SCHEMBL478289

SCHEMBL478289

CC(C)(C)OC(=O)CC(NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.57
SYK P43405 1/20 0.57
CTSK P43235 5/20 0.54
CTSL P07711 2/20 0.53
CTSB P07858 2/20 0.53
CTSS P25774 2/20 0.53
PPARG P37231 3/20 0.52
CASP1 P29466 3/20 0.52
ITGB3 P05106 2/20 0.52
ITGA2B P08514 2/20 0.52
KLK7 P49862 1/20 0.52
KLK5 Q9Y337 1/20 0.52
ACE P12821 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2775895 1.00 PPARA (0.57) PPARASYKCTSKCTSLCTSB
SCHEMBL1143898 1.00 PPARA (0.57) PPARASYKCTSKCTSLCTSB
Water SCHEMBL29401166 0.99 PPARA (0.56) PPARASYKCTSKCTSLCTSB
Water SCHEMBL2580712 0.99 PPARA (0.56) PPARASYKCTSKCTSLCTSB
SCHEMBL14037216 0.95 CTSK (0.53) PPARASYKCTSKCTSLCTSB
SCHEMBL29398102 0.92 SYK (0.57) PPARASYKCTSKCTSLCTSB
SCHEMBL31326039 0.92 CTSL (0.57) CTSKCTSLCTSBCTSSITGB3
SCHEMBL19694832 0.91 KYNU (0.56) PPARASYKCTSKCTSLCTSB
SCHEMBL14680593 0.91 SYK (0.56) PPARASYKCTSKCTSLCTSB
SCHEMBL4256075 0.91 KYNU (0.56) PPARASYKCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260035357-A1 THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION GILEAD SCIENCE INC (US) 2026-02-05 US disclosed
US-12404262-B2 Therapeutic compounds for HIV virus infection GILEAD SCIENCES, INC. (US) 2025-09-02 US disclosed
WO-2024105205-A1 ANTIBODY-DRUG CONJUGATES (A2DCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
US-20240043379-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2024-02-08 US disclosed
US-20230390411-A1 CONJUGATE AND USE THEREOF NANJING CHEMPION BIOTECHNOLOGY CO., LTD. (CN) 2023-12-07 US disclosed
EP-4285937-A1 CONJUGATE AND USE THEREOF Nanjing Chempion Biotechnology Co., Ltd. (CN) 2023-12-06 EP disclosed
US-20230212148-A1 THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION GILEAD SCIENCES, INC. 2023-07-06 US disclosed
US-11685714-B2 Prodrugs of cytotoxic active agents having enzymatically cleavable groups BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-06-27 US disclosed
WO-2023102523-A1 THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION GILEAD SCIENCES, INC. (US) 2023-06-08 WO disclosed
CN-116059390-A Prodrugs of cytotoxic actives with enzymatically cleavable groups 拜耳制药股份公司 2023-05-05 CN disclosed
CN-1525978-A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases 伊邓药品公司 2004-09-01 CN disclosed
EP-1392280-A2 ARYLSULFONAMIDE ETHERS, AND METHODS OF USE THEREOF Abbott GmbH & Co. KG (DE) 2004-03-03 EP disclosed
EP-1351975-A2 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2003-10-15 EP disclosed
CN-1420881-A Beta-amino acid derivs. as inhibitors of matrix metalloproteases and TNF-alpha BRISTOL MYERS SQUIBB PHARMACEU (US) 2003-05-28 CN disclosed
US-20030096826-A1 Arylsulfonamide ethers, and methods of use thereof WARNER-LAMBERT COMPANY 2003-05-22 US disclosed
WO-2002089749-A2 ARYLSULFONAMIDE ETHERS, AND METHODS OF USE THEREOF ABBOTT GMBH & CO.KG (DE) 2002-11-14 WO disclosed
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed
WO-2002057298-A2 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2002-07-25 WO disclosed
WO-2002034751-A1 HEXAHYDRO-4-OXOAZEPINO[3,2,1-HI]INDOLES NOVARTIS AG (CH) 2002-05-02 WO disclosed
US-20020042376-A1 C-terminal modified oxamyl dipeptides as inhibitors of the ICE-ced-3 family of cysteine proteases CONATUS PHARMACEUTICALS, INC. 2002-04-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230390411-A1 CONJUGATE AND USE THEREOF CD44, ADCY7, ADCY4 PPARA 4675/4885SYK 27/4885CTSK 3784/4885
US-11685714-B2 Prodrugs of cytotoxic active agents having enzymatically cleavable groups BUB1B, KIF5B, TK1 PPARA 4432/4885SYK 4038/4885CTSK 378/4885
US-20030096826-A1 Arylsulfonamide ethers, and methods of use thereof CASP1, IRAK1, STS PPARA 1874/4885SYK 1265/4885CTSK 172/4885
US-20240043379-A1 PRODRUGS OF CYTOTOXIC ACTIVE AGENTS HAVING ENZYMATICALLY CLEAVABLE GROUPS BUB1B, KIF5B, TK1 PPARA 4432/4885SYK 4038/4885CTSK 378/4885
US-12404262-B2 Therapeutic compounds for HIV virus infection HAVCR2, MAVS, CD4 PPARA 2074/4885SYK 3490/4885CTSK 498/4885
US-20230212148-A1 THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION CPSF6, NFATC1, CPSF1 PPARA 2904/4885SYK 4524/4885CTSK 1382/4885
US-20020042376-A1 C-terminal modified oxamyl dipeptides as inhibitors of the ICE-ced-3 family of cysteine proteases CASP3, IAPP, DPP3 PPARA 4674/4885SYK 3174/4885CTSK 762/4885
US-20260035357-A1 THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION CCR10, CCR1, CCR3 PPARA 3141/4885SYK 3536/4885CTSK 2915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.