SCHEMBL425352

SCHEMBL425352

CC(=O)NCCCN1CCCC1=O

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.60
NPC1 O15118 2/20 0.60
KMT2A Q03164 4/20 0.59
SMN1; SMN2 Q16637 2/20 0.57
MEN1 O00255 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
ALDH1A1 P00352 2/20 0.54
TSHR P16473 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548290 0.90 KMT2A (0.71) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL11479783 0.87 KMT2A (0.67) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL5656878 0.85 RAB9A (0.61) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL16254590 0.85 KMT2A (0.65) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL6359808 0.84 RAB9A (0.60) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL17057207 0.84 KMT2A (0.83) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL425351 0.84 SMN1; SMN2 (0.57) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL22838012 0.84 KMT2A (0.63) RAB9ANPC1KMT2ASMN1; SMN2L3MBTL1
SCHEMBL9911470 0.83 RAB9A (0.56) RAB9ANPC1KMT2ASMN1; SMN2MEN1
SCHEMBL13612784 0.83 RAB9A (0.56) RAB9ANPC1KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 135 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12578322-B2 Methods and consumer products for detecting a metabolite KIMBERLY-CLARK WORLDWIDE, INC. (US) 2026-03-17 US claimed
EP-4237090-B1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER UNIV TEXAS (US) 2026-02-18 EP claimed
CN-119968213-A Methods for detecting and treating ovarian cancer 德州大学系统董事会 2025-05-09 CN claimed
EP-3967217-B1 BLOOD BASED BIOMARKERS FOR DIAGNOSING ATHEROSCLEROTIC CORONARY ARTERY DISEASE GLOBAL GENOMICS GROUP LLC (US) 2024-08-14 EP claimed
US-20240044902-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-02-08 US claimed
US-20230417734-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. 2023-12-28 US claimed
EP-4237090-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER Board of Regents, The University of Texas System (US) 2023-09-06 EP claimed
CN-116660543-A Diagnostic and prognostic markers for nonalcoholic fatty liver disease and uses thereof 中国人民解放军陆军军医大学第一附属医院 2023-08-29 CN claimed
CN-116490776-A Methods for detecting and treating ovarian cancer 德州大学系统董事会 2023-07-25 CN claimed
WO-2022125057-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. (US) 2022-06-16 WO claimed
WO-2022093960-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-05-05 WO claimed
EP-3967217-A1 BLOOD BASED BIOMARKERS FOR DIAGNOSING ATHEROSCLEROTIC CORONARY ARTERY DISEASE Global Genomics Group, LLC (US) 2022-03-16 EP claimed
CN-113156096-A Blood-based biomarkers for diagnosing coronary atherosclerotic disease 全球基因集团有限责任公司 2021-07-23 CN claimed
CN-107427221-B Blood-based biomarkers for diagnosing coronary atherosclerotic disease 全球基因集团有限责任公司 2021-03-09 CN claimed
US-8148537-B2 Substituted acetophenones useful as PDE4 inhibitors LEO PHARMA A/S (DK) 2012-04-03 US claimed
EP-2125736-B1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA AS (DK) 2011-03-30 EP claimed
US-20100035908-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA (DK) 2010-02-11 US claimed
EP-2125736-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS Leo Pharma A/S (DK) 2009-12-02 EP claimed
WO-2008077404-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA A/S (DK) 2008-07-03 WO claimed
EP-3990899-B1 QUANTITATIVE RAMAN SPECTROSCOPY AALTO UNIV FOUNDATION SR (FI) 2026-05-20 EP disclosed
US-12578322-B2 Methods and consumer products for detecting a metabolite KIMBERLY-CLARK WORLDWIDE, INC. (US) 2026-03-17 US disclosed
US-12578322-B2 Methods and consumer products for detecting a metabolite KIMBERLY-CLARK WORLDWIDE, INC. (US) 2026-03-17 US disclosed
US-12571737-B2 Quantitative Raman spectroscopy AALTO UNIVERSITY FOUNDATION SR (FI) 2026-03-10 US disclosed
US-12566161-B2 Methods and consumer products for detecting a metabolite KIMBERLY-CLARK WORLDWIDE, INC. (US) 2026-03-03 US disclosed
EP-4237090-B1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER UNIV TEXAS (US) 2026-02-18 EP disclosed
US-20250295713-A1 COMPOSITIONS AND METHODS FOR IMPROVING SKIN HEALTH AND FOR THE TREATMENT AND PREVENTION OF DISEASES, DISORDERS AND CONDITIONS ASSOCIATED WITH PATHOGENIC MICROBES DERMBIONT, INC. 2025-09-25 US disclosed
EP-4604968-A1 ENHANCED NAD+ COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME Bionadrx Holdings, Inc. (US) 2025-08-27 EP disclosed
CN-119968213-A Methods for detecting and treating ovarian cancer 德州大学系统董事会 2025-05-09 CN disclosed
CN-119968213-A Methods for detecting and treating ovarian cancer 德州大学系统董事会 2025-05-09 CN disclosed
US-20250138016-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2025-05-01 US disclosed
US-12259397-B2 Biomarkers related to organ function University of Pittsburgh—of the Commonwealth System of Higher Education (US) 2025-03-25 US disclosed
CN-114341625-B Quantitative raman spectroscopy 阿尔托大学注册基金会 2025-03-11 CN disclosed
CN-118671346-B Metabolic marker for gastric cancer diagnosis and application thereof 浙江省肿瘤医院 2024-11-15 CN disclosed
CN-118671346-A Metabolic marker for gastric cancer diagnosis and application thereof 浙江省肿瘤医院 2024-09-20 CN disclosed
US-12064459-B2 Compositions and methods for improving skin health and for the treatment and prevention of diseases, disorders and conditions associated with pathogenic microbes DERMBIONT, INC. (US) 2024-08-20 US disclosed
EP-3967217-B1 BLOOD BASED BIOMARKERS FOR DIAGNOSING ATHEROSCLEROTIC CORONARY ARTERY DISEASE GLOBAL GENOMICS GROUP LLC (US) 2024-08-14 EP disclosed
US-20240257973-A1 DISEASE SPECTRUM CLASSIFICATION PATIENTSLIKEME LLC (US) 2024-08-01 US disclosed
US-20240230622-A9 Methods and Systems for Determining Autism Spectrum Disorder Risk LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2024-07-11 US disclosed
US-20240133865-A1 Methods and Systems for Determining Autism Spectrum Disorder Risk LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2024-04-25 US disclosed
WO-2024086312-A1 ENHANCED NAD+ COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME BIONADRX HOLDINGS, INC. DBA BRYLEOS (US) 2024-04-25 WO disclosed
US-20240044902-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-02-08 US disclosed
US-11894139-B1 Disease spectrum classification PATIENTSLIKEME LLC (US) 2024-02-06 US disclosed
US-20240019417-A1 Methods and Systems for Determining Autism Spectrum Disorder Risk LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2024-01-18 US disclosed
US-20230417734-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. 2023-12-28 US disclosed
US-20230417734-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. 2023-12-28 US disclosed
US-20230400438-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. 2023-12-14 US disclosed
