2-Pyrrolidone

2-Pyrrolidone

SCHEMBL421593

C=Cc1n(C=C)cc[n+]1C.COS(=O)(=O)[O-].O=C1CCCN1

nearest known ligand 0.33

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of 2-Pyrrolidone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
OR51E2 Q9H255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Pyrrolidone SCHEMBL423278 0.90 OR51E2 (0.41) OR51E2
2-Pyrrolidone SCHEMBL5916159 0.90 OR51E2 (0.41) OR51E2
2-Pyrrolidone SCHEMBL867929 0.73 OR51E2 (0.34) OR51E2
SCHEMBL538961 0.70 NPSR1 (0.33)
SCHEMBL11272078 0.70 HDAC8 (0.35)
SCHEMBL28599017 0.67 LMNA (0.32)
SCHEMBL28604119 0.65 HTT (0.31)
Sulfuric Acid Dimethyl Ester SCHEMBL11365586 0.63 OR51E2 (0.62) OR51E2
2-Pyrrolidone SCHEMBL9518900 0.63 OR51E2 (0.62) OR51E2
Sulfuric Acid Dimethyl Ester SCHEMBL10761403 0.61 OR51E2 (0.42) OR51E2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9211425-B2 Product for keratin-containing fibers comprising at least one specific amphiphilic cationic polymer, and at least one specific amphiphilic anionic polymer HENKEL AG & CO. KGAA (DE) 2015-12-15 US disclosed
US-9044411-B2 Agent for keratinous fibers, comprising at least one acrylate/glyceryl acrylate copolymer, at least one film-forming and/or solidifying polymer and at least one ester oil HENKEL AG & CO. KGAA (DE) 2015-06-02 US disclosed
US-9034307-B2 Agent for fibers containing keratin, containing at least one specific amphiphilic cationic polymer and at least one additional film-forming cationic and/or stabilizing polymer HENKEL AG & CO. KGAA (DE) 2015-05-19 US disclosed
US-20140305462-A1 Powdery Hair Cosmetics HENKEL AG & CO. KGAA (DE) 2014-10-16 US disclosed
US-8741273-B2 Agents for fibers containing keratin, containing at least one special cross-linked amphiphilic, anionic polymer and at least one further special non-cross-linked amphiphilic anionic polymer HENKEL AG & CO. KGAA (DE) 2014-06-03 US disclosed
US-8663605-B2 Agent for fibers containing keratin, comprising at least one specific amphiphilic cationic polymer, at least one cationic styling polymer that is different therefrom and at least one film-forming non-ionic and/or stabilizing non-ionic polymer HENKEL AG & CO. KGAA (DE) 2014-03-04 US disclosed
US-20140050686-A1 AGENT FOR KERATINOUS FIBERS, COMPRISING AT LEAST ONE ACRYLATE/GLYCERYL ACRYLATE COPOLYMER, AT LEAST ONE FILM-FORMING AND/OR SOLIDIFYING POLYMER AND AT LEAST ONE ESTER OIL HENKEL AG & CO. KGAA (DE) 2014-02-20 US disclosed
US-20130295034-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER HENKEL AG & CO. KGAA (DE) 2013-11-07 US disclosed
US-8506941-B2 Agent for fibers containing keratin, containing at least one specific amphiphilic cationic polymer and at least one additional film-forming cationic and/or stabilizing polymer HENKEL AG&CO. KGAA (DE) 2013-08-13 US disclosed
US-20120204896-A1 POLYAMIDES OF FATTY ACID DIMERS AND DIAMINES FOR FIXING A HAIRSTYLE SCHWEINSBERG MATTHIAS (DE) 2012-08-16 US disclosed
US-20120199155-A1 METHOD OF CREATING HAIRSTYLES THAT CAN BE REMODELED SCHWEINSBERG MATTHIAS (DE) 2012-08-09 US disclosed
US-20120141406-A1 AGENT FOR KERATINOUS FIBERS, COMPRISING AT LEAST ONE ACRYLATE/GLYCERYL ACRYLATE COPOLYMER, AT LEAST ONE FILM-FORMING AND/OR SOLIDIFYING POLYMER AND AT LEAST ONE ESTER OIL HENKEL AG & CO. KGAA (DE) 2012-06-07 US disclosed
US-20120064023-A1 AGENTS FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIAL CROSS-LINKED AMPHIPHILIC, ANIONIC POLYMER AND AT LEAST ONE FURTHER SPECIAL NON-CROSS-LINKED AMPHIPHILIC ANIONIC POLYMER HENKEL AG & CO. KGAA (DE) 2012-03-15 US disclosed
US-20120021028-A1 Powdery Composition for Shaping Keratin Fibers and Giving Them Shine HENKEL AG & CO. KGAA (DE) 2012-01-26 US disclosed
