SCHEMBL2178802

SCHEMBL2178802

NCCCC(OP(=O)(O)C(O)(CCCN)P(=O)(O)O)(P(=O)([O-])[O-])P(=O)([O-])[O-].[Na+].[Na+].[Na+].[Na+]

nearest known ligand 0.63

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FDPS known ✓ P14324 17/20 0.63
PDE3A known ✓ Q14432 2/20 0.58
PDE4D known ✓ Q08499 1/20 0.43
LMNA P02545 1/20 0.43
ADRB3 P13945 1/20 0.43
GGPS1 O95749 7/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177948 0.87 FDPS (0.66) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL429804 0.81 FDPS (0.79) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL7831396 0.80 FDPS (0.76) FDPSPDE3ALMNAADRB3PDE4D
SCHEMBL6669236 0.79 FDPS (0.63) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL328770 0.78 FDPS (1.00) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL5608575 0.78 FDPS (0.73) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL4270336 0.77 FDPS (0.87) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL5080994 0.77 FDPS (0.71) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL3110183 0.76 FDPS (0.96) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL536412 0.76 FDPS (0.96) FDPSPDE3ALMNAADRB3PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091247-A1 MIXED AMINAL PHARMACEUTICAL COMPOSITIONS AND USES THEREOF INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2011-07-28 WO disclosed
US-20110166180-A1 METHOD FOR TREATMENT OF BONE DISEASES AND FRACTURES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166180-A1 METHOD FOR TREATMENT OF BONE DISEASES AND FRACTURES ACP3, PPP4C, PPP6C FDPS 426/4885PDE3A 298/4885PDE4D 305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.