SCHEMBL2587088

SCHEMBL2587088

O=C(NCc1ccc(F)cc1F)c1noc2ccncc12

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
P2RX7 Q99572 2/20 0.45
ROCK2 O75116 6/20 0.44
MAOB P27338 1/20 0.42
MET P08581 1/20 0.42
KCNK3 O14649 1/20 0.40
PDE10A Q9Y233 1/20 0.40
HSD17B13 Q7Z5P4 1/20 0.39
DGAT2 Q96PD7 3/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581145 0.80 TSHR (0.50) P2RX7ROCK2
SCHEMBL2585532 0.76 HIF1A (0.52) GSK3BKMT2AROCK2HIF1A
SCHEMBL2584587 0.76 ROCK2 (0.48) MEN1KMT2AP2RX7ROCK2DGAT2
SCHEMBL2582356 0.72 KMT2A (0.46) GSK3BMEN1KMT2AHIF1A
SCHEMBL6543656 0.72 THRB (0.55) GSK3BMEN1KMT2A
SCHEMBL2589092 0.72 HIF1A (0.43) GSK3BROCK2HIF1A
SCHEMBL2585927 0.71 WNT1 (0.46) HIF1A
SCHEMBL2576273 0.71 ALDH1A1 (0.48) MEN1KMT2AHIF1A
SCHEMBL5083302 0.71 CXCR4 (0.60) GSK3BMEN1KMT2AP2RX7ROCK2
SCHEMBL2585707 0.70 RAB9A (0.54) MEN1KMT2AHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed