SCHEMBL19255760

SCHEMBL19255760

O=C(N[C@H]1COC[C@@H]2CCCN2C1=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.48
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
CASP3 P42574 1/20 0.47
TSHR P16473 1/20 0.46
EPHX1 P07099 1/20 0.46
PREP P48147 4/20 0.46
DPP4 P27487 1/20 0.45
KCNH2 Q12809 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790190 0.81 CASP3 (0.49) CASP1ALDH1A1GAACTSLCTSB
SCHEMBL19207724 0.78 PLA2G7 (0.33)
SCHEMBL12873896 0.77 CASP1 (0.44) CASP1CTSKCASP3EPHX1
SCHEMBL14320141 0.77 ALDH1A1 (0.51) CASP1ALDH1A1GAACTSLCTSB
SCHEMBL10265005 0.77 CTSK (0.49) ALDH1A1GAACTSLCTSBCTSK
SCHEMBL31039728 0.77 CTSL (0.57) ALDH1A1GAACTSLCTSBCTSK
SCHEMBL31039731 0.77 CTSL (0.57) ALDH1A1GAACTSLCTSBCTSK
SCHEMBL795453 0.75 FPR2 (0.52) CASP1CTSLCTSKCASP3
SCHEMBL795454 0.75 FPR2 (0.52) CASP1CTSLCTSKCASP3
SCHEMBL19207654 0.75 RIPK1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250388601-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2025-12-25 US disclosed
US-12358928-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2025-07-15 US disclosed
US-20240150376-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2024-05-09 US disclosed
US-20230043400-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2023-02-09 US disclosed
US-20200317691-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2020-10-08 US disclosed
US-10604535-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2020-03-31 US disclosed
US-20190112318-A1 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. 2019-04-18 US disclosed
US-10131676-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2018-11-20 US disclosed
US-20180099981-A1 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. 2018-04-12 US disclosed
US-9896458-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2018-02-20 US disclosed
US-20180022759-A1 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. 2018-01-25 US disclosed
US-9815850-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2017-11-14 US disclosed
WO-2017136727-A2 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. (US) 2017-08-10 WO disclosed
US-20170226127-A1 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. 2017-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180099981-A1 COMPOUNDS, COMPOSITIONS AND METHODS PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20250388601-A1 Compounds, Compositions and Methods AURKC, WEE2, ERBB2 CASP1 2775/4885ALDH1A1 3854/4885GAA 2997/4885
US-20200317691-A1 Compounds, Compositions and Methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20240150376-A1 Compounds, Compositions and Methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-12358928-B2 Compounds, compositions and methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-10131676-B2 Compounds, compositions and methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20230043400-A1 Compounds, Compositions and Methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20180022759-A1 COMPOUNDS, COMPOSITIONS AND METHODS PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20170226127-A1 COMPOUNDS, COMPOSITIONS AND METHODS PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-10604535-B2 Compounds, compositions and methods PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885
US-20190112318-A1 COMPOUNDS, COMPOSITIONS AND METHODS PIK3CA, PLK1, PIK3CB CASP1 2041/4885ALDH1A1 4405/4885GAA 2016/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.