Iofetamine

Iofetamine

SCHEMBL1650085

CC(C)NC(C)Cc1ccc([123I])cc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.66
CYP2D6 P10635 1/20 0.66
APEX1 P27695 1/20 0.63
PMP22 Q01453 1/20 0.63
SLC6A4 P31645 8/20 0.61
SIGMAR1 Q99720 4/20 0.44
TAAR1 Q96RJ0 2/20 0.41
SLC18A2 Q05940 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iofetamine SCHEMBL29617565 0.98 APEX1 (0.67) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL20862299 0.83 CYP1A2 (0.70) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL18211455 0.81 CYP1A2 (0.68) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL11151697 0.79 CYP1A2 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL13996943 0.79 CYP2D6 (0.66) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL23986761 0.79 CYP1A2 (0.66) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL1534301 0.79 CYP1A2 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL13996924 0.79 CYP1A2 (0.66) CYP1A2CYP2D6APEX1PMP22SLC6A4
Iofetamine SCHEMBL3064259 0.79 CYP1A2 (1.00) CYP1A2CYP2D6APEX1PMP22SLC6A4
SCHEMBL10606478 0.79 CYP1A2 (0.66) CYP1A2CYP2D6APEX1PMP22SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3129065-B1 TARGETED DRUG DELIVERY THROUGH AFFINITY BASED LINKERS AKAMARA THERAPEUTICS INC (US) 2026-05-13 EP disclosed
US-12624020-B2 Compositions and methods for preparing and using azetidines UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2026-05-12 US disclosed
US-12616667-B2 Compositions and methods for improving neurological diseases and disorders CURASEN THERAPEUTICS, INC. (US) 2026-05-05 US disclosed
US-12558325-B2 Methods for improving neurological diseases and disorders CURASEN THERAPEUTICS, INC. (US) 2026-02-24 US disclosed
US-20250134835-A1 COMPOSITIONS AND METHODS FOR TREATING PATIENTS WITH AMYOTROPHIC LATERAL SCLEROSIS (ALS) CURASEN THERAPEUTICS, INC. 2025-05-01 US disclosed
CN-118335285-A Postoperative complication prediction method, postoperative complication prediction device, terminal equipment and medium 首都医科大学附属北京天坛医院 2024-07-12 CN disclosed
WO-2024137478-A1 METHODS FOR TREATING VARIOUS CONDITIONS AND INDICATIONS WITH AGONISTS AND ANTAGONISTS CURASEN THERAPEUTICS, INC. (US) 2024-06-27 WO disclosed
US-12016935-B2 Methods for detecting CCR2 receptors WASHINGTON UNIVERSITY (US) 2024-06-25 US disclosed
US-20230414588-A1 COMPOSITIONS AND METHODS FOR TREATING PATIENTS WITH AMYOTROPHIC LATERAL SCLEROSIS (ALS) CURASEN THERAPEUTICS, INC. 2023-12-28 US disclosed
WO-2023250334-A1 COMPOSITIONS AND METHODS INVOLVING ISOLATED COMPOUNDS CURASEN THERAPEUTICS, INC. (US) 2023-12-28 WO disclosed
US-20230121082-A1 COMPOSITIONS AND METHODS FOR PREPARING AND USING AZETIDINES UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2023-04-20 US disclosed
US-11607395-B2 Methods for improving neurological diseases and disorders CURASEN THERAPEUTICS, INC. (US) 2023-03-21 US disclosed
EP-4124344-A1 NOVEL USE OF HIC-5 INHIBITOR Showa University (JP) 2023-02-01 EP disclosed
US-11555082-B2 P-boronophenylalanine derivative and composition containing same, and kit for producing said derivative and composition TOKYO INSTITUTE OF TECHNOLOGY (JP) 2023-01-17 US disclosed
US-11512072-B2 Compositions and methods for preparing and using azetidines UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2022-11-29 US disclosed
EP-3757137-B1 P-BORONOPHENYLALANINE DERIVATIVE AND COMPOSITION CONTAINING SAME, AND KIT FOR PRODUCING SAID DERIVATIVE AND COMPOSITION TOKYO INST TECH (JP) 2022-09-07 EP disclosed
WO-2022051305-A1 COMPOSITIONS AND METHODS FOR IMPROVING NEUROLOGICAL DISEASES AND DISORDERS CURASEN THERAPEUTICS, INC. (US) 2022-03-10 WO disclosed
US-20140010762-A1 IMAGING AGENTS CHROMA THERAPEUTICS LTD (GB) 2014-01-09 US disclosed
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11555082-B2 P-boronophenylalanine derivative and composition containing same, and kit for producing said derivative and composition KIT, SETD7, PAH CYP1A2 3691/4885CYP2D6 2654/4885APEX1 2660/4885
US-11607395-B2 Methods for improving neurological diseases and disorders ADRA2A, ADRA1A, ADRA2B CYP1A2 2333/4885CYP2D6 2854/4885APEX1 3278/4885
US-11512072-B2 Compositions and methods for preparing and using azetidines DGKA, DGKK, PRKG2 CYP1A2 2261/4885CYP2D6 1012/4885APEX1 3087/4885
US-12558325-B2 Methods for improving neurological diseases and disorders ADRB2, ADRB1, ADRA1B CYP1A2 1554/4885CYP2D6 2911/4885APEX1 3192/4885
US-12016935-B2 Methods for detecting CCR2 receptors CCR2, CCR1, CCR5 CYP1A2 3241/4885CYP2D6 2536/4885APEX1 2958/4885
US-20140010762-A1 IMAGING AGENTS CES1, CES2, NCEH1 CYP1A2 912/4885CYP2D6 966/4885APEX1 461/4885
US-12616667-B2 Compositions and methods for improving neurological diseases and disorders ADRB2, ADRB1, ADRA2A CYP1A2 1377/4885CYP2D6 1587/4885APEX1 3723/4885
US-20250134835-A1 COMPOSITIONS AND METHODS FOR TREATING PATIENTS WITH AMYOTROPHIC LATERAL SCLEROSIS (ALS) SMN1; SMN2, HNRNPU, ADRB1 CYP1A2 3912/4885CYP2D6 4266/4885APEX1 4118/4885
US-12624020-B2 Compositions and methods for preparing and using azetidines PRKAR2A, GRK2, GRK6 CYP1A2 2660/4885CYP2D6 723/4885APEX1 3143/4885
US-20230414588-A1 COMPOSITIONS AND METHODS FOR TREATING PATIENTS WITH AMYOTROPHIC LATERAL SCLEROSIS (ALS) SMN1; SMN2, HNRNPU, ADRB1 CYP1A2 3912/4885CYP2D6 4266/4885APEX1 4118/4885
US-20230121082-A1 COMPOSITIONS AND METHODS FOR PREPARING AND USING AZETIDINES DGKA, DGKK, PRKG2 CYP1A2 2261/4885CYP2D6 1012/4885APEX1 3087/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.