SCHEMBL23716720

SCHEMBL23716720

Cc1ncn(C)c1C(=O)[O-].[Na+]

nearest known ligand 0.40

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APOBEC3A P31941 4/20 0.40
APOBEC3G Q9HC16 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.32
CTDSP1 Q9GZU7 2/20 0.32
BCAT2 O15382 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
CYP2C19 P33261 1/20 0.31
KDM2B Q8NHM5 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
GAA P10253 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23716719 0.78 APOBEC3A (0.41) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2
SCHEMBL25457959 0.74 APOBEC3A (0.46) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2
SCHEMBL7375007 0.73 APOBEC3A (0.38) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2
SCHEMBL23367000 0.73 APOBEC3A (0.41) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2
SCHEMBL5937208 0.72 ALDH1A1 (0.47) APOBEC3AAPOBEC3GSMN1; SMN2LMNAHPGD
Hydrochloric Acid SCHEMBL23354063 0.72 APOBEC3A (0.40) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1HPGD
SCHEMBL23930918 0.71 GABRA1 (0.36) APOBEC3AAPOBEC3GTP53CYP2C19ALDH1A1
SCHEMBL23354512 0.69 APOBEC3A (0.38) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2
SCHEMBL23900462 0.63 BCAT2 (0.47) BCAT2LMNAHPGDKDM4ENPC1
SCHEMBL21879818 0.63 APOBEC3A (0.42) APOBEC3AAPOBEC3GSMN1; SMN2CTDSP1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715609-B Cyclohexylbenzamide compounds 伊莱利利公司 2023-01-10 CN disclosed
EP-3487840-B1 CYCLOHEXYL BENZAMIDE COMPOUNDS LILLY CO ELI (US) 2021-08-11 EP disclosed
CN-109715609-A Cyclohexylbenzoyl amine compounds 伊莱利利公司 2019-05-03 CN disclosed