SCHEMBL8264642

SCHEMBL8264642

Oc1cc2c(cn1)CNCC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADCY6 O43306 1/20 0.47
ADCY3 O60266 1/20 0.47
ADCY9 O60503 1/20 0.47
ADCY5 O95622 1/20 0.47
ADCY8 P40145 1/20 0.47
ADCY7 P51828 1/20 0.47
ADCY2 Q08462 1/20 0.47
ADCY1 Q08828 1/20 0.47
ADCY4 Q8NFM4 1/20 0.47
ASIC3 Q9UHC3 2/20 0.43
PNMT P11086 5/20 0.41
CD44 P16070 1/20 0.41
MAOB P27338 1/20 0.41
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
HTR2B P41595 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL587014 0.98 ADCY6 (0.45) ADCY6ADCY3ADCY9ADCY5ADCY8
SCHEMBL25574541 0.92 PNMT (0.43) ADCY6ADCY3ADCY9ADCY5ADCY8
SCHEMBL29627699 0.84 MB (0.31)
SCHEMBL12090705 0.77 PNMT (0.47) ASIC3PNMTCD44MAOBDRD2
SCHEMBL20038301 0.77 PNMT (0.47) ADCY6ADCY3ADCY9ADCY5ADCY8
SCHEMBL10067119 0.77 ASIC3 (0.43) ASIC3PNMTCD44MAOBDRD2
SCHEMBL25574634 0.77 NOS3 (0.57) ASIC3PNMTCD44MAOBDRD2
Hydrochloric Acid SCHEMBL12077907 0.76 PNMT (0.46) ASIC3PNMTCD44MAOBDRD2
Hydrochloric Acid SCHEMBL30062686 0.76 PNMT (0.46) ASIC3PNMTCD44MAOBDRD2
SCHEMBL30524466 0.75 ASIC3 (0.39) ADCY6ADCY3ADCY9ADCY5ADCY8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637455-B2 Naphthyridine and pyrido[3,4-c]pyridazine derivatives as GABAA α5 receptor modulators RICHTER GEDEON NYRT. (HU) 2026-05-26 US disclosed
US-20240067637-A1 NAPHTHYRIDINE AND PYRIDO[3,4-c]PYRIDAZINE DERIVATIVES AS GABAA ALPHA 5 RECEPTOR MODULATORS RICHTER GEDEON NYRT. (HU) 2024-02-29 US disclosed
US-20240067637-A1 NAPHTHYRIDINE AND PYRIDO[3,4-c]PYRIDAZINE DERIVATIVES AS GABAA ALPHA 5 RECEPTOR MODULATORS RICHTER GEDEON NYRT. (HU) 2024-02-29 US disclosed
EP-4126859-A1 NAPHTHYRIDINE AND PYRIDO[3,4-C]PYRIDAZINE DERIVATIVES AS GABAA ALPHA5 RECEPTOR MODULATORS Richter Gedeon Nyrt. (HU) 2023-02-08 EP disclosed
CN-115348962-A As GABA A Naphthyridines and pyrido [3,4-c ] of alpha 5 receptor modulators]Pyridazine derivatives 吉瑞工厂 2022-11-15 CN disclosed
WO-2021191838-A1 NAPHTHYRIDINE AND PYRIDO[3,4-c]PYRIDAZINE DERIVATIVES AS GABAA α5 RECEPTOR MODULATORS RICHTER GEDEON NYRT. (HU) 2021-09-30 WO disclosed
EP-1831199-B1 MMP inhibitors ASTRAZENECA AB (SE) 2012-02-15 EP disclosed
US-20100256166-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2010-10-07 US disclosed
US-20100256166-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2010-10-07 US disclosed
US-7700604-B2 Hydantoin derivatives as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2010-04-20 US disclosed
US-7700604-B2 Hydantoin derivatives as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2010-04-20 US disclosed
US-7655664-B2 Hydantoin derivatives as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2010-02-02 US disclosed
US-7655664-B2 Hydantoin derivatives as metalloproteinase inhibitors ASTRAZENECA AB (SE) 2010-02-02 US disclosed
US-20080293743-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-11-27 US disclosed
US-20080293743-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-11-27 US disclosed
US-20080032997-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-02-07 US disclosed
US-20080032997-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors ASTRAZENECA AB (SE) 2008-02-07 US disclosed
WO-2006065216-A1 NOVEL HYDANTOIN DERIVATIVES AS METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2006-06-22 WO disclosed
WO-2006065215-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2006-06-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100256166-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors MMP1, MMP2, MMP9 ADCY6 2072/4885ADCY3 2222/4885ADCY9 1598/4885
US-20080032997-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors MMP1, MMP2, MMP9 ADCY6 2072/4885ADCY3 2222/4885ADCY9 1598/4885
US-12637455-B2 Naphthyridine and pyrido[3,4-c]pyridazine derivatives as GABAA α5 receptor modulators GABRA5, GABRA1, GABRB1 ADCY6 2284/4885ADCY3 1622/4885ADCY9 1926/4885
US-20240067637-A1 NAPHTHYRIDINE AND PYRIDO[3,4-c]PYRIDAZINE DERIVATIVES AS GABAA ALPHA 5 RECEPTOR MODULATORS GABRA5, GABRA1, GABRA3 ADCY6 3223/4885ADCY3 2574/4885ADCY9 2771/4885
US-20080293743-A1 Novel Hydantoin Derivatives as Metalloproteinase Inhibitors MMP1, MMP2, MMP9 ADCY6 2072/4885ADCY3 2222/4885ADCY9 1598/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.