EP-4237090-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER Board of Regents, The University of Texas System (US) 2023-09-06 EP disclosed
CN-116490776-A Methods for detecting and treating ovarian cancer 德州大学系统董事会 2023-07-25 CN disclosed
US-11674948-B2 Methods and systems for determining autism spectrum disorder risk LABORATORY CORPORATION OF AMERICA HOLDINGS (US) 2023-06-13 US disclosed
US-20230158088-A1 COMPOSITIONS FOR MODULATING GUT MICROFLORA POPULATIONS, ENHANCING DRUG POTENCY AND TREATING VIRAL INFECTIONS, AND METHODS FOR MAKING AND USING SAME PERSEPHONE BIOSCIENCES INC (US) 2023-05-25 US disclosed
US-20220364997-A1 QUANTITATIVE RAMAN SPECTROSCOPY AALTO UNIVERSITY FOUNDATION SR (FI) 2022-11-17 US disclosed
WO-2022125057-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. (US) 2022-06-16 WO disclosed
WO-2022125057-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. (US) 2022-06-16 WO disclosed
WO-2022125056-A1 METHODS AND CONSUMER PRODUCTS FOR DETECTING A METABOLITE KIMBERLY-CLARK WORLDWIDE, INC. (US) 2022-06-16 WO disclosed
US-20220160617-A1 COMPOSITIONS AND METHODS FOR IMPROVING SKIN HEALTH AND FOR THE TREATMENT AND PREVENTION OF DISEASES, DISORDERS AND CONDITIONS ASSOCIATED WITH PATHOGENIC MICROBES DERMBIONT, INC. 2022-05-26 US disclosed
WO-2022093960-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-05-05 WO disclosed
WO-2022093960-A1 METHODS FOR THE DETECTION AND TREATMENT OF OVARIAN CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2022-05-05 WO disclosed
EP-3990899-A1 QUANTITATIVE RAMAN SPECTROSCOPY Aalto University Foundation sr (FI) 2022-05-04 EP disclosed
CN-114341625-A Quantitative Raman spectroscopy 阿尔托大学注册基金会 2022-04-12 CN disclosed
US-20220102000-A1 PREDICTING BLOOD METABOLITES YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2022-03-31 US disclosed
EP-3967217-A1 BLOOD BASED BIOMARKERS FOR DIAGNOSING ATHEROSCLEROTIC CORONARY ARTERY DISEASE Global Genomics Group, LLC (US) 2022-03-16 EP disclosed
EP-3954991-A2 METHODS AND SYSTEMS FOR DETERMINING AUTISM SPECTRUM DISORDER RISK Laboratory Corporation of America Holdings (US) 2022-02-16 EP disclosed
CN-113156096-A Blood-based biomarkers for diagnosing coronary atherosclerotic disease 全球基因集团有限责任公司 2021-07-23 CN disclosed
CN-107427221-B Blood-based biomarkers for diagnosing coronary atherosclerotic disease 全球基因集团有限责任公司 2021-03-09 CN disclosed
WO-2020260625-A1 QUANTITATIVE RAMAN SPECTROSCOPY AALTO UNIVERSITY FOUNDATION SR (FI) 2020-12-30 WO disclosed
EP-2881394-B1 CONDENSED RING HETEROCYCLIC COMPOUND KYOWA HAKKO KIRIN CO LTD (JP) 2018-03-21 EP disclosed
CN-107427221-A Blood-based biomarkers for diagnosing coronary atherosclerotic disease 全球基因集团有限责任公司 2017-12-01 CN disclosed
WO-2017040450-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE BRISTOL-MYERS SQUIBB COMPANY (US) 2017-03-09 WO disclosed
US-9540366-B2 Ring-fused heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2017-01-10 US disclosed
US-9540366-B2 Ring-fused heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2017-01-10 US disclosed
US-9493439-B1 Proteasome inhibitors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2016-11-15 US disclosed
US-9493439-B1 Proteasome inhibitors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2016-11-15 US disclosed
US-20150284384-A1 RING-FUSED HETEROCYCLIC COMPOUND KYOWA KIRIN CO., LTD. (JP) 2015-10-08 US disclosed
