Xylamidine

Xylamidine

SCHEMBL123846

COc1cccc(OC(C)CNC(=N)Cc2cccc(C)c2)c1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Xylamidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 9/20 0.50
MTNR1B P49286 9/20 0.50
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 3/20 0.41
RECQL P46063 1/20 0.40
POLB P06746 1/20 0.39
PTGER1 P34995 1/20 0.39
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Xylamidine SCHEMBL31307218 0.89 MTNR1A (0.58) MTNR1AMTNR1BALDH1A1POLBMAOB
Xylamidine SCHEMBL12481373 0.84 LMNA (0.40) MTNR1AMTNR1BPKML3MBTL1ALDH1A1
Xylamidine SCHEMBL30201100 0.84 MTNR1A (0.53) MTNR1AMTNR1BALDH1A1MAOB
SCHEMBL30201287 0.73 MTNR1A (0.56) MTNR1AMTNR1BALDH1A1
SCHEMBL31231248 0.69 MTNR1A (0.48) MTNR1AMTNR1BL3MBTL1ALDH1A1
SCHEMBL7539405 0.68 PKM (0.50) PKML3MBTL1POLB
SCHEMBL31231364 0.68 MTNR1A (0.56) MTNR1AMTNR1BALDH1A1RECQL
SCHEMBL30200767 0.67 MTNR1A (0.42) MTNR1AMTNR1BALDH1A1
Xylamidine SCHEMBL2107805 0.66 MAOB (0.47) MTNR1AMTNR1BMAOB
SCHEMBL30200879 0.66 MTNR1A (0.55) MTNR1AMTNR1BL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 226 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11278549-B2 Method of treating obesity MCMASTER UNIVERSITY (CA) 2022-03-22 US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20090220429-A1 METHOD AND A SYSTEM FOR ASSESSING NEUROLOGICAL CONDITIONS METIS CURA EHF (IS) 2009-09-03 US claimed
CN-101155548-A Methods and systems for assessing neurological conditions MENTIS CURA EHF (IS) 2008-04-02 CN claimed
EP-1861003-A1 A METHOD AND A SYSTEM FOR ASSESSING NEUROLOGICAL CONDITIONS Mentis Cura ehf. (IS) 2007-12-05 EP claimed
WO-2006094797-A1 A METHOD AND A SYSTEM FOR ASSESSING NEUROLOGICAL CONDITIONS MENTIS CURA EHF. (IS) 2006-09-14 WO claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
US-20250339367-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-06 US disclosed
US-12403090-B2 Oral film compositions and dosage forms having precise active dissolution profiles AQUESTIVE THERAPEUTICS, INC. (US) 2025-09-02 US disclosed
US-20010023254-A1 Psychological disorders CINCINNATI, UNIVERSITY OF 2001-09-20 US disclosed
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates LUITPOLD PHARMACEUTICALS, INC. 2001-05-31 US disclosed
WO-2000050020-A2 USE OF SULFAMATE DERIVATIVES FOR TREATING IMPULSE CONTROL DISORDERS UNIVERSITY OF CINCINNATI (US) 2000-08-31 WO disclosed
WO-1999030690-A1 ORAL DELIVERY FORMULATION AXIA THERAPEUTICS, INC. (US) 1999-06-24 WO disclosed
US-5795909-A ANTICARCINOGENIC AND ANTITUMOR AGENTS; BREAST, COLON, OVARIANCANCERS NEUROMEDICA, INC. (US) 1998-08-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11278549-B2 Method of treating obesity GPR119, HTR2A, GIPR MTNR1A 14/4885MTNR1B 11/4885PKM 2391/4885
US-20010002404-A1 Fatty acid-pharmaceutical agent conjugates FABP7, FFAR2, FFAR4 MTNR1A 490/4885MTNR1B 641/4885PKM 2367/4885
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES SORD, SLC6A13, CACNA1A MTNR1A 3999/4885MTNR1B 4039/4885PKM 194/4885
US-20010023254-A1 Psychological disorders DRD2, DRD3, DRD1 MTNR1A 458/4885MTNR1B 382/4885PKM 3406/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.