SCHEMBL181531

SCHEMBL181531

O=C1CN(C2NC(=O)NC2=O)C(=O)N1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
CRBN Q96SW2 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
RGS12 O14924 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9838534 0.73 MEN1 (0.35) TSHRTDP1MAPTRGS12LMNA
SCHEMBL7534039 0.69 BRD4 (0.33) TSHRTDP1
SCHEMBL181582 0.68 ALDH1A1 (0.33) ALDH1A1MAPT
SCHEMBL7539678 0.67 CRBN (0.42) CRBNTDP1ALDH1A1MAPT
SCHEMBL1809020 0.67 TSHR (0.38) TSHRTDP1ALDH1A1RGS12
SCHEMBL6632635 0.67 TSHR (0.38) TSHRTDP1ALDH1A1RGS12
SCHEMBL11363682 0.67 TSHR (0.34) TSHRTDP1
SCHEMBL5495774 0.65 TSHR (0.37) TSHRTDP1ALDH1A1
SCHEMBL9402295 0.64 ADAMTS5 (0.33) TSHRCRBNRGS12
SCHEMBL6236013 0.64 OPRM1 (0.46) TSHRCRBNALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9691999-B2 Photoelectric conversion device vapor deposition material, photoelectric conversion device, sensor, and imaging device FUJIFILM CORPORATION (JP) 2017-06-27 US disclosed
US-20150129861-A1 ORGANIC MATERIAL FOR DEPOSITION, AND ORGANIC PHOTOELECTRIC CONVERSION ELEMENT, IMAGING ELEMENT, DEPOSITION METHOD, AND MANUFACTURING METHOD FOR ORGANIC PHOTOELECTRONIC ONVERSION ELEMENT OBTAINED USING THE SAME FUJIFILM CORPORATION (JP) 2015-05-14 US disclosed
US-20140138522-A1 PHOTOELECTRIC CONVERSION DEVICE VAPOR DEPOSITION MATERIAL, PHOTOELECTRIC CONVERSION DEVICE, SENSOR, AND IMAGING DEVICE FUJIFILM CORPORATION (JP) 2014-05-22 US disclosed
US-20120080585-A1 PHOTOELECTRIC CONVERSION ELEMENT, PRODUCTION METHOD THEREOF, PHOTOSENSOR, IMAGING DEVICE AND THEIR DRIVING METHOD FUJIFILM CORPORATION (JP) 2012-04-05 US disclosed
US-20120025179-A1 PHOTOELECTRIC CONVERSION ELEMENT AND IMAGING DEVICE FUJIFILM CORPORATION (JP) 2012-02-02 US disclosed
EP-2403027-A1 Photoelectric conversion device and imaging device Fujifilm Corporation (JP) 2012-01-04 EP disclosed
US-8053661-B2 Photoelectric conversion element and imaging device FUJIFILM CORPORATION (JP) 2011-11-08 US disclosed
US-20110263610-A1 COMPOUNDS AND COMPOSITIONS AS ITPKB INHIBITORS IRM LLC (BM) 2011-10-27 US disclosed
US-20110220843-A1 POLYMER FILM, ULTRAVIOLET ABSORBER, MEROCYANINE COMPOUND AND PROCESS FOR PREPARING MEROCYANINE COMPOUND FUJIFILM CORPORATION (JP) 2011-09-15 US disclosed
WO-2011111589-A1 PHOTOELECTRIC CONVERSION DEVICE AND IMAGING DEVICE FUJIFILM CORPORATION (JP) 2011-09-15 WO disclosed
US-20110056562-A1 PHOTOELECTRIC CONVERSION MATERIAL, FILM CONTAINING THE MATERIAL, PHOTOELECTRIC CONVERSION DEVICE, PRODUCTION METHOD THEREOF, PHOTOSENSOR, IMAGING DEVICE AND THEIR USE METHODS FUJIFILM CORPORATION (JP) 2011-03-10 US disclosed
EP-2292586-A2 Photoelectric conversion material, film containing the material, photoelectric conversion device, production method thereof, photosensor, imaging device and their use methods Fujifilm Corporation (JP) 2011-03-09 EP disclosed
US-20110012075-A1 INFRARED ABSORPTIVE COMPOUND, AND FINE PARTICLE CONTAINING THE COMPOUND FUJIFILM CORPORATION (JP) 2011-01-20 US disclosed
EP-2274302-A2 COMPOUNDS AND COMPOSITIONS AS ITPKB INHIBITORS IRM LLC (BM) 2011-01-19 EP disclosed
EP-2272849-A1 COMPOUND CAPABLE OF ABSORBING INFRARED RAY, AND MICROPARTICLES COMPRISING THE COMPOUND FUJIFILM Corporation (JP) 2011-01-12 EP disclosed
US-7557175-B2 Poly(carbonate-co-urea) copolymers and melt transesterification method of preparing these copolymers SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2009-07-07 US disclosed
US-20030134148-A1 Novel methine compound, material for organic luminescence element, and organic luminescence element using the same FUJI PHOTO FILM CO., LTD. 2003-07-17 US disclosed
EP-0822447-B1 Photopolymerizable composition FUJI PHOTO FILM CO LTD (JP) 2000-10-11 EP disclosed
US-5939465-A COMPRISING N-HETEROCYCLE COMPOUND, COMPOUND CONTAINING AT LEAST ONE ADDITION-POLYMERIZABLE, ETHYLENICALLY UNSATURATED BOND, AND COMPOUND WHICH GENERATES AN ACTIVE RADICAL UPON IRRADIATION OF LIGHT FUJI PHOTO FILM CO., LTD. (JP) 1999-08-17 US disclosed
EP-0822447-A1 Photopolymerizable composition FUJI PHOTO FILM CO., LTD. (JP) 1998-02-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120080585-A1 PHOTOELECTRIC CONVERSION ELEMENT, PRODUCTION METHOD THEREOF, PHOTOSENSOR, IMAGING DEVICE AND THEIR DRIVING METHOD SUN2, CYBA, PPOX TSHR 3845/4885CRBN 3566/4885TDP1 4072/4885
US-20110056562-A1 PHOTOELECTRIC CONVERSION MATERIAL, FILM CONTAINING THE MATERIAL, PHOTOELECTRIC CONVERSION DEVICE, PRODUCTION METHOD THEREOF, PHOTOSENSOR, IMAGING DEVICE AND THEIR USE METHODS H1-0, CRY1, PYM1 TSHR 938/4885CRBN 3981/4885TDP1 3996/4885
US-20110220843-A1 POLYMER FILM, ULTRAVIOLET ABSORBER, MEROCYANINE COMPOUND AND PROCESS FOR PREPARING MEROCYANINE COMPOUND HAMP, CRY1, CRY2 TSHR 4451/4885CRBN 599/4885TDP1 4468/4885
US-20110012075-A1 INFRARED ABSORPTIVE COMPOUND, AND FINE PARTICLE CONTAINING THE COMPOUND RRP1B, C9, MRPS22 TSHR 182/4885CRBN 1531/4885TDP1 4085/4885
US-20110263610-A1 COMPOUNDS AND COMPOSITIONS AS ITPKB INHIBITORS IP6K1, IP6K2, IP6K3 TSHR 3960/4885CRBN 1880/4885TDP1 1634/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.