SCHEMBL2270366

SCHEMBL2270366

CC(C)(C)OC(=O)c1ccc(Oc2ccccc2)cc1NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
STK39 Q9UEW8 3/20 0.47
TLR8 Q9NR97 4/20 0.44
TLR7 Q9NYK1 2/20 0.44
HDAC1 Q13547 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
SERPINE1 P05121 1/20 0.42
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK1 P28482 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275857 0.85 SERPINE1 (0.54) STK39TLR8TLR7HDAC1HDAC8
SCHEMBL2277921 0.84 ACLY (0.49) HDAC1HDAC8HDAC6KMT2AMEN1
SCHEMBL2275549 0.82 SLC16A3 (0.43) KMT2AMEN1POLBALDH1A1
SCHEMBL2275596 0.82 FABP1 (0.51) HDAC1HDAC8HDAC6KMT2AMEN1
SCHEMBL2269667 0.81 F10 (0.53) HDAC1HDAC8HDAC6SERPINE1KMT2A
SCHEMBL2276220 0.81 L3MBTL1 (0.55) TLR8KMT2AMEN1ALDH1A1NPSR1
SCHEMBL2276375 0.81 GRIK1 (0.49) HDAC1HDAC8HDAC6KMT2AMEN1
SCHEMBL2274026 0.80 PGR (0.61) KMT2AMEN1MAPK1
SCHEMBL2271662 0.80 KMT2A (0.57) KMT2AMEN1NPSR1MAPK1
SCHEMBL2269139 0.80 CYP2C9 (0.47) HDAC1HDAC8HDAC6SERPINE1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101094829-B novel anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO.,LTD. (JP) 2012-02-08 CN disclosed
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
CN-101094829-A Novel anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO LTD (JP) 2007-12-26 CN disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 STK39 1878/4885TLR8 1001/4885TLR7 394/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.