US-20150284384-A1 RING-FUSED HETEROCYCLIC COMPOUND KYOWA KIRIN CO., LTD. (JP) 2015-10-08 US disclosed
EP-2881394-A1 CONDENSED RING HETEROCYCLIC COMPOUND Kyowa Hakko Kirin Co., Ltd. (JP) 2015-06-10 EP disclosed
EP-1642880-B1 HSP90 FAMILY PROTEIN INHIBITORS KYOWA HAKKO KIRIN CO LTD (JP) 2013-09-04 EP disclosed
US-8497380-B2 Substituted acetophenones useful as PDE4 inhibitors LEO PHARMA A/S (DK) 2013-07-30 US disclosed
US-8389442-B2 N-phenyl-′(4-pyridyl)-azinyl!amine derivatives as plant protection agents SYNGENTA CROP PROTECTION LLC (US) 2013-03-05 US disclosed
US-8389442-B2 N-phenyl-′(4-pyridyl)-azinyl!amine derivatives as plant protection agents SYNGENTA CROP PROTECTION LLC (US) 2013-03-05 US disclosed
US-20130012716-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS FELDING JAKOB (DK) 2013-01-10 US disclosed
US-8324394-B2 Substituted acetophenones useful as PDE4 inhibitors LEO PHARMA A/S (DK) 2012-12-04 US disclosed
US-20120165539-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS FELDING JAKOB (DK) 2012-06-28 US disclosed
US-8148537-B2 Substituted acetophenones useful as PDE4 inhibitors LEO PHARMA A/S (DK) 2012-04-03 US disclosed
US-20120070409-A1 TETRACYCLIC FUSED HETEROCYCLIC COMPOUND AND USE THEREOF AS HCV POLYMERASE INHIBITOR JAPAN TOBACCO INC. (JP) 2012-03-22 US disclosed
US-20120020920-A1 5-5-MEMBERED FUSED HETEROCYCLIC COMPOUND AND USE THEREOF AS HCV POLYMERASE INHIBITOR JAPAN TOBACCO INC. (JP) 2012-01-26 US disclosed
EP-1928236-B1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC (BM) 2011-11-23 EP disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7919623-B2 Naphthyridine derivatives having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2011-04-05 US disclosed
US-7919623-B2 Naphthyridine derivatives having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2011-04-05 US disclosed
US-7919517-B2 Indazole derivatives KYOWA HAKKO KIRIN CO., LTD. (JP) 2011-04-05 US disclosed
US-7919517-B2 Indazole derivatives KYOWA HAKKO KIRIN CO., LTD. (JP) 2011-04-05 US disclosed
EP-2125736-B1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA AS (DK) 2011-03-30 EP disclosed
US-7767693-B2 Hsp90 family protein inhibitors KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-08-03 US disclosed
US-7767693-B2 Hsp90 family protein inhibitors KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-08-03 US disclosed
EP-2206715-A1 Fused heterotetracyclic compounds and use thereof as hcv polymerase inhibitor Japan Tobacco, Inc. (JP) 2010-07-14 EP disclosed
US-20100035908-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA (DK) 2010-02-11 US disclosed
US-7659263-B2 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2010-02-09 US disclosed
EP-2125736-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS Leo Pharma A/S (DK) 2009-12-02 EP disclosed
US-20090247522-A1 Hsp90 FAMILY PROTEIN INHIBITORS KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-10-01 US disclosed
US-20090247522-A1 Hsp90 FAMILY PROTEIN INHIBITORS KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-10-01 US disclosed
US-20090227621-A1 Naphthyridine derivatives having inhibitory activity against hiv integrase SHIONOGI & CO., LTD. (JP) 2009-09-10 US disclosed
US-20090227621-A1 Naphthyridine derivatives having inhibitory activity against hiv integrase SHIONOGI & CO., LTD. (JP) 2009-09-10 US disclosed
US-7538224-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
