SCHEMBL5039623

SCHEMBL5039623

O=C(Cl)CCCO[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
TP53 P04637 1/20 0.39
CA12 O43570 4/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA4 P22748 4/20 0.37
CA9 Q16790 4/20 0.37
ESR2 Q92731 3/20 0.37
TSHR P16473 2/20 0.37
PTGS2 P35354 2/20 0.35
MEN1 O00255 1/20 0.30
CYP2C9 P11712 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
HSD17B10 Q99714 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL400376 0.94 ALDH1A1 (0.40) ALDH1A1TP53CA12CA1CA2
SCHEMBL6029546 0.92 ALDH1A1 (0.34) ALDH1A1TP53CA12CA1CA2
SCHEMBL401034 0.92 ALDH1A1 (0.43) ALDH1A1TP53CA12CA1CA2
SCHEMBL22958440 0.82 DGKA (0.41) ALDH1A1CA12CA1CA2CA4
SCHEMBL14696961 0.82 ALDH1A1 (0.42) ALDH1A1TP53TSHR
SCHEMBL396155 0.81 CA12 (0.41) ALDH1A1CA12CA1CA2CA4
SCHEMBL457635 0.80 LMNA (0.44) ALDH1A1CA12CA1CA2CA4
SCHEMBL2014045 0.80 CA12 (0.41) ALDH1A1CA12CA1CA2CA4
Silver SCHEMBL2239077 0.78 CA1 (0.38) ALDH1A1CA12CA1CA2CA4
Methane SCHEMBL2013629 0.78 LMNA (0.43) ALDH1A1CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10450260-B2 NO- and H2S-releasing compounds RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2019-10-22 US disclosed
US-10450260-B2 NO- and H2S-releasing compounds RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2019-10-22 US disclosed
US-20170260124-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK 2017-09-14 US disclosed
US-20170260124-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK 2017-09-14 US disclosed
US-9688607-B2 No- and H2S-releasing compounds RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2017-06-27 US disclosed
US-9688607-B2 No- and H2S-releasing compounds RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2017-06-27 US disclosed
EP-2744487-B1 NO- AND H2S- RELEASING COMPOUNDS UNIV CITY NEW YORK RES FOUND (US) 2016-10-05 EP disclosed
US-20140221316-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2014-08-07 US disclosed
US-20140221316-A1 NO- AND H2S- RELEASING COMPOUNDS RESEARCH FOUNDATION OF THE CITY UNIVERSITY OF NEW YORK (US) 2014-08-07 US disclosed
EP-2744487-A2 NO- AND H2S- RELEASING COMPOUNDS Research Foundation Of The City University Of New York (US) 2014-06-25 EP disclosed
EP-1727787-A2 NEW PROCESS FOR THE PREPARATION OF NITROOXYDERIVATIVES OF PARACETAMOL NicOx S.A. (FR) 2006-12-06 EP disclosed
US-20060167003-A1 Probucol derivatives NICOX S.A. (FR) 2006-07-27 US disclosed
WO-2005054175-A2 NEW PROCESS FOR THE PREPARATION OF NITROOXYDERIVATIVES OF PARACETAMOL NICOX S.A. (FR) 2005-06-16 WO disclosed
EP-1521740-A2 PROBUCOL DERIVATIVES Nicox S.A. (FR) 2005-04-13 EP disclosed
US-6673819-B2 NITRIC OXIDE RELEASING COMPOUND ASTRAZENECA AB (SE) 2004-01-06 US disclosed
WO-2003080568-A2 PROBUCOL DERIVATIVES NICOX S.A. (FR) 2003-10-02 WO disclosed
US-20020111370-A1 Compounds useful as antibacterial agents ASTRAZENECA AB (SE) 2002-08-15 US disclosed
EP-0192829-B1 AMINO PROPANOL DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICINES CONTAINING THESE COMPOUNDS AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1990-09-26 EP disclosed
US-4801596-A Nitroxy amino propanols for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1989-01-31 US disclosed
EP-0192829-A1 Amino propanol derivatives, process for their preparation, medicines containing these compounds and intermediates Roche Diagnostics GmbH (DE) 1986-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221316-A1 NO- AND H2S- RELEASING COMPOUNDS PTGS1, NOS2, NOS1 ALDH1A1 363/4885TP53 1179/4885CA12 3042/4885
US-20170260124-A1 NO- AND H2S- RELEASING COMPOUNDS NOS2, NOS3, NOS1 ALDH1A1 961/4885TP53 302/4885CA12 2261/4885
US-20060167003-A1 Probucol derivatives PNLIP, APOB, LIPC ALDH1A1 511/4885TP53 2075/4885CA12 4215/4885
US-10450260-B2 NO- and H2S-releasing compounds NOS2, NOS3, NOS1 ALDH1A1 961/4885TP53 302/4885CA12 2261/4885
US-20020111370-A1 Compounds useful as antibacterial agents NOS1, NOS2, PTGS1 ALDH1A1 1397/4885TP53 4652/4885CA12 3795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.