SCHEMBL11560437

SCHEMBL11560437

Cc1ncn(-c2ccc(Cl)cc2)c(=O)c1C(=O)[O-].[Na+]

nearest known ligand 0.46

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 1/20 0.39
CA1 known ✓ P00915 1/20 0.38
CA2 known ✓ P00918 1/20 0.38
ESR2 known ✓ Q92731 1/20 0.36
PDK2 known ✓ Q15119 1/20 0.36
RAB9A P51151 2/20 0.46
GRM1 Q13255 8/20 0.42
CYP11B2 P19099 1/20 0.39
GRM5 P41594 1/20 0.38
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11562101 0.97 RAB9A (0.46) RAB9AGRM1CYP11B2PTGS2GRM5
SCHEMBL11560097 0.89 SMN1; SMN2 (0.45) RAB9AGRM1CYP11B2PTGS2GRM5
SCHEMBL11562309 0.86 RAB9A (0.48) RAB9AGRM1CYP11B2GRM5NPC1
Ammonia Solution, Strong SCHEMBL11559116 0.84 RAB9A (0.47) RAB9AGRM1CYP11B2GRM5NPC1
Potassium Ion SCHEMBL11564252 0.80 NPC1 (0.42) RAB9ACA1CA2NPC1
SCHEMBL11563739 0.80 GABRA2 (0.51) RAB9APTGS2CA1CA2NPC1
SCHEMBL14516990 0.75 RAB9A (0.51) RAB9AGRM1CYP11B2PTGS2GRM5
SCHEMBL13985485 0.75 RAB9A (0.51) RAB9AGRM1CYP11B2PTGS2GRM5
SCHEMBL11565008 0.74 SMN1; SMN2 (0.47) RAB9AGRM1CYP11B2GRM5NPC1
SCHEMBL11564209 0.72 HTT (0.46) CA1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4147528-A 6-Oxopyrimidine plant growth regulators ROHM AND HAAS COMPANY (US) 1979-04-03 US disclosed