SCHEMBL17007494

SCHEMBL17007494

Cc1c(C)c(S(=O)(=O)Cl)c(C)c2c1OC(C)(C)C2

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
F2 P00734 1/20 0.31
PLG P00747 1/20 0.31
PLAU P00749 1/20 0.31
ST14 Q9Y5Y6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29506779 1.00 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL12811732 0.85 HSP90AA1 (0.38) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL29402889 0.84 CYP1A2 (0.39) ALDH1A1SMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL838416 0.84 CYP1A2 (0.39) ALDH1A1SMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL2477502 0.83 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL4047614 0.83 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL29793307 0.83 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL29561615 0.83 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL4569875 0.82 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2
SCHEMBL4569895 0.82 HSP90AA1 (0.37) HSP90AA1HSP90AB1ALDH1A1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777071-A Preparation method of methyl arginine 南京药坦生物科技有限公司 2024-03-29 CN claimed
US-20260137821-A1 PEPTIDE STRUCTURE TARGETING CARBONIC DEHYDROGENASE IX AND USE THEREOF C-BIOMEX CO., LTD. (KR) 2026-05-21 US disclosed
US-20260117257-A1 MRNA Delivery System Targeting DC Cells and Preparation Method Therefor WINLEIN TIANJIN BIOTECHNOLOGY CO LTD (CN) 2026-04-30 US disclosed
EP-4608452-A2 PEPTIDE-ANTISENSE OLIGONUCLEOTIDES AND THEIR USE FOR TREATMENT OF NEURODEGENERATIVE DISORDERS Eisai R&D Management Co., Ltd. (JP) 2025-09-03 EP disclosed
US-20250136545-A1 NOVEL SULFONAMIDE DERIVATIVES HAVING SELECTIVE NOX INHIBITING ACTIVITY GLUCOX BIOTECH AB (SE) 2025-05-01 US disclosed
WO-2025023747-A1 PEPTIDE STRUCTURE TARGETING CARBONIC DEHYDROGENASE IX AND USE THEREOF (주)씨바이오멕스 2025-01-30 WO disclosed
US-12202790-B2 Sulfonamide derivatives having selective Nox inhibiting activity GLUCOX BIOTECH AB (SE) 2025-01-21 US disclosed
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2024-12-05 US disclosed
WO-2024208277-A1 CALCITONIN ANALOGUE, AND DERIVATIVE THEREOF AND USE THEREOF 杭州先为达生物科技股份有限公司 2024-10-10 WO disclosed
US-20240325307-A1 HIGH DENSITY PEPTIDE POLYMERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-10-03 US disclosed
WO-2019215291-A1 NOVEL SULFONAMIDE DERIVATIVES HAVING SELECTIVE NOX INHIBITING ACTIVITY GLUCOX BIOTECH AB (SE) 2019-11-14 WO disclosed
US-20190135776-A1 THERAPEUTICS TARGETING TRUNCATED ADENOMATOUS POLYPOSIS COLI (APC) PROTEINS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2019-05-09 US disclosed
EP-3398957-A1 METHOD FOR SYNTHESIZING ETELCALCETIDE Hybio Pharmaceutical Co., Ltd (CN) 2018-11-07 EP disclosed
US-20180042843-A1 HIGH DENSITY PEPTIDE POLYMERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2018-02-15 US disclosed
US-9856233-B2 Therapeutics targeting truncated adenomatous polyposis coli (APC) proteins BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2018-01-02 US disclosed
WO-2017100154-A1 INHIBITORS FOR PROLIFERATING CELL NUCLEAR ANTIGEN AND USES PURDUE RESEARCH FOUNDATION (US) 2017-06-15 WO disclosed
EP-3044218-A2 THERAPEUTICS TARGETING TRUNCATED ADENOMATOUS POLYPOSIS COLI (APC) PROTEINS Board Of Regents Of the University Of Texas System (US) 2016-07-20 EP disclosed
EP-2299821-B1 TRICYCLIC COMPOUNDS ABBVIE INC (US) 2015-11-04 EP disclosed
US-20150232444-A1 THERAPEUTICS TARGETING TRUNCATED ADENOMATOUS POLYPOSIS COLI (APC) PROTEINS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM 2015-08-20 US disclosed
CN-100453537-C Process for preparing amino-acid with dual protection YIFURUI INDUSTRY CO LTD (CN) 2009-01-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150232444-A1 THERAPEUTICS TARGETING TRUNCATED ADENOMATOUS POLYPOSIS COLI (APC) PROTEINS APC, VHL, TP53 HSP90AA1 907/4885HSP90AB1 719/4885ALDH1A1 4595/4885
US-12202790-B2 Sulfonamide derivatives having selective Nox inhibiting activity NOX4, NOX1, NOX5 HSP90AA1 1069/4885HSP90AB1 691/4885ALDH1A1 493/4885
US-20190135776-A1 THERAPEUTICS TARGETING TRUNCATED ADENOMATOUS POLYPOSIS COLI (APC) PROTEINS APC, VHL, TP53 HSP90AA1 907/4885HSP90AB1 719/4885ALDH1A1 4595/4885
US-20250136545-A1 NOVEL SULFONAMIDE DERIVATIVES HAVING SELECTIVE NOX INHIBITING ACTIVITY NOX4, NOX1, NOX5 HSP90AA1 1264/4885HSP90AB1 847/4885ALDH1A1 473/4885
US-20180042843-A1 HIGH DENSITY PEPTIDE POLYMERS ERMP1, PARL, PRAP1 HSP90AA1 2448/4885HSP90AB1 1336/4885ALDH1A1 4678/4885
US-20260117257-A1 MRNA Delivery System Targeting DC Cells and Preparation Method Therefor RNMT, RNGTT, CD4 HSP90AA1 1360/4885HSP90AB1 1476/4885ALDH1A1 3800/4885
US-20260137821-A1 PEPTIDE STRUCTURE TARGETING CARBONIC DEHYDROGENASE IX AND USE THEREOF CA5A, CA1, CA9 HSP90AA1 2329/4885HSP90AB1 1750/4885ALDH1A1 949/4885
US-20240325307-A1 HIGH DENSITY PEPTIDE POLYMERS IAPP, LCP1, LNPEP HSP90AA1 453/4885HSP90AB1 706/4885ALDH1A1 4773/4885
US-20240400499-A1 NOVEL AMINO ACID DERIVATIVES BCAT1, BCAT2, PELP1 HSP90AA1 906/4885HSP90AB1 1464/4885ALDH1A1 4472/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.