SCHEMBL17324271

SCHEMBL17324271

C=CCOC(=O)NC[C@H](N)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GFPT1 Q06210 1/20 0.45
GRIK1 P39086 2/20 0.40
GRIK2 Q13002 2/20 0.40
DDAH1 O94760 1/20 0.38
CASP1 P29466 7/20 0.38
MAPT P10636 1/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC1A3 P43003 1/20 0.33
SLC1A1 P43005 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25660591 1.00 GFPT1 (0.45) GFPT1GRIK1GRIK2DDAH1CASP1
Hydrochloric Acid SCHEMBL31496724 0.98 GFPT1 (0.44) GFPT1GRIK1GRIK2DDAH1CASP1
SCHEMBL16446798 0.89 GFPT1 (0.40) GFPT1GRIK1GRIK2DDAH1CASP1
SCHEMBL15746590 0.84 DDAH1 (0.39) GFPT1GRIK1GRIK2DDAH1CASP1
SCHEMBL24185361 0.83 DDAH1 (0.46) GRIK1GRIK2DDAH1CASP1MAPT
SCHEMBL7194971 0.81 DDAH1 (0.57) GRIK1GRIK2DDAH1CASP1MEN1
SCHEMBL22281180 0.81 DDAH1 (0.57) GRIK1GRIK2DDAH1CASP1MEN1
SCHEMBL28297586 0.81 DDAH1 (0.57) GRIK1GRIK2DDAH1CASP1MEN1
SCHEMBL18159716 0.81 TDP1 (0.39) CASP1MAPTCACNA1BAPBA1MEN1
SCHEMBL1700571 0.80 ARG1 (0.37) GRIK1GRIK2DDAH1CASP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4695268-A1 ANTIBACTERIAL COVALENT PEPTIDE INHIBITORS Université de Bordeaux (FR) 2026-02-18 EP disclosed
CN-113226375-B Methods and compositions 英国研究与创新署 2025-05-13 CN disclosed
EP-4448547-A1 APELINERGIC MACROCYCLES AND USES THEREOF Socpra Sciences Santé Et Humaines S.E.C. (CA) 2024-10-23 EP disclosed
WO-2024213701-A1 ANTIBACTERIAL COVALENT PEPTIDE INHIBITORS UNIVERSITÉ DE BORDEAUX (FR) 2024-10-17 WO disclosed
US-20240343761-A1 APELINERGIC MACROCYCLES AND USES THEREOF SOCPRA SCIENCES SANTÉ ET HUMAINES S.E.C. (CA) 2024-10-17 US disclosed
EP-4445957-A1 ANTIBACTERIAL COVALENT PEPTIDE INHIBITORS Université de Bordeaux (FR) 2024-10-16 EP disclosed
US-20240218041-A1 MOLECULAR DESIGN OF GLUCOSE SENSORS IN GLUCOSE-RESPONSIVE INSULIN ANALOGUES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2024-07-04 US disclosed
US-20240140991-A1 ANTIBIOTIC NATURAL PRODUCT ANALOGUES UNIV BELFAST (GB) 2024-05-02 US disclosed
US-11952379-B2 Small molecule modulators of PAR2 and uses thereof ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2024-04-09 US disclosed
EP-4284816-A1 ANTIBIOTIC NATURAL PRODUCT ANALOGUES The Queen's University of Belfast (GB) 2023-12-06 EP disclosed
WO-2023108291-A9 APELINERGIC MACROCYCLES AND USES THEREOF SOCPRA SCIENCES SANTÉ ET HUMAINES S.E.C. (CA) 2023-09-28 WO disclosed
WO-2023108291-A1 APELINERGIC MACROCYCLES AND USES THEREOF SOCPRA SCIENCES SANTÉ ET HUMAINES S.E.C. (CA) 2023-06-22 WO disclosed
WO-2022162332-A1 ANTIBIOTIC NATURAL PRODUCT ANALOGUES THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2022-08-04 WO disclosed
US-20220010296-A1 METHODS AND COMPOSITIONS UNITED KINGDOM RESEARCH AND INNOVATION (GB) 2022-01-13 US disclosed
CN-113226375-A Methods and compositions 英国研究与创新署 2021-08-06 CN disclosed
US-9764037-B2 Conjugate compounds VICTORIA LINK LIMITED (NZ) 2017-09-19 US disclosed
US-20150352219-A1 CONJUGATE COMPOUNDS VICTORIA LINK LIMITED (NZ) 2015-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240343761-A1 APELINERGIC MACROCYCLES AND USES THEREOF APLNR, AP3D1, AP3B1 GFPT1 2874/4885GRIK1 746/4885GRIK2 586/4885
US-20240218041-A1 MOLECULAR DESIGN OF GLUCOSE SENSORS IN GLUCOSE-RESPONSIVE INSULIN ANALOGUES IAPP, GPR119, INSR GFPT1 119/4885GRIK1 2409/4885GRIK2 2488/4885
US-11952379-B2 Small molecule modulators of PAR2 and uses thereof F2RL1, F2R, TBXA2R GFPT1 3745/4885GRIK1 2209/4885GRIK2 958/4885
US-20240140991-A1 ANTIBIOTIC NATURAL PRODUCT ANALOGUES NRDC, RPS14, SCN11A GFPT1 3824/4885GRIK1 3787/4885GRIK2 3797/4885
US-20150352219-A1 CONJUGATE COMPOUNDS SGMS1, SGMS2, ENPP2 GFPT1 1329/4885GRIK1 1793/4885GRIK2 1999/4885
US-20220010296-A1 METHODS AND COMPOSITIONS TRMT1, TARBP1, RNGTT GFPT1 395/4885GRIK1 3659/4885GRIK2 3471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.