SCHEMBL264176

SCHEMBL264176

Ic1ccc2[nH]ncc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 6/20 1.00
ROCK2 O75116 5/20 0.59
MAPT P10636 3/20 0.59
ROCK1 Q13464 2/20 0.59
METAP2 P50579 2/20 0.59
KDM4E B2RXH2 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
CSNK2A1 P68400 1/20 0.59
ALDH1A1 P00352 1/20 0.59
GAA P10253 1/20 0.59
HPGD P15428 1/20 0.59
RAB9A P51151 1/20 0.59
HIF1A Q16665 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
GSK3B P49841 4/20 0.53
DYRK1A Q13627 3/20 0.53
CLK1 P49759 2/20 0.53
DYRK3 O43781 1/20 0.53
CLK2 P49760 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29402104 0.83 NOS1 (0.70) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL1141578 0.83 NOS1 (0.70) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL907620 0.74 NOS1 (0.59) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL3497213 0.74 TRPA1 (0.59) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL31315056 0.74 NOS1 (0.59) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL3995547 0.74 NOS1 (0.59) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL5562 0.74 NOS1 (1.00) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL277777 0.74 ROCK2 (0.59) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL117208 0.74 ROCK2 (1.00) NOS1ROCK2MAPTROCK1METAP2
SCHEMBL3540025 0.74 NOS1 (1.00) NOS1ROCK2MAPTROCK1METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 358 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260138998-A1 GLP-1 RECEPTOR AGONISTS AND METHODS OF USE MERCK SHARP & DOHME LLC (US) 2026-05-21 US disclosed
US-20260049071-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF BEYANG THERAPEUTICS CO LTD (CN) 2026-02-19 US disclosed
US-12545689-B2 Macrocyclic LRRK2 kinase inhibitors ONCODESIGN PRECISION MEDICINE (FR) 2026-02-10 US disclosed
US-12545648-B2 Benzopyrazole compound MEDSHINE DISCOVERY INC. (CN) 2026-02-10 US disclosed
US-20250388577-A1 METTL3 INHIBITORY COMPOUNDS STORM THERAPEUTICS LTD (GB) 2025-12-25 US disclosed
EP-4146658-B1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS ONCODESIGN PREC MEDICINE OPM (FR) 2025-10-29 EP disclosed
US-12358915-B2 METTL3 inhibitory compounds STORM Therapeutics Ltd. (GB) 2025-07-15 US disclosed
US-12344605-B2 Substituted pyrrolidine amides II GRUENENTHAL GMBH (DE) 2025-07-01 US disclosed
EP-4556466-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF Beyang Therapeutics Co., Ltd. (CN) 2025-05-21 EP disclosed
WO-2025082316-A1 OPHTHALMIC FORMATION, AND PREPARATION METHOD THEREFOR AND USE THEREOF 苏州必扬医药科技有限公司 2025-04-24 WO disclosed
US-20020161022-A1 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation AGOURON PHARMACEUTICALS 2002-10-31 US disclosed
EP-1250326-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2002-10-23 EP disclosed
US-6451819-B2 PYRROLIDINE-3-YL-SULFANYL, OR SUFONYL OR SUFINYL DERIVATIVES USED IN THE TREATMENT OF NEURODEGENERATIVE DISEASES HOFFMANN-LA ROCHE INC. 2002-09-17 US disclosed
US-20010047031-A1 Heterocyclic compounds useful as NMDA receptor selective subtype blockers HOFFMANN-LA ROCHE INC. 2001-11-29 US disclosed
WO-2001081303-A1 PYRROLIDINE AND PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREAMENT OF NEURODEGENERATIVE DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2001-11-01 WO disclosed
WO-2001053268-A2 INDAZOLE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND THEIR USE FOR MEDIATING OR INHIBITING CELL PROLIFERATION AGOURON PHARMACEUTICALS, INC. (US) 2001-07-26 WO disclosed
EP-0137223-B1 PHOTOGRAPHIC IMAGE-RECEIVING ELEMENT FOR SILVER SALT DIFFUSION TRANSFER PROCESS FUJI PHOTO FILM CO., LTD. (JP) 1988-05-11 EP disclosed
US-4585725-A STORAGE STABILITY FUJI PHOTO FILM CO., LTD. (JP) 1986-04-29 US disclosed
EP-0137223-A2 Photographic image-receiving element for silver salt diffusion transfer process FUJI PHOTO FILM CO., LTD. (JP) 1985-04-17 EP disclosed
US-3963495-A Image-receiving element for silver salt diffusion transfer with layer of monoacrylates or monomethacrylates of polyhydric alcohols FUJI PHOTO FILM CO., LTD. (JA) 1976-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12358915-B2 METTL3 inhibitory compounds METTL3, METTL16, DIMT1 NOS1 1520/4885ROCK2 2678/4885MAPT 3077/4885
US-12545689-B2 Macrocyclic LRRK2 kinase inhibitors LRRK2, SNCA, ROS1 NOS1 1180/4885ROCK2 98/4885MAPT 717/4885
US-20260138998-A1 GLP-1 RECEPTOR AGONISTS AND METHODS OF USE GLP1R, GIPR, GPR119 NOS1 3486/4885ROCK2 1806/4885MAPT 4844/4885
US-12344605-B2 Substituted pyrrolidine amides II NR3C1, NR3C2, MC2R NOS1 1524/4885ROCK2 3294/4885MAPT 4458/4885
US-20020161022-A1 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation CDK3, MKI67, ROCK1 NOS1 131/4885ROCK2 12/4885MAPT 902/4885
US-20250388577-A1 METTL3 INHIBITORY COMPOUNDS METTL3, RNMT, TPMT NOS1 550/4885ROCK2 3543/4885MAPT 4317/4885
US-12545648-B2 Benzopyrazole compound CYP3A43, CYP4B1, ABCB11 NOS1 3463/4885ROCK2 1827/4885MAPT 3452/4885
US-20010047031-A1 Heterocyclic compounds useful as NMDA receptor selective subtype blockers GRIN1, GRM1, GRIN2B NOS1 1959/4885ROCK2 3731/4885MAPT 1856/4885
US-20260049071-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF KDR, FLT1, ERBB2 NOS1 444/4885ROCK2 351/4885MAPT 4181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.