SCHEMBL4035688

SCHEMBL4035688

CN(C)CCC1CN(c2ccc(Cl)c(Cl)c2)CCN1S(=O)(=O)c1ccc(-c2ccccc2)cc1.NC(=O)NC=O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.39
CA2 P00918 3/20 0.39
MMP9 P14780 2/20 0.39
MMP2 P08253 1/20 0.39
OPRK1 P41145 4/20 0.38
PTGDR Q13258 1/20 0.37
THRB P10828 1/20 0.37
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038524 0.77 MMP2 (0.34) CA12MMP9MMP2CA9
SCHEMBL4035190 0.72 ADAMTS4 (0.42) MMP9
SCHEMBL4033743 0.71 RAB9A (0.45) CA12CA2MMP9CA1CA9
SCHEMBL4035748 0.69 MMP1 (0.40) MMP9MMP2
SCHEMBL4032668 0.66 THRB (0.36) CA12CA2PTGDRTHRBCA1
SCHEMBL4037368 0.66 CCR1 (0.39) OPRK1
SCHEMBL4035430 0.65 MMP1 (0.47) MMP9
SCHEMBL1470570 0.63 NOTUM (0.42) PTGDRTHRB
SCHEMBL1662635 0.62 HDAC3 (0.49) MMP9MMP2
SCHEMBL5800067 0.61 PTGDR (0.53) PTGDRTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed