Tromethamine

Tromethamine

SCHEMBL3104874

Cc1ccc(P)cc1.NC(CO)(CO)CO

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DHFRGARTPTGFRPTGIRPTGS1PTGS2TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8envmurAthyA

The experimentally established mechanism targets of Tromethamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ACHE P22303 3/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 2/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
S1PR1 P21453 4/20 0.34
S1PR3 Q99500 3/20 0.34
TNNC1 P63316 5/20 0.33
SGPL1 O95470 1/20 0.33
S1PR4 O95977 1/20 0.33
GPR183 P32249 1/20 0.33
CERS2 Q96G23 1/20 0.33
S1PR5 Q9H228 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GSK3B P49841 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tromethamine SCHEMBL5702541 0.83 LMNA (0.43) LMNAMEN1KMT2AACHETDP1
P-Cresol SCHEMBL1904230 0.80 ACHE (0.59) LMNAMEN1KMT2AACHETDP1
Tromethamine SCHEMBL5564327 0.80 ACHE (0.59) LMNAMEN1KMT2AACHETDP1
Tromethamine SCHEMBL7181961 0.78 LMNA (0.43) LMNAMEN1KMT2AACHETDP1
Tromethamine SCHEMBL7101299 0.78 ALDH1A1 (0.42) LMNAMEN1KMT2ATDP1ALDH1A1
SCHEMBL193486 0.75
Tromethamine SCHEMBL1290395 0.75 CES2 (0.42) LMNAMEN1KMT2ACES2CES1
Tromethamine SCHEMBL4329786 0.75 NQO1 (0.50) KMT2ATDP1ALDH1A1
SCHEMBL15362252 0.74 CYP1A2 (0.41) LMNAMEN1KMT2AACHES1PR1
Bromide SCHEMBL7197581 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230382856-A1 METHOD OF PRODUCING 3-METHYL-4-HALO-INDOLE DERIVATIVE DAIICHI SANKYO COMPANY, LIMITED (JP) 2023-11-30 US disclosed
EP-4238961-A1 METHOD OF PRODUCING 3-METHYL-4-HALO-INDOLE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2023-09-06 EP disclosed
US-8242217-B2 Epoxy resin curing agent, process for preparing the same, and epoxy resin composition SHOWA DENKO K.K. (JP) 2012-08-14 US disclosed
US-20100273940-A1 EPOXY RESIN CURING AGENT, PROCESS FOR PREPARING THE SAME, AND EPOXY RESIN COMPOSITION SHOWA DENKO K.K. (JP) 2010-10-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230382856-A1 METHOD OF PRODUCING 3-METHYL-4-HALO-INDOLE DERIVATIVE INMT, TDO2, HNMT LMNA 2502/4885MEN1 3840/4885KMT2A 99/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.