US-20110165109-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING AND/OR STABILIZING POLYMER SELECTED FROM CHITOSAN AND DERIVATES THEREOF MUELLER BURKHARD 2011-07-07 US disclosed
US-20110142780-A1 AGENT FOR KERATIN-CONTAINING FIBERS, COMPRISING AT LEAST ONE PARTICULAR AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE POLYMER WITH SILICON-CONTAINING SIDECHAINS AND ANIONIC GROUPS HENTRICH DIRK 2011-06-16 US disclosed
US-20110135589-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER, AND AT LEAST ONE SPECIFIC AMPHIPHILIC ANIONIC POLYMER HENKEL AG & CO. KGAA (DE) 2011-06-09 US disclosed
US-20110135590-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC, CATIONIC POLYMER, AND AT LEAST ONE POLYOL KNAPPE THORSTEN 2011-06-09 US disclosed
US-20110135591-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER HENKEL AG & CO. KGAA (DE) 2011-06-09 US disclosed
US-20110132389-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER, AT LEAST ONE CATIONIC STYLING POLYMER THAT IS DIFFERENT THEREFROM AND AT LEAST ONE FILM-FORMING NON-IONIC AND/OR STABILIZING NON-IONIC POLYMER HENKEL AG & CO. KGAA (DE) 2011-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (14 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110135590-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC, CATIONIC POLYMER, AND AT LEAST ONE POLYOL KRT18, F12, H1-10 OR51E2 561/4885
US-20120064023-A1 AGENTS FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIAL CROSS-LINKED AMPHIPHILIC, ANIONIC POLYMER AND AT LEAST ONE FURTHER SPECIAL NON-CROSS-LINKED AMPHIPHILIC ANIONIC POLYMER KRT18, DSG1, CUTA OR51E2 3036/4885
US-20110135591-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER KRT18, POLR1C, F12 OR51E2 44/4885
US-20140050686-A1 AGENT FOR KERATINOUS FIBERS, COMPRISING AT LEAST ONE ACRYLATE/GLYCERYL ACRYLATE COPOLYMER, AT LEAST ONE FILM-FORMING AND/OR SOLIDIFYING POLYMER AND AT LEAST ONE ESTER OIL KRT18, ACR, CUTA OR51E2 1484/4885
US-20110135589-A1 PRODUCT FOR KERATIN-CONTAINING FIBERS COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER, AND AT LEAST ONE SPECIFIC AMPHIPHILIC ANIONIC POLYMER KRT18, H1-10, F12 OR51E2 896/4885
US-20110132389-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER, AT LEAST ONE CATIONIC STYLING POLYMER THAT IS DIFFERENT THEREFROM AND AT LEAST ONE FILM-FORMING NON-IONIC AND/OR STABILIZING NON-IONIC POLYMER KRT18, POLR1C, ZYX OR51E2 35/4885
US-20120204896-A1 POLYAMIDES OF FATTY ACID DIMERS AND DIAMINES FOR FIXING A HAIRSTYLE FFAR2, DGAT2, FAAH2 OR51E2 3065/4885
US-20140305462-A1 Powdery Hair Cosmetics CUTA, SHH, H1-0 OR51E2 3835/4885
US-20120021028-A1 Powdery Composition for Shaping Keratin Fibers and Giving Them Shine KRT18, CUTA, KIF23 OR51E2 1757/4885
US-20130295034-A1 AGENT FOR FIBERS CONTAINING KERATIN, CONTAINING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING CATIONIC AND/OR STABILIZING POLYMER KRT18, POLR1C, F12 OR51E2 44/4885
US-20120141406-A1 AGENT FOR KERATINOUS FIBERS, COMPRISING AT LEAST ONE ACRYLATE/GLYCERYL ACRYLATE COPOLYMER, AT LEAST ONE FILM-FORMING AND/OR SOLIDIFYING POLYMER AND AT LEAST ONE ESTER OIL KRT18, ACR, CUTA OR51E2 1484/4885
US-20110142780-A1 AGENT FOR KERATIN-CONTAINING FIBERS, COMPRISING AT LEAST ONE PARTICULAR AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE POLYMER WITH SILICON-CONTAINING SIDECHAINS AND ANIONIC GROUPS KRT18, DSG1, H1-10 OR51E2 876/4885
US-20110165109-A1 AGENT FOR FIBERS CONTAINING KERATIN, COMPRISING AT LEAST ONE SPECIFIC AMPHIPHILIC CATIONIC POLYMER AND AT LEAST ONE ADDITIONAL FILM-FORMING AND/OR STABILIZING POLYMER SELECTED FROM CHITOSAN AND DERIVATES THEREOF KRT18, F12, POLR1C OR51E2 29/4885
US-20120199155-A1 METHOD OF CREATING HAIRSTYLES THAT CAN BE REMODELED FASN, ACSL5, DGAT2 OR51E2 3770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.