SCHEMBL11200690

SCHEMBL11200690

Nc1ccc(N=Nc2ccc(S(=O)(=O)[O-])cc2)cc1Br.[Na+]

nearest known ligand 0.51

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 known ✓ O43570 7/20 0.51
CA2 known ✓ P00918 7/20 0.51
CA1 known ✓ P00915 1/20 0.51
CA4 known ✓ P22748 1/20 0.51
PTGS1 known ✓ P23219 5/20 0.45
PTGS2 known ✓ P35354 5/20 0.45
THRB known ✓ P10828 1/20 0.43
CA9 Q16790 7/20 0.51
CA7 P43166 2/20 0.51
CA6 P23280 1/20 0.51
CA5A P35218 1/20 0.51
CA14 Q9ULX7 1/20 0.51
CA5B Q9Y2D0 1/20 0.51
SLC7A11 Q9UPY5 2/20 0.51
PLCG1 P19174 1/20 0.49
PHLPP2 Q6ZVD8 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11200679 1.00 CA12 (0.51) CA12CA2CA9CA7CA1
SCHEMBL11200935 0.85 CA2 (0.47) CA12CA2CA9CA7CA1
SCHEMBL11200933 0.85 CA2 (0.47) CA12CA2CA9CA7CA1
SCHEMBL11200703 0.83 POLB (0.53) CA12CA2CA9CA7CA1
SCHEMBL4881910 0.82 SLC7A11 (0.52) CA12CA2CA9CA7SLC7A11
SCHEMBL339834 0.82 SLC7A11 (0.52) CA12CA2CA9CA7SLC7A11
SCHEMBL11202854 0.81 PTGS1 (0.53) CA12CA2CA9CA7CA1
SCHEMBL11202850 0.81 PTGS1 (0.53) CA12CA2CA9CA7CA1
SCHEMBL29837421 0.78 SENP2 (0.50) SLC7A11PLCG1PTGS1PTGS2THRB
SCHEMBL2394481 0.77 CA12 (0.68) CA12CA2CA9CA7CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4419290-A COLORFASTNESS BASF AKTIENGESELLSCHAFT (DE) 1983-12-06 US disclosed