Trolamine

Trolamine

SCHEMBL3283288

O=P(O)(O)OP(=O)(O)O.O=[N+]([O-])O.O=[N+]([O-])O.O=[N+]([O-])O.OCCN(CCO)CCO

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ERG11

The experimentally established mechanism targets of Trolamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
FDPS P14324 1/20 0.40
BLM P54132 1/20 0.40
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
CA5A P35218 1/20 0.32
CA5B Q9Y2D0 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trolamine SCHEMBL2390784 0.98 FDPS (0.39) TDP1FDPSBLMALDH1A1KDM4E
Trolamine SCHEMBL3283293 0.87 CA5A (0.38) TDP1ALDH1A1KDM4ECA5ACA5B
Trolamine SCHEMBL2869748 0.87 FDPS (0.53) TDP1FDPSBLMKDM4ESMN1; SMN2
Trolamine SCHEMBL2396169 0.82 CA5A (0.47) TDP1ALDH1A1KDM4ECA5ACA5B
Trolamine SCHEMBL725388 0.82 CA5A (0.47) TDP1ALDH1A1KDM4ECA5ACA5B
Trolamine SCHEMBL9299420 0.80 CA5A (0.44) TDP1ALDH1A1KDM4ECA5ACA5B
Trolamine SCHEMBL28050292 0.80 CA5A (0.44) TDP1ALDH1A1KDM4ECA5ACA5B
Triphosphate SCHEMBL7796776 0.79 FDPS (0.41) TDP1FDPSBLMKDM4ESMN1; SMN2
Trolamine SCHEMBL9300209 0.78 CA5A (0.42) TDP1ALDH1A1KDM4ECA5ACA5B
Pyrophosphoric Acid SCHEMBL8931250 0.78 FDPS (0.59) TDP1FDPSBLMCA5ACA5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805730-A1 Nitric oxide donor for the treatment of chronic fatigue syndrome Bergen Teknologioverforing AS (NO) 2014-11-26 EP claimed
US-20080317679-A1 FOAMABLE COMPOSITIONS AND KITS COMPRISING ONE OR MORE OF A CHANNEL AGENT, A CHOLINERGIC AGENT, A NITRIC OXIDE DONOR, AND RELATED AGENTS AND THEIR USES FOAMIX LTD. (IL) 2008-12-25 US claimed
JP-2008540509-A 2008-11-20 JP claimed
WO-2008110872-A2 FOAMABLE COMPOSITIONS AND KITS COMPRISING ONE OR MORE OF A CHANNEL AGENT, A CHOLINERGIC AGENT, A NITRIC OXIDE DONOR, AND RELATED AGENTS AND THEIR USES FOAMIX LTD. (US) 2008-09-18 WO claimed
EP-1919448-A2 VASOACTIVE KIT AND COMPOSITION AND USES THEREOF Foamix Ltd. (IL) 2008-05-14 EP claimed
WO-2007023396-A2 VASOACTIVE KIT AND COMPOSITION AND USES THEREOF FOAMIX LTD. (US) 2007-03-01 WO claimed
US-20050271596-A1 Vasoactive kit and composition and uses thereof FOAMIX LTD. 2005-12-08 US claimed
EP-4277592-A1 TOPICAL COMPOSITION Liliger Ltd (IL) 2023-11-22 EP disclosed
US-20230355500-A1 TOPICAL COMPOSITION LILIGER LTD (IL) 2023-11-09 US disclosed
CN-116685302-A Topical compositions 利勒格有限公司 2023-09-01 CN disclosed
US-11433025-B2 Oil foamable carriers and formulations VYNE THERAPEUTICS INC. (US) 2022-09-06 US disclosed
WO-2022153308-A1 TOPICAL COMPOSITION RICH PSC LTD. (IL) 2022-07-21 WO disclosed
US-20210386944-A1 GAS-EVOLVING COMPOSITIONS AND CONTAINER AND DELIVERY SYSTEMS SANOTIZE RESEARCH DEVELOPMENT CORP. (CA) 2021-12-16 US disclosed
US-4834979-A Medical bandage for administering beneficial drug ALZA CORPORATION (US) 1989-05-30 US disclosed
US-4812313-A Method for lessening the incidence of anginal attacks ALZA CORPORATION (US) 1989-03-14 US disclosed
US-4725272-A Novel bandage for administering beneficial drug ALZA CORPORATION (US) 1988-02-16 US disclosed
US-4704119-A Method comprising transdermal and buccal treatment of angina ALZA CORPORATION (US) 1987-11-03 US disclosed
US-4661105-A Medical bandage for administering vasodilator drug ALZA CORPORATION (US) 1987-04-28 US disclosed
US-4650484-A Method for treating ischemic conditions ALZA CORPORATION (US) 1987-03-17 US disclosed
US-4486193-A Method for treating ischemic conditions by administering drug by two routes ALZA CORPORATION (US) 1984-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11433025-B2 Oil foamable carriers and formulations LIPA, PTGER1, TTPA TDP1 3437/4885FDPS 446/4885BLM 543/4885
US-20210386944-A1 GAS-EVOLVING COMPOSITIONS AND CONTAINER AND DELIVERY SYSTEMS GMPS, SQOR, GSS TDP1 2909/4885FDPS 875/4885BLM 2109/4885
US-20230355500-A1 TOPICAL COMPOSITION NOS1, NOS3, NOS2 TDP1 446/4885FDPS 1984/4885BLM 3770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.