SCHEMBL288413

SCHEMBL288413

O=C(O)n1ccc2ncccc21

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.56
MET P08581 9/20 0.54
RPS6KA5 O75582 5/20 0.50
PARP1 P09874 1/20 0.41
RPS6KA4 O75676 1/20 0.41
CDC7 O00311 1/20 0.41
CDK2 P24941 1/20 0.41
RAPGEF4 Q8WZA2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30241905 1.00 SLC22A12 (0.56) SLC22A12METRPS6KA5PARP1RPS6KA4
SCHEMBL30532842 0.98 SLC22A12 (0.55) SLC22A12METRPS6KA5PARP1RPS6KA4
SCHEMBL14312991 0.87 PARP1 (0.56) SLC22A12METRPS6KA5PARP1RPS6KA4
SCHEMBL31200457 0.84 SLC22A12 (0.55) SLC22A12METRPS6KA5PARP1RPS6KA4
SCHEMBL4714519 0.83 SLC22A12 (0.66) SLC22A12METRPS6KA5SMN1; SMN2
SCHEMBL759396 0.76 SLC22A12 (0.48) SLC22A12METRPS6KA5RAPGEF4
SCHEMBL29962730 0.76 SLC22A12 (0.48) SLC22A12METRPS6KA5RAPGEF4
SCHEMBL857765 0.73 SMN1; SMN2 (0.61) SMN1; SMN2
SCHEMBL5803359 0.73 SLC22A12 (0.45) SLC22A12METRPS6KA5RPS6KA4CDC7
SCHEMBL29898292 0.73 SLC22A12 (1.00) SLC22A12METRPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025235719-A1 DIMERIC SMAC MIMETICS USEFUL IN HIV THERAPY VIIV HEALTHCARE COMPANY (US) 2025-11-13 WO disclosed
US-12275729-B2 Substituted tetrahydroquinolin compounds as indoleamine 2,3-dioxygenase (IDO) inhibitors MERCK SHARP & DOHME LLC (US) 2025-04-15 US disclosed
US-20240124493-A1 Monocyclic And Bicyclic Ring System Substituted Carbanucleoside Analogues For Use As PRMT5 Inhibitors JANSSEN PHARMACEUTICA NV (BE) 2024-04-18 US disclosed
WO-2023230541-A1 PIPERAZINE DERIVATIVES USEFUL IN HIV THERAPY VIIV HEALTHCARE COMPANY (US) 2023-11-30 WO disclosed
CN-116731016-A Tricyclic heterocyclic compounds as IAP antagonists 苏州亚盛药业有限公司 2023-09-12 CN disclosed
US-20230234967-A1 Fused Azole Heterocycles as AHR Antagonists SAIL BIOMEDICINES, INC. 2023-07-27 US disclosed
CN-109803971-B Monocyclic and bicyclic substituted carbanucleoside analogs as PRMT5 inhibitors 詹森药业有限公司 2022-10-28 CN disclosed
US-11339177-B2 Heteroaryl compounds as inhibitors of necrosis, composition and method using the same ACCRO BIOSCIENCE (HK) LIMITED (HK) 2022-05-24 US disclosed
US-11274100-B2 EP300/CREBBP inhibitor DAIICHI SANKYO COMPANY, LIMITED (JP) 2022-03-15 US disclosed
EP-3728252-A1 4-AZAINDOLE COMPOUNDS Bristol-Myers Squibb Company (US) 2020-10-28 EP disclosed
CN-104011050-A 2, 4-diamino-pyrimidine derivatives as serine/threonine kinase inhibitors HOFFMANN LA ROCHE 2014-08-27 CN disclosed
EP-2427448-A1 Gpr 119 modulators Pfizer Inc. (US) 2012-03-14 EP disclosed
EP-2427450-A1 GPR 119 MODULATORS Pfizer Inc. (US) 2012-03-14 EP disclosed
US-20120052130-A1 GPR 119 MODULATORS PFIZER INC. 2012-03-01 US disclosed
EP-2342202-A1 AZAINDOLE DERIVATIVE Merck Patent GmbH (DE) 2011-07-13 EP disclosed
WO-2010128414-A1 GPR 119 MODULATORS PFIZER INC. (US) 2010-11-11 WO disclosed
WO-2010128425-A1 GPR 119 MODULATORS PFIZER INC. (US) 2010-11-11 WO disclosed
US-20100285145-A1 GPR 119 MODULATORS PFIZER INC 2010-11-11 US disclosed
WO-2010046013-A1 AZAINDOLE DERIVATIVE MERCK PATENT GMBH (DE) 2010-04-29 WO disclosed
CN-1244798-A Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds RHONE POULENC RORER PHARMA (US) 2000-02-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11274100-B2 EP300/CREBBP inhibitor EP300, CREBBP, CREB1 SLC22A12 3271/4885MET 2938/4885RPS6KA5 543/4885
US-20120052130-A1 GPR 119 MODULATORS GPR119, GPR39, GPR65 SLC22A12 618/4885MET 555/4885RPS6KA5 1934/4885
US-20230234967-A1 Fused Azole Heterocycles as AHR Antagonists AHR, ARNT, AIPL1 SLC22A12 3925/4885MET 491/4885RPS6KA5 2590/4885
US-11339177-B2 Heteroaryl compounds as inhibitors of necrosis, composition and method using the same BAX, LITAF, PNLIP SLC22A12 3370/4885MET 3056/4885RPS6KA5 764/4885
US-20100285145-A1 GPR 119 MODULATORS GPR119, GPR65, GPR39 SLC22A12 1054/4885MET 924/4885RPS6KA5 1884/4885
US-12275729-B2 Substituted tetrahydroquinolin compounds as indoleamine 2,3-dioxygenase (IDO) inhibitors IDO1, IDO2, INMT SLC22A12 1804/4885MET 4158/4885RPS6KA5 2307/4885
US-20240124493-A1 Monocyclic And Bicyclic Ring System Substituted Carbanucleoside Analogues For Use As PRMT5 Inhibitors PRMT5, PRMT1, PRMT8 SLC22A12 3896/4885MET 2519/4885RPS6KA5 199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.