SCHEMBL337724

SCHEMBL337724

O=C1CCC(C(=O)O)=NN1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 3/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
SMYD3 Q9H7B4 1/20 0.42
ALDH1A1 P00352 4/20 0.40
GFER P55789 1/20 0.40
RXFP1 Q9HBX9 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 1/20 0.37
RECQL P46063 1/20 0.37
MME P08473 1/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13938473 0.80 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL5201218 0.80 SMYD3 (0.44) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL7875062 0.79
SCHEMBL10045647 0.77 LMNA (0.44) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL27040299 0.71 LMNA (0.40) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL13779949 0.69 ALDH1A1 (0.59) NPC1RAB9AMAPTALDH1A1GFER
SCHEMBL338764 0.68 SMN1; SMN2 (0.39) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL27040200 0.68 SMN1; SMN2 (0.39) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL5865621 0.67
SCHEMBL6503803 0.66 SMN1; SMN2 (0.67) SMN1; SMN2MAPTLMNAMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 146 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11912666-B2 Synthesis of 6-oxo-1,4,5,6-tetrahydropyridizin-3-carboxylic acid MILLENNIUM ENTPR INC (US) 2024-02-27 US claimed
US-11800869-B2 Use of 6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxylic acid, 1-methyl 6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxylic acid and 1-alkyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxylic acid for improving growth performance in plants Advanced Crop Chem LLP (US) 2023-10-31 US claimed
US-20220372002-A1 SYNTHESIS OF 6-OXO-1,4,5,6-TETRAHYDROPYRIDIZIN-3-CARBOXYLIC ACID Millennium Enterprises, Inc. (US) 2022-11-24 US claimed
EP-1814880-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS, COMPOSITIONS, USES AND METHODS RELATED THERETO FERRER INT (ES) 2009-01-28 EP claimed
US-20080200473-A1 Imidazo [1,2-a]Pyridine Compounds, Compositions, Uses and Methods Thereto FERRER INTERNACIONAL, S.A. (ES) 2008-08-21 US claimed
US-6946462-B2 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents HOFFMANN-LA ROCHE INC. (US) 2005-09-20 US claimed
US-6869953-B2 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents HOFFMAN-LA ROCHE INC. (US) 2005-03-22 US claimed
US-20040192744-A1 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents HAAG RAINER (DE) 2004-09-30 US claimed
US-20030139404-A1 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents HOFFMANN-LA ROCHE INC. 2003-07-24 US claimed
US-20250382240-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SALARIUS PHARMACEUTICALS INC (US) 2025-12-18 US disclosed
US-20250302838-A1 3-(SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME DEUTERX LLC (US) 2025-10-02 US disclosed
EP-4554674-A1 BIARYL ETHER UREA COMPOUNDS AS FAAH INHIBITORS Jazz Pharmaceuticals Ireland Limited (IE) 2025-05-21 EP disclosed
US-20240101552-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF SHANGHAI PHARMACEUTICALS HOLDING CO., LTD. (CN) 2024-03-28 US disclosed
US-11935803-B2 Resin composition, laminate, semiconductor wafer with resin composition layer, substrate for mounting semiconductor with resin composition layer and semiconductor device MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2024-03-19 US disclosed
US-5559232-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1996-09-24 US disclosed
EP-0641779-A1 Novel 1-amidinopiperdines and 4-amidinomorpholines as aggregation inhibitions F. HOFFMANN-LA ROCHE AG (CH) 1995-03-08 EP disclosed
US-5229386-A Anticoagulants, hypotensive agents, antiallergens, antiinflammatory agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-07-20 US disclosed
US-5145860-A Anticoagulants, vasodilators, antiinflammatory, antiallergens, enzyme inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-09-08 US disclosed
WO-1992002513-A1 HETEROCYCLIC COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-02-20 WO disclosed
EP-0388909-A2 Thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-09-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040192744-A1 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents NAT1, CYP1A1, UGT1A1 NPC1 71/4885RAB9A 2425/4885SMN1; SMN2 2811/4885
US-20220372002-A1 SYNTHESIS OF 6-OXO-1,4,5,6-TETRAHYDROPYRIDIZIN-3-CARBOXYLIC ACID OGDH, PGD, HPD NPC1 3824/4885RAB9A 4695/4885SMN1; SMN2 4045/4885
US-20240101552-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF LANCL2, CBS, LCP2 NPC1 1564/4885RAB9A 2591/4885SMN1; SMN2 3536/4885
US-20250302838-A1 3-(SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME AQP3, AQP4, AQP1 NPC1 571/4885RAB9A 2873/4885SMN1; SMN2 1263/4885
US-20250382240-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME IL5, TLR5, IDO1 NPC1 2138/4885RAB9A 2388/4885SMN1; SMN2 1721/4885
US-20080200473-A1 Imidazo [1,2-a]Pyridine Compounds, Compositions, Uses and Methods Thereto GABRA1, GABRA2, GABRA3 NPC1 807/4885RAB9A 1380/4885SMN1; SMN2 1951/4885
US-11912666-B2 Synthesis of 6-oxo-1,4,5,6-tetrahydropyridizin-3-carboxylic acid OGDH, PGD, HPD NPC1 3824/4885RAB9A 4695/4885SMN1; SMN2 4045/4885
US-20030139404-A1 N-monoacylated derivatives of o-phenylenediamines, their analogs and their use as pharmaceutical agents NAT1, CYP1A1, UGT1A1 NPC1 71/4885RAB9A 2425/4885SMN1; SMN2 2811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.