SCHEMBL4492513

SCHEMBL4492513

CCc1c(C(=O)O)c(C=O)n(Cc2ccccc2)c1-c1cc2ccccc2o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
KDM4E B2RXH2 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TSHR P16473 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
ALOX12 P18054 1/20 0.42
POLB P06746 2/20 0.39
MKNK1 Q9BUB5 3/20 0.38
CCR2 P41597 1/20 0.37
GRIN2B Q13224 1/20 0.36
S1PR1 P21453 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
HTR1A P08908 1/20 0.36
HTR2B P41595 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4485204 0.82 ALDH1A1 (0.42) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL4494579 0.80 ALDH1A1 (0.43) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL4488093 0.76 VDR (0.40) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL4504869 0.76 ALDH1A1 (0.42) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL4559832 0.75 TP53 (0.46) ALDH1A1MEN1KMT2ATSHRHPGD
SCHEMBL4490747 0.75 PGR (0.43) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL4492331 0.75 LMNA (0.42) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL4485664 0.75 KDM4E (0.40) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL4490040 0.73 GFER (0.47) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL4482567 0.73 PLA2G2A (0.43) ALDH1A1KDM4EKMT2AHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed