SCHEMBL7656276

SCHEMBL7656276

O=C(O)c1cc(-c2ccc(C(F)(F)F)cc2)c2c3c(ccc2c1)OCO3

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 15/20 0.46
SLC6A2 P23975 3/20 0.44
TMEM97 Q5BJF2 5/20 0.43
HTR1A P08908 2/20 0.43
ADRB3 P13945 2/20 0.43
DRD5 P21918 2/20 0.43
AGTR1 P30556 2/20 0.43
ADRA1B P35368 2/20 0.43
DRD3 P35462 2/20 0.43
SLC6A3 Q01959 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
CYP3A4 P08684 1/20 0.43
KCNH2 Q12809 1/20 0.43
PDE2A O00408 1/20 0.43
PDE5A O76074 1/20 0.43
EGFR P00533 1/20 0.43
INSR P06213 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656847 0.86 AURKA (0.46)
SCHEMBL7652092 0.84 ALDH1A1 (0.50)
SCHEMBL7656725 0.82 NR4A2 (0.45)
SCHEMBL8082276 0.78 FABP4 (0.38) GPR35
SCHEMBL7662193 0.76 ABL1 (0.44) SLC6A2SLC6A4
SCHEMBL7652482 0.74 CHEK2 (0.47) CYP3A4
SCHEMBL8086618 0.73 ALOX5 (0.52) PDE5APTGS2PDE3BPDE3A
SCHEMBL7663316 0.71 GABRA1 (0.45) PDE5A
SCHEMBL7657293 0.71 UCHL1 (0.46)
SCHEMBL8085105 0.71 TDP2 (0.39) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6340704-B1 TREATING NERVE DISEASE OR BONE/JOINT DISEASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-01-22 US disclosed
EP-0975621-A1 CELL DIFFERENTIATION INDUCING AMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-02-02 EP disclosed
WO-1998049155-A1 CELL DIFFERENTIATION INDUCING AMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-05 WO disclosed