SCHEMBL4045912

SCHEMBL4045912

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1)Oc1cccc2ccccc12

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 8/20 0.34
ITGB7 P26010 7/20 0.34
POLB P06746 1/20 0.33
F12 P00748 1/20 0.33
CTSK P43235 2/20 0.33
CAPN1 P07384 1/20 0.32
ITGB1 P05556 2/20 0.32
F10 P00742 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
ACE P12821 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044157 0.90 CNR1 (0.38) ITGA4ITGB7POLBCTSKITGB1
SCHEMBL4045610 0.90 POLB (0.33) POLBF12CTSKCAPN1F10
SCHEMBL4041433 0.88 ALDH1A1 (0.35) ITGA4ITGB7POLBF12ITGB1
SCHEMBL4046036 0.88 P2RX7 (0.36) ITGA4ITGB7CTSKITGB1ACE
SCHEMBL4044768 0.85 CTSL (0.44) CTSKCTSLCTSBCTSS
SCHEMBL4041901 0.83 P2RX7 (0.39) ITGA4ITGB7CTSKITGB1P2RX7
SCHEMBL4044603 0.82 MC4R (0.37) ITGA4ITGB7POLBCTSKCTSL
SCHEMBL4045047 0.82 CTSL (0.37) ITGA4ITGB7POLBF12CTSK
SCHEMBL4043833 0.82 F10 (0.36) ITGA4ITGB7CTSKITGB1F10
SCHEMBL4041712 0.82 ITGA4 (0.40) ITGA4ITGB7CTSKITGB1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed