SCHEMBL805010

SCHEMBL805010

Brc1cccc(-c2ccc3oc4ccccc4c3c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 5/20 0.56
GABRD O14764 5/20 0.56
GABRA1 P14867 5/20 0.56
GABRB1 P18505 5/20 0.56
GABRG2 P18507 5/20 0.56
GABRB3 P28472 5/20 0.56
GABRA5 P31644 5/20 0.56
GABRA3 P34903 5/20 0.56
GABRA2 P47869 5/20 0.56
GABRB2 P47870 5/20 0.56
GABRA4 P48169 5/20 0.56
GABRE P78334 5/20 0.56
GABRA6 Q16445 5/20 0.56
GABRG1 Q8N1C3 5/20 0.56
GABRG3 Q99928 5/20 0.56
GABRQ Q9UN88 5/20 0.56
MAOB P27338 2/20 0.50
MAOA P21397 1/20 0.50
IDO1 P14902 1/20 0.50
NPC1 O15118 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29632081 1.00 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL30449000 1.00 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL19152582 0.98 GABRP (0.55) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL30038100 0.95 GABRP (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL21890577 0.95 GABRP (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29316451 0.92 GABRP (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL9106871 0.91 GABRP (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL15836118 0.90 GABRA1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL30704825 0.90 GABRA1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL16752108 0.90 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 134 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250393469-A1 ORGANIC ELECTROLUMINESCENCE DEVICE AND POLYCYCLIC COMPOUND FOR ORGANIC ELECTROLUMINESCENCE DEVICE SAMSUNG DISPLAY CO LTD (KR) 2025-12-25 US disclosed
US-20250359477-A1 ORGANIC ELECTROLUMINESCENT ELEMENT, COMPOUND, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2025-11-20 US disclosed
US-12433150-B2 Organic electroluminescence device and polycyclic compound for organic electroluminescence device SAMSUNG DISPLAY CO., LTD. (KR) 2025-09-30 US disclosed
US-20250221309-A1 LIGHT-EMITTING DEVICE INCLUDING CONDENSED CYCLIC COMPOUND, ELECTRONIC APPARATUS INCLUDING THE LIGHT-EMITTING DEVICE, AND THE CONDENSED CYCLIC COMPOUND SAMSUNG DISPLAY CO., LTD. (KR) 2025-07-03 US disclosed
US-20250214956-A1 ORGANIC ELECTRONIC DEVICE AND DISPLAY APPARATUS USING COMPOSITION FOR ORGANIC ELECTRONIC DEVICE DUK SAN NEOLUX CO., LTD. (KR) 2025-07-03 US disclosed
EP-4580379-A1 LIGHT-EMITTING DEVICE COMPRISING CONDENSED CYCLIC COMPOUND, ELECTRONIC APPARATUS COMPRISING THE LIGHT-EMITTING DEVICE, AND THE CONDENSED CYCLIC COMPOUND Samsung Display Co., Ltd. (KR) 2025-07-02 EP disclosed
US-20250051636-A1 HOST MATERIAL, COMPOSITION, AND ORGANIC ELECTROLUMINESCENT ELEMENT KYULUX INC (JP) 2025-02-13 US disclosed
US-12163074-B2 Host material, composition, and organic electroluminescent element KYULUX, INC. (JP) 2024-12-10 US disclosed
US-20240391906-A1 COMPOUND, COMPOSITION, HOST MATERIAL, ELECTRON BARRIER MATERIAL AND ORGANIC LIGHT-EMITTING DEVICE KYULUX, INC. (JP) 2024-11-28 US disclosed
EP-4410789-A1 COMPOUND, COMPOSITION, HOST MATERIAL, ELECTRON BARRIER MATERIAL AND ORGANIC LIGHT EMITTING ELEMENT Kyulux, Inc. (JP) 2024-08-07 EP disclosed
EP-2163550-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME Idemitsu Kosan Co., Ltd. (JP) 2010-03-17 EP disclosed
US-20100001636-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2010-01-07 US disclosed
US-20100001636-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2010-01-07 US disclosed
US-20090030202-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT EMPLOYING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2009-01-29 US disclosed
US-20090030202-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT EMPLOYING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2009-01-29 US disclosed
US-20090017331-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE AND ORGANIC ELECTROLUMINESCENCE DEVICE UTILIZING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2009-01-15 US disclosed
US-20090017331-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE AND ORGANIC ELECTROLUMINESCENCE DEVICE UTILIZING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2009-01-15 US disclosed
US-20080315754-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2008-12-25 US disclosed
US-20080315754-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2008-12-25 US disclosed
US-20080315754-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2008-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12433150-B2 Organic electroluminescence device and polycyclic compound for organic electroluminescence device ODC1, LEF1, L1CAM GABRP 4535/4885GABRD 4486/4885GABRA1 3672/4885
US-20250393469-A1 ORGANIC ELECTROLUMINESCENCE DEVICE AND POLYCYCLIC COMPOUND FOR ORGANIC ELECTROLUMINESCENCE DEVICE SOD1, LIFR, LEF1 GABRP 4086/4885GABRD 4267/4885GABRA1 3309/4885
US-20080315754-A1 ANTHRACENE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME APRT, ETFA, MLLT3 GABRP 4498/4885GABRD 2998/4885GABRA1 3831/4885
US-20250359477-A1 ORGANIC ELECTROLUMINESCENT ELEMENT, COMPOUND, AND ELECTRONIC DEVICE CCNE2, L1CAM, CCNE1 GABRP 4837/4885GABRD 4806/4885GABRA1 4396/4885
US-20090030202-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT EMPLOYING THE SAME EMC2, L1CAM, EMC1 GABRP 3698/4885GABRD 4301/4885GABRA1 3809/4885
US-20240391906-A1 COMPOUND, COMPOSITION, HOST MATERIAL, ELECTRON BARRIER MATERIAL AND ORGANIC LIGHT-EMITTING DEVICE C5, MCM5, CRY1 GABRP 4730/4885GABRD 4535/4885GABRA1 4520/4885
US-20250051636-A1 HOST MATERIAL, COMPOSITION, AND ORGANIC ELECTROLUMINESCENT ELEMENT TRPA1, CRY1, MCM5 GABRP 4698/4885GABRD 4466/4885GABRA1 3288/4885
US-20090017331-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE AND ORGANIC ELECTROLUMINESCENCE DEVICE UTILIZING THE SAME ICMT, ORAI2, ILK GABRP 4200/4885GABRD 4823/4885GABRA1 4577/4885
US-20250214956-A1 ORGANIC ELECTRONIC DEVICE AND DISPLAY APPARATUS USING COMPOSITION FOR ORGANIC ELECTRONIC DEVICE OCIAD2, OCIAD1, EPHA4 GABRP 3537/4885GABRD 2329/4885GABRA1 3505/4885
US-12163074-B2 Host material, composition, and organic electroluminescent element TRPA1, CRY1, MCM5 GABRP 4698/4885GABRD 4466/4885GABRA1 3288/4885
US-20100001636-A1 AROMATIC AMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENCE DEVICE TYR, TERF2, SAT1 GABRP 4721/4885GABRD 4143/4885GABRA1 4344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.