SCHEMBL5366533

SCHEMBL5366533

CCOP(=O)(OCC)C(Nc1cccnc1)P(=O)(OCC)OCC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.59
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
CFTR P13569 1/20 0.43
GOPC Q9HD26 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 2/20 0.42
TRPV1 Q8NER1 1/20 0.42
ALPL P05186 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7793582 0.81 KDM4E (0.43) FDPSPOLBMAPTLMNANPSR1
SCHEMBL8159782 0.81 FDPS (0.60) FDPSPOLBNPC1RAB9ACFTR
SCHEMBL4743968 0.78 NPSR1 (0.64) FDPSPOLBTSHRNPC1RAB9A
SCHEMBL5367565 0.77 KMT2A (0.50) FDPSPOLBTSHRPKMALDH1A1
SCHEMBL7793634 0.75 FDFT1 (0.42) POLBMAPTLMNA
SCHEMBL7793613 0.75 L3MBTL1 (0.45) POLBMAPTALDH1A1LMNA
SCHEMBL21501951 0.75 FDPS (0.39) FDPSPOLBSMN1; SMN2ALDH1A1LMNA
SCHEMBL8166203 0.75 FDPS (0.69) FDPSPOLBNPC1RAB9ACFTR
SCHEMBL5359859 0.75 TSHR (0.42) FDPSPOLBTSHRNPC1RAB9A
SCHEMBL8159300 0.74 FDPS (1.00) FDPSCFTRGOPCLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7208481-B2 Aminodiphosphonate apolipoprotein E modulators ILEX PRODUCTS, INC. (US) 2007-04-24 US claimed
US-20050075317-A1 Aminodiphosphonate apolipoprotein e modulators PHAN HIEU TRUNG (CH) 2005-04-07 US claimed
EP-1482897-A2 AMINODIPHOSPHONATE APOLIPOPROTEIN E MODULATORS Ilex Products, Inc. (US) 2004-12-08 EP claimed
WO-2003070169-A2 AMINODIPHOSPHONATE APOLIPOPROTEIN E MODULATORS ILEX PRODUCTS, INC. (US) 2003-08-28 WO claimed
US-7208481-B2 Aminodiphosphonate apolipoprotein E modulators ILEX PRODUCTS, INC. (US) 2007-04-24 US disclosed
US-20050075317-A1 Aminodiphosphonate apolipoprotein e modulators PHAN HIEU TRUNG (CH) 2005-04-07 US disclosed
EP-1482897-A2 AMINODIPHOSPHONATE APOLIPOPROTEIN E MODULATORS Ilex Products, Inc. (US) 2004-12-08 EP disclosed
WO-2003070169-A2 AMINODIPHOSPHONATE APOLIPOPROTEIN E MODULATORS ILEX PRODUCTS, INC. (US) 2003-08-28 WO disclosed
EP-0563107-B1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 2000-05-03 EP disclosed
US-5393748-A Treating bone disorders, Paget* s disease, calcium metabolism disorders LEIRAS OY (FI) 1995-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050075317-A1 Aminodiphosphonate apolipoprotein e modulators APOB, APOL1, NAPEPLD FDPS 526/4885POLB 2745/4885TSHR 4299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.