SCHEMBL3373434

SCHEMBL3373434

CC(C)[C@](C)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CTSK P43235 9/20 0.41
CTSS P25774 8/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CA12 O43570 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CYP2D6 P10635 1/20 0.38
APLNR P35414 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.35
DGAT1 O75907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3528810 1.00 CA1 (0.42) CA1CA2CA7CTSKCTSS
SCHEMBL3528813 1.00 CA1 (0.42) CA1CA2CA7CTSKCTSS
SCHEMBL19578354 0.85 CA12 (0.33) CA1CA2CA7CTSKCTSS
SCHEMBL12175227 0.85 CA12 (0.33) CA1CA2CA7CTSKCTSS
SCHEMBL22577436 0.84 CA1 (0.40) CA1CA2CA7CTSKCTSS
SCHEMBL22362794 0.84 APLNR (0.41) CA1CA2CA7CTSKCTSS
SCHEMBL19209627 0.83 CTSK (0.44) CA1CA2CA7CTSKCTSS
SCHEMBL28000287 0.83 CTSK (0.44) CA1CA2CA7CTSKCTSS
SCHEMBL19209615 0.83 CTSK (0.44) CA1CA2CA7CTSKCTSS
SCHEMBL18709073 0.82 DGAT1 (0.47) CA1CA2CA7CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12612420-B2 Arginase inhibitors and methods of use thereof MOLECURE S.A. (PL) 2026-04-28 US disclosed
EP-4678238-A2 ARGINASE INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2026-01-14 EP disclosed
US-12503452-B2 Antimicrobial compounds and methods CURZA GLOBAL, LLC (US) 2025-12-23 US disclosed
US-20250313578-A1 Arginase Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2025-10-09 US disclosed
EP-3752251-B1 ARGINASE INHIBITORS AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2025-09-10 EP disclosed
US-12195485-B2 Arginase inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2025-01-14 US disclosed
US-11912727-B2 Arginase inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2024-02-27 US disclosed
CN-117186134-A Arginase inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2023-12-08 CN disclosed
US-20230365599-A1 Arginase Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2023-11-16 US disclosed
EP-4267590-A1 ARGINASE INHIBITORS AND METHODS OF USE THEREOF ONCOARENDI THERAPEUTICS S.A. (PL) 2023-11-01 EP disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-20090186869-A1 Antiviral compounds GILEAD SCIENCES, INC. (US) 2009-07-23 US disclosed
US-20090186869-A1 Antiviral compounds GILEAD SCIENCES, INC. (US) 2009-07-23 US disclosed
US-20090186869-A1 Antiviral compounds GILEAD SCIENCES, INC. (US) 2009-07-23 US disclosed
WO-2009005677-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2009-01-08 WO disclosed
EP-1877391-A1 PRO-DRUGS OF N-THIAZOL-2YL-BENZAMIDE DERIVATIVES H. Lundbeck A/S (DK) 2008-01-16 EP disclosed
WO-2006114093-A1 PRO-DRUGS OF N-THIAZOL-2YL-BENZAMIDE DERIVATIVES H. LUNDBECK A/S (DK) 2006-11-02 WO disclosed
US-20060229336-A1 Ccr5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORPORATION 2006-10-12 US disclosed
EP-1569646-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2005-09-07 EP disclosed
WO-2004054974-A2 PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2004-07-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11912727-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 CA1 413/4885CA2 544/4885CA7 683/4885
US-12195485-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, PRMT1 CA1 456/4885CA2 556/4885CA7 739/4885
US-20230365599-A1 Arginase Inhibitors and Methods of Use Thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 CA1 413/4885CA2 544/4885CA7 683/4885
US-20250313578-A1 Arginase Inhibitors and Methods of Use Thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 CA1 413/4885CA2 544/4885CA7 683/4885
US-20090186869-A1 Antiviral compounds MAVS, EIF2AK2, ZC3HAV1 CA1 4745/4885CA2 4564/4885CA7 3839/4885
US-12612420-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, ARGLU1 CA1 600/4885CA2 204/4885CA7 2113/4885
US-20060229336-A1 Ccr5 antagonists as therapeutic agents CCR5, CCR1, CXCR3 CA1 4808/4885CA2 4267/4885CA7 4713/4885
US-12503452-B2 Antimicrobial compounds and methods MPO, NISCH, RPN2 CA1 4525/4885CA2 2151/4885CA7 1619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.