SCHEMBL20118231

SCHEMBL20118231

CCC1=NN(c2ccc(F)cc2Cl)C(=O)[C@]12CC[C@H](NC(=O)c1cc(Br)cc3c1OCC3)CC2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 3/20 0.37
CRHR2 Q13324 1/20 0.37
CXCR2 P25025 1/20 0.37
PTGES O14684 3/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HPGD P15428 1/20 0.36
HTR3A P46098 2/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
DRD3 P35462 1/20 0.34
HTR4 Q13639 2/20 0.33
HTR1A P08908 1/20 0.33
ADRA2C P18825 1/20 0.33
ACHE P22303 1/20 0.33
PTGS1 P23219 1/20 0.33
ADRA1A P35348 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118187 0.77 PDE4B (0.41) CRHR1CRHR2HPGDCNR1CNR2
SCHEMBL20118213 0.77 LMNA (0.42) CRHR1CRHR2HPGDHTR1A
SCHEMBL20118174 0.76 CRHR1 (0.40) CRHR1CRHR2HPGD
SCHEMBL20118184 0.76 CRHR1 (0.39) CRHR1CRHR2HPGDKCNH2
SCHEMBL20118188 0.75 KDM4E (0.47)
SCHEMBL20118220 0.75 ALDH1A1 (0.50) CRHR1CRHR2MAPTHPGD
SCHEMBL20118407 0.74 PDE4B (0.40) CRHR1CRHR2HTR1A
SCHEMBL20118169 0.74 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118172 0.74 P2RX7 (0.35) CRHR1CRHR2
SCHEMBL20118401 0.71 PSEN1 (0.37) CRHR1CRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed