SCHEMBL7445756

SCHEMBL7445756

NC(=O)C(c1cccc(C(F)(F)F)c1)N1CCC(=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.46
EPHX1 P07099 3/20 0.44
CACNA2D1 P54289 1/20 0.44
CACNA1B Q00975 1/20 0.44
CACNB1 Q02641 1/20 0.44
CACNA1C Q13936 1/20 0.44
TRPV1 Q8NER1 1/20 0.43
PNMT P11086 1/20 0.43
TEAD1 P28347 2/20 0.42
OPRM1 P35372 3/20 0.41
OPRD1 P41143 3/20 0.41
OPRK1 P41145 3/20 0.41
OPRL1 P41146 3/20 0.41
SLC6A9 P48067 1/20 0.41
ACP3 P15309 1/20 0.40
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441378 0.85 TEAD1 (0.54) CES2CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL7445606 0.80 ADRA1D (0.41) CACNA2D1CACNA1BCACNB1CACNA1COPRM1
SCHEMBL7434817 0.79 LMNA (0.51) OPRM1OPRD1OPRK1OPRL1
SCHEMBL6246702 0.74 PNMT (0.57) CES2EPHX1PNMTACP3
SCHEMBL7434643 0.74 CES2 (0.38) CES2EPHX1TEAD1CHRM2
SCHEMBL7426489 0.73 CHRM2 (0.38) TEAD1CHRM2
Hydrochloric Acid SCHEMBL14815137 0.73 ALDH1A1 (0.52) CES2CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL15797668 0.72 TEAD1 (0.55) CES2CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL7437442 0.72 TSHR (0.45) CACNA2D1CACNA1BCACNB1CACNA1CTEAD1
SCHEMBL8234510 0.71 PNMT (0.54) CES2EPHX1PNMTACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed