SCHEMBL703952

SCHEMBL703952

CC(C)(C)OC(=O)N1CC(F)(F)C[C@H]1CO

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.40
CNR2 P34972 1/20 0.37
RIPK1 Q13546 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SCN9A Q15858 2/20 0.34
HDAC8 Q9BY41 1/20 0.34
TACR1 P25103 6/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL703953 1.00 NR1H2 (0.40) NR1H2CNR2RIPK1MEN1KMT2A
SCHEMBL17001728 1.00 NR1H2 (0.40) NR1H2CNR2RIPK1MEN1KMT2A
SCHEMBL12424302 0.89 NR1H2 (0.35) NR1H2HDAC8CHRM2CHRM1CHRM3
SCHEMBL19127641 0.88 NR1H2 (0.34) NR1H2HDAC8CHRM2CHRM1CHRM3
SCHEMBL21730405 0.88 NR1H2 (0.34) NR1H2HDAC8CHRM2CHRM1CHRM3
SCHEMBL19540623 0.88 NR1H2 (0.34) NR1H2HDAC8CHRM2CHRM1CHRM3
SCHEMBL26922100 0.88 NR1H2 (0.34) NR1H2HDAC8CHRM2CHRM1CHRM3
SCHEMBL17924712 0.86 NR1H2 (0.34) NR1H2MEN1KMT2AHDAC8CHRM2
SCHEMBL16551797 0.86 NR1H2 (0.34) NR1H2MEN1KMT2AHDAC8CHRM2
SCHEMBL16749349 0.86 NR1H2 (0.34) NR1H2MEN1KMT2AHDAC8CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4746969-A1 HETEROCYCLIC PAD4 INHIBITORS Bristol-Myers Squibb Company (US) 2026-05-27 EP disclosed
US-12612414-B2 Nitrile SUMO inhibitors and uses thereof CIT THERAPEUTICS, INC. (US) 2026-04-28 US disclosed
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON INC (US) 2026-03-12 US disclosed
US-20260035365-A1 1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVES AS IRREVERSIBLE INHIBITORS OF MUTANT EGFR FOR THE TREATMENT OF CANCER BAYER AKTIENGESELLSCHAFT (DE) 2026-02-05 US disclosed
US-12509474-B2 Inhibitors of complement factors and uses thereof ANNEXON, INC. (US) 2025-12-30 US disclosed
US-12415789-B2 Macrocycles comprising a 4-amido-2,4-pentadienoate moiety for the treatment of hypoxic cancers AARHUS UNIVERSITET (DK) 2025-09-16 US disclosed
WO-2025125621-A1 CANCER-ASSOCIATED PROTEIN-TARGETED STRONG OR COVALENTLY BINDING PRECURSOR COMPOUNDS AND RADIOTRACERS RADIOVAXX GMBH (DE) 2025-06-19 WO disclosed
EP-4565584-A1 1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVES AS IRREVERSIBLE INHIBITORS OF MUTANT EGFR FOR THE TREATMENT OF CANCER Bayer Aktiengesellschaft (DE) 2025-06-11 EP disclosed
CN-115867282-B 5-Amino-8- (4-pyridyl) - [1,2,4] triazolo [4,3-C ] pyrimidin-3-one compounds for anticancer use 奈克斯拉制药英国有限公司 2025-05-27 CN disclosed
EP-3853234-B1 FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATASE INHIBITORS NIKANG THERAPEUTICS INC (US) 2025-04-23 EP disclosed
WO-2011053705-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed
US-20110105520-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, NV (BE) 2011-05-05 US disclosed
US-20110082165-A1 PYRROLIDINE GPR40 MODULATORS BRISTOL-MYERS SQUIBB COMPANY 2011-04-07 US disclosed
EP-2280970-A1 IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS F. Hoffmann-La Roche AG (CH) 2011-02-09 EP disclosed
WO-2009132986-A1 IMIDAZOLIDINONE DERIVATIVES AS 11B-HSD1 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-11-05 WO disclosed
US-20090275573-A1 Imidazolidinone Derivatives as 11B-HSD1 Inhibitors HOFFMANN-LA ROCHE, INC. 2009-11-05 US disclosed
US-20090257978-A1 Antiviral coumpounds GILEAD SCIENCES, INC. (US) 2009-10-15 US disclosed
US-20090257978-A1 Antiviral coumpounds GILEAD SCIENCES, INC. (US) 2009-10-15 US disclosed
WO-2009005676-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2009-01-08 WO disclosed
US-6221865-B1 INHIBITORS OF PROTEIN FARNESYLTRANSFERASE AND PROTEIN GERANYLGERANYLTRANSFERASE. UNIVERSITY OF PITTSBURGH 2001-04-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090257978-A1 Antiviral coumpounds MAVS, ZC3HAV1, EIF2AK2 NR1H2 1128/4885CNR2 4297/4885RIPK1 3153/4885
US-20110105520-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS OPRD1, OPRK1, OPRM1 NR1H2 39/4885CNR2 52/4885RIPK1 2341/4885
US-12612414-B2 Nitrile SUMO inhibitors and uses thereof SUMO1, SUMO3, PSMB6 NR1H2 2552/4885CNR2 3255/4885RIPK1 2996/4885
US-20090275573-A1 Imidazolidinone Derivatives as 11B-HSD1 Inhibitors HSD11B1, HSD17B1, HSD17B11 NR1H2 138/4885CNR2 3302/4885RIPK1 2335/4885
US-12509474-B2 Inhibitors of complement factors and uses thereof SSB, UACA, CFH NR1H2 1312/4885CNR2 297/4885RIPK1 2710/4885
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFH, CFB, C5 NR1H2 550/4885CNR2 155/4885RIPK1 2681/4885
US-20260035365-A1 1H-PYRROLO[3,2-B]PYRIDINE DERIVATIVES AS IRREVERSIBLE INHIBITORS OF MUTANT EGFR FOR THE TREATMENT OF CANCER EGFR, ERBB2, ERBB3 NR1H2 3296/4885CNR2 390/4885RIPK1 2050/4885
US-20110082165-A1 PYRROLIDINE GPR40 MODULATORS GPR55, GPR65, GPR27 NR1H2 160/4885CNR2 79/4885RIPK1 2241/4885
US-12415789-B2 Macrocycles comprising a 4-amido-2,4-pentadienoate moiety for the treatment of hypoxic cancers DLD, HIF1A, DPYD NR1H2 3171/4885CNR2 818/4885RIPK1 2575/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.