SCHEMBL4037038

SCHEMBL4037038

CCCCS(=O)(=O)N1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2CC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.39
CXCR3 P49682 1/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
KMT2A Q03164 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 2/20 0.36
PKM P14618 2/20 0.36
GAA P10253 1/20 0.36
CCR5 P51681 2/20 0.36
CYP2D6 P10635 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SLC6A9 P48067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041414 0.88 KMT2A (0.46) SMN1; SMN2KMT2AHTTMAPTPKM
SCHEMBL3917728 0.83 SMN1; SMN2 (0.39) SMN1; SMN2NPC1CYP1A2CYP2C9UBE2M
SCHEMBL4034055 0.83 L3MBTL1 (0.45) KMT2AHTTMAPTPKMGAA
SCHEMBL3927380 0.83 CYP2D6 (0.45) SMN1; SMN2KMT2AHTTMAPTGAA
SCHEMBL2934783 0.83 CCR5 (0.40) SMN1; SMN2CXCR3KMT2AGAACCR5
SCHEMBL4041277 0.83 KMT2A (0.41) SMN1; SMN2CXCR3KMT2AHTTMAPT
SCHEMBL4041475 0.82 MMP2 (0.39) SMN1; SMN2CXCR3KMT2AHTTMAPT
SCHEMBL4038204 0.80 EPHX2 (0.47) KMT2ACCR5CYP2D6
SCHEMBL4035567 0.79 LMNA (0.48) CYP1A2KMT2AHTTMAPTPKM
SCHEMBL4032408 0.79 ALDH1A1 (0.52) SMN1; SMN2KMT2AHTTMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed