SCHEMBL2184085

SCHEMBL2184085

CCc1cccc(CC)c1N1C(=O)C(Cl)=C(Cl)C1=O

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.56
CRHR2 Q13324 1/20 0.56
ANPEP P15144 2/20 0.54
DPP4 P27487 2/20 0.54
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
MGLL Q99685 1/20 0.41
GABRA1 P14867 3/20 0.40
GABRB2 P47870 3/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
DAO P14920 1/20 0.39
NPEPPS P55786 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28187917 0.91 CRHBP (0.49) CRHBPCRHR2ANPEPDPP4PKM
SCHEMBL29431569 0.89 L3MBTL1 (0.51) CRHBPCRHR2ANPEPDPP4PKM
SCHEMBL2840556 0.89 L3MBTL1 (0.51) CRHBPCRHR2ANPEPDPP4PKM
SCHEMBL10734022 0.83 DPP4 (0.58) CRHBPCRHR2ANPEPDPP4MGLL
SCHEMBL29382376 0.80 DPP4 (0.68) CRHBPCRHR2ANPEPDPP4L3MBTL1
SCHEMBL987346 0.80 DPP4 (0.68) CRHBPCRHR2ANPEPDPP4L3MBTL1
SCHEMBL22221562 0.78 ANPEP (0.66) CRHBPCRHR2ANPEPDPP4L3MBTL1
SCHEMBL8766123 0.78 KDM5A (0.49) PKML3MBTL1MGLLLMNAMAPT
SCHEMBL10483855 0.78 GABRA1 (0.41) CRHBPCRHR2ANPEPDPP4L3MBTL1
SCHEMBL8765659 0.78 PKM (0.49) CRHBPCRHR2PKMMGLLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 161 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10858521-B2 Antifouling coating compositions, antifouling coating films, antifouling substrates, methods for producing antifouling substrates, and methods of storing antifouling coating compositions CHUGOKU MARINE PAINTS, LTD. (JP) 2020-12-08 US claimed
EP-3299427-B1 ANTIFOULING COATING MATERIAL COMPOSITION, ANTIFOULING COATING FILM, ANTIFOULING BASE, METHOD FOR PRODUCING ANTIFOULING BASE, AND METHOD FOR STORING ANTIFOULING COATING MATERIAL COMPOSITION CHUGOKU MARINE PAINTS (JP) 2020-06-17 EP claimed
US-20180105703-A1 ANTIFOULING COATING COMPOSITIONS, ANTIFOULING COATING FILMS, ANTIFOULING SUBSTRATES, METHODS FOR PRODUCING ANTIFOULING SUBSTRATES, AND METHODS OF STORING ANTIFOULING COATING COMPOSITIONS CHUGOKU MARINE PAINTS, LTD. (JP) 2018-04-19 US claimed
EP-3299427-A1 ANTIFOULING COATING MATERIAL COMPOSITION, ANTIFOULING COATING FILM, ANTIFOULING BASE, METHOD FOR PRODUCING ANTIFOULING BASE, AND METHOD FOR STORING ANTIFOULING COATING MATERIAL COMPOSITION Chugoku Marine Paints, Ltd. (JP) 2018-03-28 EP claimed
EP-2551309-B1 ANTIFOULING COATING COMPOSITION AND USE FOR SAME CHUGOKU MARINE PAINTS (JP) 2017-05-17 EP claimed
US-8840910-B2 Antifouling coating composition and uses of the same CHUGOKU MARINE PAINTS, LTD. (JP) 2014-09-23 US claimed
US-20130045264-A1 ANTIFOULING COATING COMPOSITION AND USES OF THE SAME CHUGOKU MARINE PAINTS, LTD. (JP) 2013-02-21 US claimed
EP-2551309-A1 ANTIFOULING COATING COMPOSITION AND USE FOR SAME Chugoku Marine Paints, Ltd. (JP) 2013-01-30 EP claimed
US-20100209381-A1 COPPER COMPOUND-CONTAINING ANTIFOULING COATING COMPOSITION HAVING IMPROVED SLIME RESISTANCE AND STORAGE STABILITY CHUGOKU MARINE PAINTS, LTD. (JP) 2010-08-19 US claimed
EP-2206755-A1 ANTI-STAIN COATING COMPOSITION CONTAINING COPPER COMPOUND AND HAVING IMPROVED SLIME RESISTANCE AND STORAGE STABILITY CHUGOKU MARINE PAINTS, LTD. (JP) 2010-07-14 EP claimed
EP-2161318-A1 TRIPHENYLBORON COMPOUND-CONTAINING ANTIFOULING COATING COMPOSITION HAVING IMPROVED STABILITY, ANTIFOULING AGENT SET USED THEREFOR, AND METHOD FOR SUPPRESSING/CONTROLLING DECOMPOSITION OF TRIPHENYLBORON COMPOUND CHUGOKU MARINE PAINTS, LTD. (JP) 2010-03-10 EP claimed
US-12637573-B2 Antifouling coating composition CHUGOKU MARINE PAINTS, LTD. (JP) 2026-05-26 US disclosed
EP-4726003-A1 UNDERWATER ANTIFOULING COATING COMPOSITION Chugoku Marine Paints, Ltd. (JP) 2026-04-15 EP disclosed
EP-4726002-A1 UNDERWATER ANTI-FOULING COATING MATERIAL COMPOSITION Chugoku Marine Paints, Ltd. (JP) 2026-04-15 EP disclosed
EP-4691768-A1 LAMINATED ANTIFOULING COATING FILM Chugoku Marine Paints, Ltd. (JP) 2026-02-11 EP disclosed
US-5760091-A ADDING TO SEAWATER SYSTEM AN AMINE COMPOUND AND A POLYAMINE COMPOUND KATAYAMA CHEMICAL, INC. (JP) 1998-06-02 US disclosed
US-5658375-A ACRYLONITRILE COMPOUND CONTAINING THIAZOLE RING STRUCTURE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1997-08-19 US disclosed
US-5603755-A 1-(4-ALKYL- OR ARYL-THIAZOL-2-YL)-2-(ALKYL- OR ARYL-SULFONYLOXY)-2-HALOPHENYL-ACRYLONITRILE DERIVATIVES; POTENCY, STABILITY; ANTIGROWTH AGENTS IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1997-02-18 US disclosed
EP-0706758-A1 MARINE ANTIFOULING AGENT IHARA CHEMICAL INDUSTRY Co., Ltd. (JP) 1996-04-17 EP disclosed
US-5290834-A Method for controlling elution rate of agent ROHM & HAAS COMPANY (US) 1994-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12637573-B2 Antifouling coating composition COL1A1, COL2A1, HBS1L CRHBP 3926/4885CRHR2 3502/4885ANPEP 2039/4885
US-20130045264-A1 ANTIFOULING COATING COMPOSITION AND USES OF THE SAME ADRB2, OPRM1, CHRM2 CRHBP 1624/4885CRHR2 133/4885ANPEP 3306/4885
US-10858521-B2 Antifouling coating compositions, antifouling coating films, antifouling substrates, methods for producing antifouling substrates, and methods of storing antifouling coating compositions ITGA5, SIGMAR1, ITGB6 CRHBP 1948/4885CRHR2 778/4885ANPEP 3607/4885
US-20180105703-A1 ANTIFOULING COATING COMPOSITIONS, ANTIFOULING COATING FILMS, ANTIFOULING SUBSTRATES, METHODS FOR PRODUCING ANTIFOULING SUBSTRATES, AND METHODS OF STORING ANTIFOULING COATING COMPOSITIONS ITGA5, SIGMAR1, ITGB6 CRHBP 1948/4885CRHR2 778/4885ANPEP 3607/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.