Cocarboxylase

Cocarboxylase

SCHEMBL344290

Cc1ncc(C[n+]2csc(CCOP(=O)(O)OP(=O)(O)O)c2C)c(N)n1.O.O.O.O.[Cl-]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Cocarboxylase. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.96
TKT P29401 7/20 0.83
TDP1 Q9NUW8 1/20 0.82
HSP90AA1 P07900 1/20 0.62
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 1/20 0.53
PPP5C P53041 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cocarboxylase SCHEMBL27898926 0.99 LMNA (0.98) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL21111 0.99 LMNA (0.98) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL8923435 0.99 LMNA (0.98) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL23151784 0.98 LMNA (0.96) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL662896 0.98 LMNA (0.96) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL30192281 0.98 LMNA (1.00) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL80028 0.98 LMNA (1.00) LMNATKTTDP1HSP90AA1ALDH1A1
Hydrochloric Acid SCHEMBL9766249 0.97 LMNA (0.94) LMNATKTTDP1HSP90AA1ALDH1A1
Hydrochloric Acid SCHEMBL478202 0.97 LMNA (0.94) LMNATKTTDP1HSP90AA1ALDH1A1
Cocarboxylase SCHEMBL23151785 0.97 LMNA (0.98) LMNATKTTDP1HSP90AA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 113 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4537826-A1 METHOD FOR TREATING MENTAL DISEASES Shanghai Raising Pharmaceutical Co., Ltd. (CN) 2025-04-16 EP claimed
CN-119384278-A Method for treating mental diseases 上海日馨医药科技股份有限公司 2025-01-28 CN claimed
CN-117756852-A Preparation method of cocarboxylase tetrahydrate 燃点(南京)生物医药科技有限公司 2024-03-26 CN claimed
WO-2023236781-A1 METHOD FOR TREATING MENTAL DISEASES 上海日馨医药科技股份有限公司 2023-12-14 WO claimed
CN-116270503-A Preparation method of 12 compound vitamins for injection 天津汉瑞药业有限公司 2023-06-23 CN claimed
CN-113402555-B Preparation method of cocarboxylase and tetrahydrate or salt thereof 上海医药工业研究院 2022-12-30 CN claimed
CN-113402555-A Preparation method of cocarboxylase and tetrahydrate or salt thereof 上海医药工业研究院 2021-09-17 CN claimed
CN-111007162-A Method for simultaneously detecting contents of two impurities of cocarboxylase tetrahydrate 济南康和医药科技有限公司 2020-04-14 CN claimed
CN-110988233-A Method for detecting impurity A content of cocarboxylase tetrahydrate 济南康和医药科技有限公司 2020-04-10 CN claimed
CN-108634093-A It is a kind of can strengthen immunity piglet feed 南安市创培电子科技有限公司 2018-10-12 CN claimed
US-20130287757-A1 COMPOSITION FOR THE REGENERATION OF ATROPHIC TISSUES MEDESTEA INTERNAZIONALE S.P.A. (IT) 2013-10-31 US claimed
CN-103351407-A Novel crystal form of cocarboxylase tetrahydrate SICHUAN HAISCO PHARMACEUTICAL CO LTD 2013-10-16 CN claimed
WO-2012095702-A1 A COMPOSITION FOR THE REGENERATION OF ATROPHIC TISSUES MEDESTEA INTERNAZIONALE S.P.A. (IT) 2012-07-19 WO claimed
CN-102068453-B Stable complex vitamin composition and preparation method thereof BEIJING JINGWEI XINKANG MEDICAL TECHNOLOGY CO LTD 2012-01-11 CN claimed
CN-102068453-A Stable complex vitamin composite and preparation method thereof BEIJING JINGWEI XINKANG MEDICAL TECHNOLOGY CO LTD 2011-05-25 CN claimed
CN-101787049-B Novel crystal form of cocarboxylase tetrahydrate and preparation method thereof BEIJING JINGWEI XINKANG MED TECH CO LTD 2011-04-20 CN claimed
CN-101787048-B Preparation method of cocarboxylase tetrahydrate BEIJING JINGWEI XINKANG MED TECH CO LTD 2011-04-06 CN claimed
CN-101787049-A Novel crystal form of cocarboxylase tetrahydrate and preparation method thereof BEIJING JINGWEI XINKANG MED TE 2010-07-28 CN claimed
CN-101787048-A Preparation method of cocarboxylase tetrahydrate BEIJING JINGWEI XINKANG MED TE 2010-07-28 CN claimed
CN-101711769-A Stable injection composite of 12 complex vitamins and preparation method thereof BEIJING JINGWEIXINKANG PHARMAC 2010-05-26 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130287757-A1 COMPOSITION FOR THE REGENERATION OF ATROPHIC TISSUES CUTA, UNG, MMP1 LMNA 3710/4885TKT 661/4885TDP1 942/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.