SCHEMBL367333

SCHEMBL367333

O=C(O)c1c2ccccc2n2cc(C(=O)N3CCOCC3)ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.52
TSHR P16473 1/20 0.49
CNR2 P34972 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
ALDH1A1 P00352 4/20 0.46
CNR1 P21554 1/20 0.46
PHGDH O43175 1/20 0.45
KDM4E B2RXH2 2/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
CYP1A2 P05177 1/20 0.44
LMNA P02545 1/20 0.42
GRM5 P41594 1/20 0.42
POLB P06746 1/20 0.42
DNMT1 P26358 1/20 0.42
PTPN7 P35236 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365229 0.89 HPGD (0.48) HPGDTSHRCNR2SMN1; SMN2ALDH1A1
SCHEMBL365335 0.86 CNR2 (0.47) HPGDCNR2ALDH1A1CNR1KDM4E
SCHEMBL367332 0.81 HPGD (0.50) HPGDTSHRCNR2SMN1; SMN2GAA
SCHEMBL365668 0.80 KMT2A (0.55) HPGDTSHRSMN1; SMN2ALDH1A1KDM4E
SCHEMBL365935 0.80 KDM4E (0.47) HPGDALDH1A1KDM4ECYP1A2POLB
SCHEMBL366310 0.77 ALDH1A1 (0.52) HPGDSMN1; SMN2ALDH1A1CNR1KDM4E
SCHEMBL366876 0.76 EGFR (0.44) HPGDSMN1; SMN2ALDH1A1KDM4EPOLB
SCHEMBL366811 0.76 EGFR (0.44) HPGDTSHRALDH1A1KDM4EPOLB
SCHEMBL367205 0.73 EGFR (0.45) HPGDALDH1A1KDM4EHDAC1HDAC6
SCHEMBL365912 0.73 CES1 (0.45) HPGDALDH1A1KDM4ECYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed