SCHEMBL11200933

SCHEMBL11200933

Nc1c(Br)cc(/N=N/c2ccc(S(=O)(=O)[O-])cc2)cc1Br.[Na+]

nearest known ligand 0.47

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 known ✓ P00918 8/20 0.47
CA12 known ✓ O43570 7/20 0.47
CA1 known ✓ P00915 1/20 0.44
THRB known ✓ P10828 1/20 0.43
PTGS2 known ✓ P35354 3/20 0.42
PTGS1 known ✓ P23219 2/20 0.42
CA9 Q16790 8/20 0.47
SLC7A11 Q9UPY5 3/20 0.47
PLCG1 P19174 1/20 0.47
CA3 P07451 1/20 0.44
APP P05067 1/20 0.43
GLB1 P16278 1/20 0.43
CHAT P28329 1/20 0.43
ENPP2 Q13822 1/20 0.43
PHLPP2 Q6ZVD8 1/20 0.43
CTRC Q99895 1/20 0.43
CA7 P43166 1/20 0.42
FTO Q9C0B1 1/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11200935 1.00 CA2 (0.47) CA2CA9CA12SLC7A11PLCG1
SCHEMBL11200679 0.85 CA12 (0.51) CA2CA9CA12SLC7A11PLCG1
SCHEMBL11200690 0.85 CA12 (0.51) CA2CA9CA12SLC7A11PLCG1
SCHEMBL11200940 0.82 POLB (0.54) CA2CA9CA12CA1CA3
SCHEMBL2394481 0.78 CA12 (0.68) CA2CA9CA12SLC7A11PLCG1
SCHEMBL9618266 0.78 CA12 (0.68) CA2CA9CA12SLC7A11PLCG1
SCHEMBL3511719 0.78 CA2 (0.64) CA2CA9CA12CA1CA3
SCHEMBL4881910 0.73 SLC7A11 (0.52) CA2CA9CA12SLC7A11PLCG1
SCHEMBL339834 0.73 SLC7A11 (0.52) CA2CA9CA12SLC7A11PLCG1
SCHEMBL11658995 0.73 ALDH1A1 (0.50) CA2CA9CA12CA1CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4419290-A COLORFASTNESS BASF AKTIENGESELLSCHAFT (DE) 1983-12-06 US disclosed