US-7538224-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
US-7538241-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
US-7538241-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
EP-1613156-B1 N-PHENYL- \" (4-PYRIDYL)- AZINYL]AMINE DERIVATIVES AS PLANT PROTECTION AGENTS SYNGENTA PARTICIPATIONS AG (CH) 2009-05-06 EP disclosed
EP-1719773-B1 FUSED HETEROTETRACYCLIC COMPOUNDS AND USE TEHREOF AS HCV POLYMERASE INHIBITOR JAPAN TOBACCO INC (JP) 2009-04-15 EP disclosed
US-7517875-B2 Piperidine derivatives having CCR3 antagonism TEIJIN LIMITED (JP) 2009-04-14 US disclosed
US-7517875-B2 Piperidine derivatives having CCR3 antagonism TEIJIN LIMITED (JP) 2009-04-14 US disclosed
US-20090082348-A1 INDAZOLE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-03-26 US disclosed
US-20090082348-A1 INDAZOLE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-03-26 US disclosed
US-20090042883-A1 ANTITUMOR AGENT KYOWA HAKKOKOGYO CO. (JP) 2009-02-12 US disclosed
US-20090042883-A1 ANTITUMOR AGENT KYOWA HAKKOKOGYO CO. (JP) 2009-02-12 US disclosed
US-7488752-B2 nor-seco himbacine derivatives; thrombosis, anticoagulants, anticancer agents; antiinflammatory agents; anticholesterol agents; cardiovascular disorders; antiarrhythmia agents; antiischemic agents; strokes; antiarthritic agents SCHERING CORPORATION (US) 2009-02-10 US disclosed
US-20090036444-A1 5-5-Membered fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2009-02-05 US disclosed
US-7470717-B2 Indazole derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-12-30 US disclosed
US-7470717-B2 Indazole derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-12-30 US disclosed
WO-2008052072-A9 COMPOUNDS FOR THE TREATMENT OF PAIN AND SCREENING METHODS THEREFOR ACADIA PHARM INC (US) 2008-07-10 WO disclosed
WO-2008077404-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA A/S (DK) 2008-07-03 WO disclosed
WO-2008052072-A2 COMPOUNDS FOR THE TREATMENT OF PAIN AND SCREENING METHODS THEREFOR ACADIA PHARMACEUTICALS INC. (US) 2008-05-02 WO disclosed
EP-1852112-A1 ANTI-TUMOR AGENT KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-11-07 EP disclosed
US-20070155813-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-07-05 US disclosed
US-20070155813-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-07-05 US disclosed
US-20070117856-A1 Indazole derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-05-24 US disclosed
US-20070117856-A1 Indazole derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-05-24 US disclosed
US-20070078146-A1 Antiinflamamtory agents; antiarthritic agents; inflammatory bowel disorders; multiple sclerosis; asthma PHARMACIA CORPORATION 2007-04-05 US disclosed
US-20070049593-A1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2007-03-01 US disclosed
US-20070032532-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-02-08 US disclosed
US-20070032532-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-02-08 US disclosed
US-20070032490-A1 N-Phenyl-'(4-pyridyl)-azinyl!amine derivatives as plant protection agents SYNGENTA CROP PROTECTION, INC. 2007-02-08 US disclosed
US-20070032490-A1 N-Phenyl-'(4-pyridyl)-azinyl!amine derivatives as plant protection agents SYNGENTA CROP PROTECTION, INC. 2007-02-08 US disclosed
EP-1719773-A1 FUSED HETEROTETRACYCLIC COMPOUNDS AND USE TEHREOF AS HCV POLYMERASE INHIBITOR Japan Tobacco, Inc. (JP) 2006-11-08 EP disclosed
