SCHEMBL29449939

SCHEMBL29449939

COC1C(=O)N2C(C(=O)[O-])=C(CSc3nnnn3CCO)COC12.[Na+]

nearest known ligand 0.43

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 1/20 0.37
HSD17B10 Q99714 5/20 0.43
TDP1 Q9NUW8 4/20 0.43
ELANE P08246 5/20 0.42
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.37
POLB P06746 1/20 0.37
APEX1 P27695 1/20 0.37
PTPN7 P35236 1/20 0.37
BLM P54132 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.37
CMA1 P23946 6/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29727496 0.92 ELANE (0.44) HSD17B10TDP1ELANEALDH1A1KDM4E
SCHEMBL29501762 0.91 ELANE (0.43) HSD17B10TDP1ELANEALDH1A1KDM4E
SCHEMBL29501744 0.82 CMA1 (0.55) ELANEPTGS1CMA1
SCHEMBL11497346 0.78 ELANE (0.40) HSD17B10TDP1ELANEMAPTALDH1A1
Flomoxef SCHEMBL30531854 0.73 HSD17B10 (0.58) HSD17B10TDP1MAPTBLMSMN1; SMN2
Flomoxef SCHEMBL30716855 0.73 HSD17B10 (0.58) HSD17B10TDP1MAPTBLMSMN1; SMN2
Flomoxef SCHEMBL30515667 0.69 PTGS1 (0.44) HSD17B10TDP1PTGS1CMA1
Flomoxef SCHEMBL14423926 0.66 PTGS1 (0.57) HSD17B10TDP1PTGS1CMA1
Flomoxef SCHEMBL49438 0.66 PTGS1 (0.57) HSD17B10TDP1PTGS1CMA1
SCHEMBL11046775 0.66 TDP1 (0.54) HSD17B10TDP1MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114315858-A Synthesis method of flomoxef intermediate 深圳市立国药物研究有限公司 2022-04-12 CN disclosed