Fluralaner

Fluralaner

SCHEMBL121934

Cc1cc(C2=NOC(c3cc(Cl)cc(Cl)c3)(C(F)(F)F)C2)ccc1C(=O)NCC(=O)NCC(F)(F)F

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
PTGES O14684 1/20 0.32
HDAC4 P56524 1/20 0.31
ORAI1 Q96D31 4/20 0.31
GABRA5 P31644 1/20 0.31
LMNA P02545 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ELOVL6 Q9H5J4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluralaner SCHEMBL29362559 1.00 CA1 (0.32) CA1CA2PTGESHDAC4ORAI1
Fluralaner SCHEMBL8513367 1.00 CA1 (0.32) CA1CA2PTGESHDAC4ORAI1
Fluralaner SCHEMBL29399660 1.00 CA1 (0.32) CA1CA2PTGESHDAC4ORAI1
Fluralaner SCHEMBL8515337 1.00 CA1 (0.32) CA1CA2PTGESHDAC4ORAI1
SCHEMBL23546689 0.95 GABRA5 (0.31) CA1CA2PTGESGABRA5
SCHEMBL22919822 0.94 PTGES (0.33) PTGESHDAC4KDM4E
SCHEMBL120084 0.94 PTGES (0.33) PTGESHDAC4KDM4E
SCHEMBL15999841 0.94 PTGES (0.31) CA1CA2PTGESGABRA5LMNA
SCHEMBL119374 0.94 PTGES (0.35) CA1CA2PTGESORAI1GABRA5
SCHEMBL23530405 0.93 LMNA (0.32) CA1CA2PTGESORAI1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1644 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2658541-B2 TOPICAL LOCALIZED ISOXAZOLINE FORMULATION COMPRISING GLYCOFUROL INTERVET INT BV (NL) 2025-12-17 EP claimed
US-12396945-B2 Soft chewable pharmaceutical products INTERVET INC. (US) 2025-08-26 US claimed
EP-4008329-B1 ISOXAZOLINE COMPOUNDS FOR USE IN TREATING DEMODICOSIS INTERVET INT BV (NL) 2025-06-11 EP claimed
EP-2658542-B2 TOPICAL LOCALIZED ISOXAZOLINE FORMULATION INTERVET INT BV (NL) 2025-06-04 EP claimed
EP-2833866-B2 SOFT CHEWABLE PHARMACEUTICAL PRODUCTS INTERVET INT BV (NL) 2024-11-27 EP claimed
US-11911503-B2 Manufacturing of semi-plastic pharmaceutical dosage units INTERVET INC. (US) 2024-02-27 US claimed
US-20230276803-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING THIETANYLOXY COMPOUND, OXIDES OR SALTS THEREOF PI INDUSTRIES LTD. (IN) 2023-09-07 US claimed
US-20230276804-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING PYRAZOLOPYRIDINE ANTHRANILAMIDE COMPOUND, OXIDES OR SALTS THEREOF PI INDUSTRIES LTD. (IN) 2023-09-07 US claimed
EP-4188094-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING PYRAZOLOPYRIDINE ANTHRANILAMIDE COMPOUND, OXIDES OR SALTS THEREOF PI Industries Ltd. (IN) 2023-06-07 EP claimed
EP-4175476-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING THIETANYLOXY COMPOUND, OXIDES OR SALTS THEREOF PI Industries Ltd. (IN) 2023-05-10 EP claimed
WO-2011157778-A1 ACTIVE SUBSTANCE COMBINATIONS WITH INSECTICIDE AND ACARICIDE PROPERTIES BAYER CROPSCIENCE AG (DE) 2011-12-22 WO claimed
WO-2011147952-A1 PESTICIDAL MIXTURES BASF SE (DE) 2011-12-01 WO claimed
US-8022089-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-09-20 US claimed
WO-2011025789-A2 FOAMABLE PESTICIDE COMPOSITIONS AND METHODS OF APPLICATION BASF CORPORATION (US) 2011-03-03 WO claimed
US-20100322892-A1 PESTICIDE COMPOSITIONS AND APPLICATORS BASF CORPORATION (US) 2010-12-23 US claimed
US-20100323897-A1 FOAMABLE PESTICIDE COMPOSITIONS BASF CORPORATION (US) 2010-12-23 US claimed
US-20100322990-A1 METHODS FOR CONTROLLING PESTS BASF CORPORATION (US) 2010-12-23 US claimed
WO-2010129345-A2 FOAMABLE PESTICIDE COMPOSITIONS BASF CORPORATION (US) 2010-11-11 WO claimed
WO-2010127019-A1 PESTICIDE COMPOSITIONS AND APPLICATORS BASF CORPORATION (US) 2010-11-04 WO claimed
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-12-17 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11911503-B2 Manufacturing of semi-plastic pharmaceutical dosage units PUF60, RPS11, RPS20 CA1 4870/4885CA2 4861/4885PTGES 99/4885
US-20100323897-A1 FOAMABLE PESTICIDE COMPOSITIONS DDT, PON1, ACHE CA1 2387/4885CA2 2507/4885PTGES 1994/4885
US-20230276804-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING PYRAZOLOPYRIDINE ANTHRANILAMIDE COMPOUND, OXIDES OR SALTS THEREOF ACHE, NOX3, NOX5 CA1 528/4885CA2 40/4885PTGES 2476/4885
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE ATM, CHRM1, NAT1 CA1 1945/4885CA2 725/4885PTGES 4055/4885
US-12396945-B2 Soft chewable pharmaceutical products PAM, TAS2R46, TAS2R16 CA1 1332/4885CA2 158/4885PTGES 203/4885
US-20100322990-A1 METHODS FOR CONTROLLING PESTS DDT, ACHE, PON1 CA1 2289/4885CA2 2176/4885PTGES 2010/4885
US-20230276803-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING THIETANYLOXY COMPOUND, OXIDES OR SALTS THEREOF DDT, ACHE, TH CA1 1246/4885CA2 248/4885PTGES 941/4885
US-20100322892-A1 PESTICIDE COMPOSITIONS AND APPLICATORS DDT, ACHE, CHRM2 CA1 2802/4885CA2 2561/4885PTGES 3958/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.