SCHEMBL432970

SCHEMBL432970

NC(=O)c1ccc(C2(C(=O)NCC(c3ccccc3)N3CCCC3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
CYP2C19 P33261 1/20 0.44
TP53 P04637 5/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
LMNA P02545 4/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
P2RX7 Q99572 2/20 0.41
MAPT P10636 1/20 0.41
TRPA1 O75762 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL433923 0.89 HSD11B1 (0.49) CYP1A2CYP2C9HPGDMAPK1CYP2C19
SCHEMBL433444 0.89 SLC6A4 (0.47) CYP1A2CYP2C9HPGDMAPK1CYP2C19
SCHEMBL433860 0.87 P2RX7 (0.55) CYP2C9CYP2C19TP53LMNAP2RX7
SCHEMBL433922 0.85 SMN1; SMN2 (0.53) CYP1A2CYP2C9HPGDMAPK1CYP2C19
Hydrochloric Acid SCHEMBL433170 0.84 SMN1; SMN2 (0.52) CYP1A2CYP2C9HPGDMAPK1CYP2C19
SCHEMBL435915 0.84 P2RX7 (0.60) TP53LMNAMEN1ALDH1A1KMT2A
SCHEMBL435467 0.83 ALDH1A1 (0.44) CYP1A2CYP2C9HPGDMAPK1CYP2C19
SCHEMBL434779 0.82 POLB (0.52) MAPK1TP53LMNAALDH1A1KMT2A
SCHEMBL434790 0.81 OPRM1 (0.47) MEN1ALDH1A1GLAGAAKMT2A
SCHEMBL434036 0.79 TP53 (0.54) MAPK1TP53LMNAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed