(R)-Trolox

(R)-Trolox

SCHEMBL615168

Cc1c(C)c2c(c(C)c1O)CC[C@](C)(C(=O)O)O2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 1.00
PTGS2 P35354 1/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
TSHR P16473 1/20 1.00
PSEN1 P49768 4/20 0.56
ALOX5 P09917 3/20 0.49
NR1I2 O75469 1/20 0.49
BCHE P06276 5/20 0.47
ACHE P22303 5/20 0.47
CAPN1 P07384 1/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
GSTP1 P09211 1/20 0.45
TTPA P49638 1/20 0.45
KMT2A Q03164 1/20 0.45
USP2 O75604 1/20 0.45
THRB P10828 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trolox SCHEMBL1927837 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL3226 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL29375939 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL29653919 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL4647438 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL1651402 1.00 PTGS1 (1.00) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL7895023 0.96 PTGS1 (0.91) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL17713594 0.94 PTGS1 (0.89) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL8523345 0.93 PTGS1 (0.86) PTGS1PTGS2CYP1A2CYP3A4TSHR
Trolox SCHEMBL20746198 0.92 PTGS1 (0.84) PTGS1PTGS2CYP1A2CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 209 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509434-B2 Optically resolved Trolox intermediate and method for producing same PTC THERAPEUTICS, INC. (US) 2025-12-30 US claimed
EP-4661890-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS Purdue Research Foundation (US) 2025-12-17 EP claimed
CN-115066420-B Optically resolved Trolox intermediates and methods of making the same PTC医疗公司 2024-12-10 CN claimed
WO-2024167565-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS PURDUE RESEARCH FOUNDATION (US) 2024-08-15 WO claimed
US-20230029044-A1 OPTICALLY RESOLVED TROLOX INTERMEDIATE AND METHOD FOR PRODUCING SAME PTC THERAPEUTICS, INC. 2023-01-26 US claimed
EP-4108658-A1 OPTICALLY RESOLVED TROLOX INTERMEDIATE AND METHOD FOR PRODUCING SAME Sumitomo Pharma Co., Ltd. (JP) 2022-12-28 EP claimed
CN-115066420-A Optically resolved Trolox intermediates and process for producing the same 住友制药株式会社 2022-09-16 CN claimed
US-10072043-B2 Inhibitors of protein tyrosine phosphatases INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2018-09-11 US claimed
US-20180170892-A1 COMPOUND FOR THE PROPHYLAXIS OR TREATMENT OF ORGAN DAGAMAGE SULFATEQ B.V. (NL) 2018-06-21 US claimed
EP-3297625-A1 COMPOUND FOR THE PROPHYLAXIS OR TREATMENT OF ORGAN DAMAGE Sulfateq B.V. (NL) 2018-03-28 EP claimed
EP-1504002-B1 METHOD FOR THE PRODUCTION OF OPTICALLY ACTIVE BETA-AMINOKETONES AND OPTICALLY ACTIVE 1,3-AMINOALCOHOLS SANOFI AVENTIS DEUTSCHLAND (DE) 2012-12-19 EP claimed
US-20120088720-A1 INHIBITORS OF PROTEIN TYROSINE PHOSPHATASES INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATI (US) 2012-04-12 US claimed
WO-2010118241-A2 INHIBITORS OF PROTEIN TYROSINE PHOSPHATASES INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION (US) 2010-10-14 WO claimed
US-7161008-B2 Optically active β-aminoketones, optically active 1,3-amino alcohols and processes for preparing them Sanofi - Aventis Deutschland GmbH (DE) 2007-01-09 US claimed
EP-1504002-A1 OPTICALLY ACTIVE &bgr;-AMINOKETONES, OPTICALLY ACTIVE 1,3-AMINOALCOHOLS AND METHOD FOR THE PRODUCTION THEREOF Aventis Pharma Deutschland GmbH (DE) 2005-02-09 EP claimed
US-20040030145-A1 Optically active B-aminoketones, optically active 1,3-amino alcohols and processes for preparing them AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-02-12 US claimed
WO-2003093259-A1 OPTICALLY ACTIVE β-AMINOKETONES, OPTICALLY ACTIVE 1,3-AMINOALCOHOLS AND METHOD FOR THE PRODUCTION THEREOF AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-11-13 WO claimed
US-20030064972-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis MPM ASSET MANAGEMENT INVESTORS 2002 BVIII LLC 2003-04-03 US claimed
EP-1276730-A2 THIAZOLIDINEDIONE ANALOGUES AND THEIR USE FOR THE TREATMENT OF DIABETES ARYx Therapeutics (US) 2003-01-22 EP claimed
WO-2001081328-A2 THIAZOLIDINEDIONE ANALOGUES AND THEIR USE FOR THE TREATMENT OF DIABETES ARYX THERAPEUTICS (US) 2001-11-01 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509434-B2 Optically resolved Trolox intermediate and method for producing same CYP11B2, ACAD9, TXNRD2 PTGS1 2003/4885PTGS2 1078/4885CYP1A2 395/4885
US-10072043-B2 Inhibitors of protein tyrosine phosphatases PTPRCAP, PTPRF, PTPRS PTGS1 3346/4885PTGS2 3853/4885CYP1A2 4223/4885
US-20040030145-A1 Optically active B-aminoketones, optically active 1,3-amino alcohols and processes for preparing them ORMDL3, OR10J3, BCAT2 PTGS1 3472/4885PTGS2 3604/4885CYP1A2 429/4885
US-20030064972-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis LIPA, LIPC, CETP PTGS1 1370/4885PTGS2 814/4885CYP1A2 254/4885
US-20230029044-A1 OPTICALLY RESOLVED TROLOX INTERMEDIATE AND METHOD FOR PRODUCING SAME ALDH1A2, TTPA, AOX1 PTGS1 583/4885PTGS2 217/4885CYP1A2 74/4885
US-20120088720-A1 INHIBITORS OF PROTEIN TYROSINE PHOSPHATASES PTPRCAP, PTPRF, PTPRS PTGS1 3346/4885PTGS2 3853/4885CYP1A2 4223/4885
US-20180170892-A1 COMPOUND FOR THE PROPHYLAXIS OR TREATMENT OF ORGAN DAGAMAGE LIPG, GLS, TXN2 PTGS1 75/4885PTGS2 109/4885CYP1A2 1406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.