SCHEMBL6922115

SCHEMBL6922115

CC[N+](C)(C)Oc1c(-c2ccccc2)n(C(=O)c2ccccc2)c2ccc(Br)cc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.44
AGTR1 P30556 2/20 0.44
PTGS2 P35354 2/20 0.43
ABCB1 P08183 1/20 0.38
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
HIF1A Q16665 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PLA2G2A P14555 1/20 0.35
MAPK8 P45983 1/20 0.35
P2RX4 Q99571 1/20 0.34
TSPO P30536 1/20 0.34
SRC P12931 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7128402 0.88 PTGS2 (0.47) AGTR1PTGS2ABCB1LMNACYP1A2
SCHEMBL6919741 0.87 AGTR1 (0.55) ELANEAGTR1PTGS2ABCB1LMNA
SCHEMBL6922117 0.80 ELANE (0.43) ELANEAGTR1PTGS2ABCB1LMNA
SCHEMBL6820229 0.78 ALDH1A1 (0.43) ELANEAGTR1PTGS2ABCB1LMNA
SCHEMBL6920262 0.78 AGTR1 (0.39) AGTR1PTGS2ABCB1CYP1A2CYP2C9
SCHEMBL7129936 0.78 PLA2G2A (0.41) LMNATSHRNPSR1PLA2G2AMAPK8
SCHEMBL6471641 0.75 POLB (0.45) AGTR1LMNATSHRNPSR1P2RX4
SCHEMBL7130815 0.75 ELANE (0.47) ELANETSHRNPSR1TSPO
SCHEMBL6917789 0.75 MEN1 (0.35) ABCB1TSHRNPSR1PLA2G2AMAPK8
SCHEMBL6920229 0.73 P2RX4 (0.47) ELANEAGTR1PTGS2ABCB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO claimed