SCHEMBL599583

SCHEMBL599583

CS(=O)(=O)c1ccc(C(=O)Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.54
AKR1C3 P42330 4/20 0.50
GSR P00390 2/20 0.50
MAOB P27338 1/20 0.50
PTGS2 P35354 2/20 0.49
AKR1C2 P52895 1/20 0.47
AKR1C1 Q04828 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17981319 0.94 PTGS2 (0.54) ENPP2AKR1C3GSRMAOBPTGS2
SCHEMBL724893 0.81 ALDH1A1 (0.50)
SCHEMBL4321082 0.81 ENPP2 (0.58) ENPP2AKR1C3GSRPTGS2
SCHEMBL28079560 0.79 ENPP2 (0.47) ENPP2AKR1C3GSRMAOBPTGS2
SCHEMBL35155 0.79 ALDH1A1 (0.48) MAOB
SCHEMBL28229 0.79 PTGS2 (0.57) ENPP2AKR1C3GSRPTGS2
SCHEMBL8747696 0.79 LMNA (0.52)
SCHEMBL34837 0.79 CA2 (0.61) ENPP2AKR1C3GSRPTGS2
SCHEMBL10451127 0.78 PSIP1 (0.50)
SCHEMBL9659082 0.77 LMNA (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 229 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1506355-A Diphenyl benzimidazole compound containing sulfonyl group and its prepn process, medicinal composition and use 中国医学科学院药物研究所 2004-06-23 CN claimed
CN-122010767-A Haloalkyl bisamide compound and application thereof 山东熙霖生物科技有限公司 2026-05-12 CN disclosed
US-20250145598-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF UNIV CALIFORNIA (US) 2025-05-08 US disclosed
CN-115626894-B Lappaconitine derivative with analgesic activity, and preparation method and application thereof 西南交通大学 2025-04-18 CN disclosed
CN-119409623-A Ketoxime ester photoinitiator and application thereof, and photosensitive composition 武汉尚赛光电科技有限公司 2025-02-11 CN disclosed
CN-111936471-B Non-fused thiophene derivatives and uses thereof 埃尼奥制药公司 2024-10-29 CN disclosed
US-20240342185-A1 SMALL MOLECULES INHIBITORS OF CYCLIC GMP-AMP SYNTHASE (cGAS) SHANGPHARMA INNOVATION INC. 2024-10-17 US disclosed
EP-4387617-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF The Regents of the University of California (US) 2024-06-26 EP disclosed
CN-112708644-B Preparation method of florfenicol intermediate 弈柯莱生物科技(集团)股份有限公司 2024-05-28 CN disclosed
CN-118026883-A Amide compound and preparation method and application thereof 南通泰禾化工股份有限公司 2024-05-14 CN disclosed
WO-1995017485-A1 FUEL COMPOSITIONS CONTAINING POLYALKYL AND POLY(OXYALKYLENE) AROMATIC ESTERS CHEVRON CHEMICAL COMPANY (US) 1995-06-29 WO disclosed
EP-0596326-A1 Arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes, their salts, medicaments containing the same, use thereof and precesses for their production Dr. Karl Thomae GmbH (DE) 1994-05-11 EP disclosed
US-4609610-A BY BETA-ELIMINATION EASTMAN KODAK COMPANY (US) 1986-09-02 US disclosed
US-4425282-A Preparation of 3-(arylvinyl)-2,2-dimethyl-cyclopropane-1-carboxylic acid esters and new intermediate therefor BAYER AKTIENGESELLSCHAFT (DE) 1984-01-10 US disclosed
EP-0018533-B1 SUBSTITUTED PENTANE (OR PENTENE) CARBOXYLIC ACIDS AND THEIR DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE FOR THE PREPARATION OF 3-(ARYLVINYL)-2,2-DIMETHYL-CYCLOPROPANE-1-CARBOXYLATES BAYER AG (DE) 1983-01-26 EP disclosed
US-4329456-A ACYLATION WITHOUT INTERMEDIATE ISOLATION CIBA-GEIGY AG (CH) 1982-05-11 US disclosed
US-4269848-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETICS LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1981-05-26 US disclosed
EP-0018533-A1 Substituted pentane (or pentene) carboxylic acids and their derivatives, process for their preparation and their use for the preparation of 3-(arylvinyl)-2,2-dimethyl-cyclopropane-1-carboxylates BAYER AG (DE) 1980-11-12 EP disclosed
US-4224341-A ANTIINFLAMMATORY AGENTS, ANALGESICS AND ANTIPYRETICS LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1980-09-23 US disclosed
US-4057642-A ANTIINFLAMMATORY, RHEUMATOID ARTHRITIS MERCK & CO., INC. (US) 1977-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145598-A1 ACID CERAMIDASE INHIBITORS AND USES THEREOF ASAH2, ASAH1, ACER2 ENPP2 18/4885AKR1C3 1418/4885GSR 3736/4885
US-20240342185-A1 SMALL MOLECULES INHIBITORS OF CYCLIC GMP-AMP SYNTHASE (cGAS) CGAS, GMPS, PRKG1 ENPP2 454/4885AKR1C3 2584/4885GSR 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.