EP-1688420-A1 5-5-MEMBERED FUSED HETEROCYCLIC COMPOUND AND USE THEREOF AS HCV POLYMERASE INHIBITOR JAPAN TOBACCO INC. (JP) 2006-08-09 EP disclosed
US-20060167246-A1 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2006-07-27 US disclosed
US-20060167246-A1 Thienopyrrole compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2006-07-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (21 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120165539-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS PDE4A, PDE4B, PDE3B RAB9A 4372/4885NPC1 2936/4885KMT2A 3731/4885
US-20070049593-A1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor POLI, TERT, ZC3HAV1 RAB9A 2410/4885NPC1 1131/4885KMT2A 1865/4885
US-20090036444-A1 5-5-Membered fused heterocyclic compound and use thereof as HCV polymerase inhibitor GTF3C5, ZC3HAV1, POLI RAB9A 1530/4885NPC1 1268/4885KMT2A 2259/4885
US-20120020920-A1 5-5-MEMBERED FUSED HETEROCYCLIC COMPOUND AND USE THEREOF AS HCV POLYMERASE INHIBITOR GTF3C5, ZC3HAV1, POLI RAB9A 1530/4885NPC1 1268/4885KMT2A 2259/4885
US-20100035908-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS PDE4A, PDE4B, PDE3B RAB9A 4359/4885NPC1 2847/4885KMT2A 3607/4885
US-20070032532-A1 Hsp90 family protein inhibitors HSP90AB1, HSP90B1, HSP90AB2P RAB9A 1598/4885NPC1 1079/4885KMT2A 3681/4885
US-20060167246-A1 Thienopyrrole compound and use thereof as HCV polymerase inhibitor TPMT, JAK2, GTF3C5 RAB9A 3278/4885NPC1 2385/4885KMT2A 2063/4885
US-12571737-B2 Quantitative Raman spectroscopy CWC22, ILF2, IL36G RAB9A 4182/4885NPC1 3387/4885KMT2A 4487/4885
US-20090247522-A1 Hsp90 FAMILY PROTEIN INHIBITORS HSP90AB1, HSP90B1, HSP90AB2P RAB9A 1598/4885NPC1 1079/4885KMT2A 3681/4885
US-20070032490-A1 N-Phenyl-'(4-pyridyl)-azinyl!amine derivatives as plant protection agents CYP1A1, NAT1, AKR7A2 RAB9A 579/4885NPC1 347/4885KMT2A 761/4885
US-20070117856-A1 Indazole derivatives IGF1R, NR0B2, ADRA2B RAB9A 2996/4885NPC1 2845/4885KMT2A 1477/4885
US-20120070409-A1 TETRACYCLIC FUSED HETEROCYCLIC COMPOUND AND USE THEREOF AS HCV POLYMERASE INHIBITOR POLI, TERT, ZC3HAV1 RAB9A 2410/4885NPC1 1131/4885KMT2A 1865/4885
US-20070155813-A1 Hsp90 family protein inhibitors HSP90AB1, HEATR1, HSP90AB2P RAB9A 585/4885NPC1 1090/4885KMT2A 3994/4885
US-20070078146-A1 Antiinflamamtory agents; antiarthritic agents; inflammatory bowel disorders; multiple sclerosis; asthma MAPK1, MAPK3, MAPK4 RAB9A 2090/4885NPC1 4880/4885KMT2A 1449/4885
US-20090042883-A1 ANTITUMOR AGENT MCL1, HDAC7, TP53 RAB9A 2761/4885NPC1 1842/4885KMT2A 1021/4885
US-12566161-B2 Methods and consumer products for detecting a metabolite SLC6A6, SLC7A11, CTH RAB9A 1471/4885NPC1 1733/4885KMT2A 3082/4885
US-20090227621-A1 Naphthyridine derivatives having inhibitory activity against hiv integrase PNP, CDKL1, ASNS RAB9A 2264/4885NPC1 1366/4885KMT2A 1071/4885
US-20090082348-A1 INDAZOLE DERIVATIVES IGF1R, NR0B2, ADRA2B RAB9A 2996/4885NPC1 2845/4885KMT2A 1477/4885
US-20130012716-A1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS PDE4A, PDE3B, PDE5A RAB9A 4486/4885NPC1 2749/4885KMT2A 3570/4885
US-20150284384-A1 RING-FUSED HETEROCYCLIC COMPOUND TRPV1, TRPV2, TRPV3 RAB9A 785/4885NPC1 1138/4885KMT2A 2063/4885
US-12578322-B2 Methods and consumer products for detecting a metabolite SHBG, OXGR1, OGG1 RAB9A 4417/4885NPC1 4657/4885KMT2A 1249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.