SCHEMBL9955387

SCHEMBL9955387

Nc1nc2ccc(Br)cc2c(=O)n1-c1cccc(N2CCOCC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.50
IDO2 Q6ZQW0 1/20 0.50
MAPT P10636 5/20 0.43
HTT P42858 2/20 0.43
MAPK1 P28482 1/20 0.43
AHR P35869 1/20 0.43
DHFR P00374 1/20 0.42
LRRK2 Q5S007 2/20 0.41
KMO O15229 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
FLT1 P17948 1/20 0.40
KDR P35968 1/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14247826 0.84 DHFR (0.46) TDO2IDO2MAPTHTTMAPK1
SCHEMBL9952861 0.82 TDO2 (0.46) TDO2IDO2MAPTHTTMAPK1
SCHEMBL9953980 0.81 ATM (0.51) TDO2IDO2MAPTALDH1A1KDM4E
SCHEMBL9954672 0.78 TDO2 (0.52) TDO2IDO2MAPTHTTSMN1; SMN2
SCHEMBL10289024 0.77 SMN1; SMN2 (0.55) MAPTSMN1; SMN2TP53ALDH1A1KDM4E
SCHEMBL9955586 0.77 HPD (0.44) SMN1; SMN2HSD17B10MEN1KMT2A
SCHEMBL9955016 0.76 ALDH1A1 (0.50) MAPTNPC1RAB9ATP53ALOX15
SCHEMBL9954589 0.75 ALOX12 (0.50) MAPTMAPK1RAB9AALDH1A1MEN1
SCHEMBL14247524 0.74 MAPT (0.47) MAPTHTTMAPK1AHRDHFR
SCHEMBL9955086 0.74 CCKBR (0.43) TDO2IDO2MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed