SCHEMBL4437598

SCHEMBL4437598

C(=C/c1ccccc1)\CN1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
LMNA P02545 4/20 0.58
CYP2D6 P10635 4/20 0.58
MAPK1 P28482 4/20 0.58
CYP3A4 P08684 3/20 0.58
HIF1A Q16665 3/20 0.58
CYP1A2 P05177 3/20 0.58
CYP2C9 P11712 3/20 0.58
CHRM2 P08172 2/20 0.58
CHRM4 P08173 2/20 0.58
HTR1A P08908 2/20 0.58
CHRM5 P08912 2/20 0.58
ADRA2A P08913 2/20 0.58
ADORA3 P0DMS8 2/20 0.58
CHRM1 P11229 2/20 0.58
DRD2 P14416 2/20 0.58
ADRA2B P18089 2/20 0.58
ADRA2C P18825 2/20 0.58
CHRM3 P20309 2/20 0.58
DRD1 P21728 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666143 1.00 ALDH1A1 (0.58) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL2579539 0.87 LMNA (0.72) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL11036914 0.83 LTA4H (0.77) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL613704 0.83 LTA4H (0.77) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL6293359 0.83 ALDH1A1 (0.48) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL9779468 0.83 SIGMAR1 (0.71) ALDH1A1SIGMAR1MEN1KMT2AHSP90AA1
SCHEMBL15759224 0.83 ALDH1A1 (0.51) ALDH1A1HIF1ATSHRKDM4ELTA4H
SCHEMBL17888675 0.83 ALDH1A1 (0.48) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL17888676 0.83 ALDH1A1 (0.48) ALDH1A1LMNACYP2D6MAPK1CYP3A4
SCHEMBL6293360 0.83 ALDH1A1 (0.48) ALDH1A1LMNACYP2D6MAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170362151-A1 COMPOSITIONS AND METHODS FOR REDUCTION OF KETONES, ALDEHYDES AND IMINIUMS, AND PRODUCTS PRODUCED THEREBY BOARD OF TRUSTEES OF NORTHERN ILLINOIS UNIVERSITY (US) 2017-12-21 US disclosed
US-20170349561-A1 SYNTHESIS OF NOVEL IONIC LIQUIDS FROM LIGNIN-DERIVED COMPOUNDS UNITED STATES DEPARTMENT OF ENERGY 2017-12-07 US disclosed
US-9765044-B2 Synthesis of novel ionic liquids from lignin-derived compounds THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-09-19 US disclosed
US-20160031843-A1 SYNTHESIS OF NOVEL IONIC LIQUIDS FROM LIGNIN-DERIVED COMPOUNDS UNITED STATES DEPARTMENT OF ENERGY 2016-02-04 US disclosed
US-8580990-B2 Gold catalyzed hydroamination of alkynes and allenes THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-11-12 US disclosed
US-20110166349-A1 GOLD CATALYZED HYDROAMINATION OF ALKYNES AND ALLENES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-07-07 US disclosed
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP disclosed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO disclosed
US-6359174-B1 REACTING ALLYL REACTANT WITH ACID CHLORIDE IN PRESENCE OF LEWIS ACID CATALYST THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2002-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160031843-A1 SYNTHESIS OF NOVEL IONIC LIQUIDS FROM LIGNIN-DERIVED COMPOUNDS DCXR, LCT, LARS1 ALDH1A1 185/4885LMNA 128/4885CYP2D6 4475/4885
US-20170362151-A1 COMPOSITIONS AND METHODS FOR REDUCTION OF KETONES, ALDEHYDES AND IMINIUMS, AND PRODUCTS PRODUCED THEREBY ADH1A, ADH1C, ADH5 ALDH1A1 11/4885LMNA 321/4885CYP2D6 1065/4885
US-20110166349-A1 GOLD CATALYZED HYDROAMINATION OF ALKYNES AND ALLENES AOC3, AOC2, AOC1 ALDH1A1 202/4885LMNA 2925/4885CYP2D6 1661/4885
US-20170349561-A1 SYNTHESIS OF NOVEL IONIC LIQUIDS FROM LIGNIN-DERIVED COMPOUNDS LSS, DCXR, MYB ALDH1A1 2369/4885LMNA 101/4885CYP2D6 3257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.