SCHEMBL19542

SCHEMBL19542

COc1cccc(CO)n1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
MPO P05164 1/20 0.41
CCR1 P32246 1/20 0.40
ADORA2A P29274 2/20 0.39
BTK Q06187 1/20 0.38
LIPG Q9Y5X9 1/20 0.36
GRM5 P41594 1/20 0.36
TRPV3 Q8NET8 1/20 0.35
POLB P06746 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PSMB5 P28074 1/20 0.35
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932468 0.84 KDM1A (0.42) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL23888634 0.81 LIPG (0.44) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL217520 0.81 KDM1A (0.45) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL28031732 0.81 MPO (0.49) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL1536741 0.80 MAPK8 (0.50) CCR1BTKGRM5TRPV3
SCHEMBL14067123 0.80 KDM1A (0.49) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL20099871 0.80 KCNH2 (0.46) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL10568321 0.79 MPO (0.44) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL509881 0.79 KDM1A (0.44) KDM1AMAOAMAOBMPOADORA2A
SCHEMBL128108 0.79 KDM1A (0.44) KDM1AMAOAMAOBMPOADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 316 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118271239-B Synthesis method of 3- (6-methoxy-2-pyridine) -propionic acid 聊城大学 2025-02-11 CN claimed
CN-118271239-A Synthesis method of 3- (6-methoxy-2-pyridine) -propionic acid 聊城大学 2024-07-02 CN claimed
CN-113979955-B Preparation method of heterocyclic ester compound 河南农业大学 2024-05-14 CN claimed
CN-113979955-A Preparation method of heterocyclic ester compound 河南农业大学 2022-01-28 CN claimed
JP-2011524881-A 2011-09-08 JP claimed
EP-2307385-A1 2 -ARYLAMINOQUINAZOLINES FOR TREATING PROLIFERATIVE DISEASES Novartis AG (CH) 2011-04-13 EP claimed
US-20100121052-A1 Novel compounds for treating proliferative diseases JAIN RAMA 2010-05-13 US claimed
WO-2009153313-A1 2 -ARYLAMINOQUINAZOLINES FOR TREATING PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2009-12-23 WO claimed
WO-2026098493-A1 HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 江苏恒瑞医药股份有限公司 2026-05-15 WO disclosed
US-20260078091-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer AMGEN INC (US) 2026-03-19 US disclosed
US-20260028365-A1 TYROSINE KINASE 2 INHIBITORS AND USES THEREOF BIOGEN MA INC (US) 2026-01-29 US disclosed
US-12528815-B2 5-amino-8-(4-pyridyl)-[1,2,4]triazolo[4,3-c]pyrimidin-3-one compounds for use against cancer NXERA PHARMA UK LIMITED (GB) 2026-01-20 US disclosed
US-20250325552-A1 SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES INC (US) 2025-10-23 US disclosed
US-20250197368-A1 2-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS DRAIG THERAPEUTICS LTD. (GB) 2025-06-19 US disclosed
US-6200975-B1 FOR COGNITION ENHANCEMENT THERAPY MERCK SHARP & DOHME LIMITED (GB) 2001-03-13 US disclosed
EP-0986562-A1 SUBSTITUTED 1,2,4-TRIAZOLO 3,4-A]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LTD. (GB) 2000-03-22 EP disclosed
WO-1998050385-A1 SUBSTITUTED 1,2,4-TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES AS GABA ALPHA 5 LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1998-11-12 WO disclosed
EP-0189678-B1 ELECTROCHEMICAL REDUCTIONS OF PYRIDINE CARBOXAMIDE BASES REILLY INDUSTRIES, INC. (US) 1991-11-06 EP disclosed
US-4695352-A Electrochemical reduction of pyridine carboxamide bases REILLY TAR & CHEMICAL CORPORATION (US) 1987-09-22 US disclosed
EP-0189678-A1 Electrochemical reductions of pyridine carboxamide bases REILLY INDUSTRIES, INC. (US) 1986-08-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100121052-A1 Novel compounds for treating proliferative diseases PDK1, PDK2, PDK3 KDM1A 1003/4885MAOA 4685/4885MAOB 4407/4885
US-20250325552-A1 SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS POLQ, POLK, POLH KDM1A 3330/4885MAOA 3462/4885MAOB 3551/4885
US-20260078091-A1 Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer TP53, HIF1AN, MDM2 KDM1A 117/4885MAOA 4186/4885MAOB 4346/4885
US-20250197368-A1 2-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS GABRA2, GABRA3, GABRB2 KDM1A 1315/4885MAOA 316/4885MAOB 440/4885
US-12528815-B2 5-amino-8-(4-pyridyl)-[1,2,4]triazolo[4,3-c]pyrimidin-3-one compounds for use against cancer ADORA1, ADORA3, OPRL1 KDM1A 4408/4885MAOA 483/4885MAOB 597/4885
US-20260028365-A1 TYROSINE KINASE 2 INHIBITORS AND USES THEREOF TYK2, ERBB2, ROS1 KDM1A 812/4885MAOA 1293/4885MAOB 838/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.