SCHEMBL9955086

SCHEMBL9955086

CN(C)Cc1cccc(-n2c(N)nc3ccc(Br)cc3c2=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.43
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
IDO2 Q6ZQW0 1/20 0.41
ATM Q13315 2/20 0.40
MAPT P10636 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PDE7A Q13946 1/20 0.39
HPD P32754 2/20 0.39
PI4KA P42356 2/20 0.38
PIK3CG P48736 1/20 0.38
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3R1 P27986 1/20 0.38
HTT P42858 1/20 0.38
HIF1A Q16665 1/20 0.38
BCHE P06276 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954482 0.82 CCKBR (0.40) CCKBRIDO1TDO2IDO2ATM
SCHEMBL9953980 0.81 ATM (0.51) IDO1TDO2IDO2ATMMAPT
SCHEMBL10289024 0.80 SMN1; SMN2 (0.55) CCKBRMAPTALDH1A1HPDPI4KA
SCHEMBL9955586 0.75 HPD (0.44) HPDPI4KAPIK3CGSMN1; SMN2MEN1
SCHEMBL9954589 0.75 ALOX12 (0.50) ATMMAPTALDH1A1PI4KAPIK3CG
SCHEMBL9955387 0.74 TDO2 (0.50) TDO2IDO2MAPTALDH1A1SMN1; SMN2
SCHEMBL9954470 0.74 HCAR1 (0.46) ATMMAPTALDH1A1PDE7API4KA
SCHEMBL10288659 0.73 POLB (0.53) IDO1TDO2IDO2ATMMAPT
SCHEMBL9954343 0.72 MAPT (0.49) ATMMAPTALDH1A1LMNAMEN1
SCHEMBL26856831 0.70 TDO2 (0.77) IDO1TDO2IDO2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed