Evans Blue Free Acid

Evans Blue Free Acid

SCHEMBL29601874

Cc1cc(-c2ccc(/N=N/c3ccc4c(S(=O)(=O)[O-])cc(S(=O)(=O)[O-])c(N)c4c3O)c(C)c2)ccc1/N=N/c1ccc2c(S(=O)(=O)[O-])cc(S(=O)(=O)[O-])c(N)c2c1O.[Na+].[Na+].[Na+].[Na+]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Evans Blue Free Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB known ✓ P10828 6/20 0.77
ENPP2 Q13822 3/20 1.00
HSPD1 P10809 2/20 1.00
HSPE1 P61604 2/20 1.00
TST Q16762 2/20 1.00
PTPN1 P18031 2/20 1.00
ALB P02768 1/20 1.00
CYP3A4 P08684 5/20 0.77
MAPK1 P28482 5/20 0.77
RECQL P46063 5/20 0.77
HSD17B10 Q99714 5/20 0.77
HPGD P15428 4/20 0.77
MEN1 O00255 4/20 0.77
KMT2A Q03164 4/20 0.77
KDM4E B2RXH2 3/20 0.77
TDP1 Q9NUW8 3/20 0.77
CYP2C9 P11712 2/20 0.77
CYP2C19 P33261 2/20 0.77
APEX1 P27695 2/20 0.77
USP2 O75604 2/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Evans Blue Free Acid SCHEMBL103701 1.00 ENPP2 (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Evans Blue Free Acid SCHEMBL29377040 1.00 ENPP2 (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Evans Blue Free Acid SCHEMBL30392230 1.00 ENPP2 (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Evans Blue Free Acid SCHEMBL29381789 1.00 ENPP2 (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Evans Blue Free Acid SCHEMBL2437648 1.00 ENPP2 (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Evans Blue Free Acid SCHEMBL29609615 0.87 MEN1 (0.98) ENPP2HSPD1HSPE1TSTPTPN1
Chicago Sky Blue SCHEMBL93506 0.87 THRB (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Chicago Sky Blue SCHEMBL29358365 0.87 THRB (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Chicago Sky Blue SCHEMBL29401288 0.87 THRB (1.00) ENPP2HSPD1HSPE1TSTPTPN1
Chicago Sky Blue SCHEMBL30201536 0.87 THRB (1.00) ENPP2HSPD1HSPE1TSTPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116982597-A Clear light intervention system for preventing and treating acute lung injury caused by acute hypoxia 中国人民解放军陆军军医大学 2023-11-03 CN claimed
EP-4499145-A1 TRANSIENT DISRUPTION OF THE NEUROVASCULAR BARRIER OF A HUMAN AND USES THEREOF FOR TREATING AMYOTROPHIC LATERAL SCLEROSIS SORBONNE UNIVERSITE (FR) 2025-02-05 EP disclosed
CN-118924758-A Use of BTK inhibitors and single dose medicaments 武汉人福创新药物研发中心有限公司 2024-11-12 CN disclosed
CN-118924759-A Composition containing BTK inhibitor and application thereof 武汉人福创新药物研发中心有限公司 2024-11-12 CN disclosed
CN-117100857-B Antibody gold nano-cage medicine carrying system, preparation method and application 福建医科大学附属协和医院 2024-09-10 CN disclosed
CN-118490800-B Pharmaceutical composition for clearing heat and relieving itching as well as preparation and application thereof 云南中医药大学 2024-09-06 CN disclosed
CN-118490800-A Pharmaceutical composition for clearing heat and relieving itching as well as preparation and application thereof 云南中医药大学 2024-08-16 CN disclosed
EP-4387565-A1 COMBINATORIAL THERAPIES INCLUDING IMPLANTABLE DAMPING DEVICES AND THERAPEUTIC AGENTS FOR TREATING A CONDITION AND ASSOCIATED SYSTEMS AND METHODS OF USE The Brain Protection Company Pty Ltd (AU) 2024-06-26 EP disclosed
CN-117309534-A Fungus fluorescent staining solution and preparation method and application thereof 深圳玖明医疗科技有限公司 2023-12-29 CN disclosed
CN-112391358-B Vibrio mediterranean virulent phage vB_VmeM-Yong and application thereof 宁波大学 2023-12-01 CN disclosed
CN-117100857-A Antibody gold nano-cage medicine carrying system, preparation method and application 福建医科大学附属协和医院 2023-11-24 CN disclosed
WO-2023179866-A1 TRANSIENT DISRUPTION OF THE NEUROVASCULAR BARRIER OF A HUMAN AND USES THEREOF FOR TREATING AMYOTROPHIC LATERAL SCLEROSIS SORBONNE UNIVERSITE (FR) 2023-09-28 WO disclosed
CN-115838393-B Intermediate for FAPI synthesis and preparation method and application thereof 烟台蓝纳成生物技术有限公司 2023-05-05 CN disclosed
WO-2023019320-A1 COMBINATORIAL THERAPIES INCLUDING IMPLANTABLE DAMPING DEVICES AND THERAPEUTIC AGENTS FOR TREATING A CONDITION AND ASSOCIATED SYSTEMS AND METHODS OF USE CARNEGIE VENTURE CAPITAL PTY LTD (AU) 2023-02-23 WO disclosed
WO-2022144927-A1 A METHOD OF PREPARATION OF PURE PHARMACEUTICAL COMPOUNDS AND PHARMACEUTICAL FORMULATION THEREOF KAR, SANTOSH KUMAR (IN) 2022-07-07 WO disclosed
EP-3996502-A1 COMPOSITIONS AND METHODS FOR PRESERVING ORGAN TRANSPLANTS Firststring Research, Inc. (US) 2022-05-18 EP disclosed