SCHEMBL9727464

SCHEMBL9727464

CC1(C)c2cc(OCc3ccccc3)c(CCCOc3ccccc3)cc2OC1CCc1ccc(Cl)cc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AKR1B1 P15121 1/20 0.36
BCHE P06276 1/20 0.36
CCR5 P51681 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DUSP3 P51452 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727668 0.86 TDP1 (0.36) TDP1L3MBTL1
SCHEMBL9727665 0.85 L3MBTL1 (0.38) AKR1B1L3MBTL1MEN1KMT2A
SCHEMBL9727331 0.81 MTNR1A (0.37) AKR1B1
SCHEMBL9727653 0.80 ABCB1 (0.38)
SCHEMBL9727777 0.78 AKR1B1 (0.35) KDM4EALDH1A1LMNAAKR1B1KMT2A
SCHEMBL9727725 0.74 AKR1B1 (0.32) ALDH1A1AKR1B1BCHETDP1L3MBTL1
SCHEMBL5502488 0.71 MAOA (0.40)
SCHEMBL9727700 0.69 MTNR1A (0.35) AKR1B1TDP1L3MBTL1
SCHEMBL9727633 0.69 LTA4H (0.38) ALDH1A1AKR1B1DUSP3
SCHEMBL9727620 0.68 CCR5 (0.38) KDM4EALDH1A1LMNAHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed