SCHEMBL4573758

SCHEMBL4573758

Cc1ccc2[nH]c(C(C)N)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.53
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
HTT P42858 2/20 0.50
USP2 O75604 1/20 0.50
KDM4E B2RXH2 2/20 0.45
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SCN10A Q9Y5Y9 6/20 0.43
TAAR1 Q96RJ0 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
MLKL Q8NB16 2/20 0.42
PARP1 P09874 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.38
ALPL P05186 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2757079 0.86 KDM4E (0.59) CYP1A2ALDH1A1HPGDHTTUSP2
SCHEMBL5111363 0.82 TAAR1 (0.47) CYP1A2ALDH1A1HPGDHTTUSP2
SCHEMBL4154842 0.81 CSNK2A1 (0.45) CYP1A2ALDH1A1HTTKDM4ELMNA
SCHEMBL5101171 0.81 CSNK2A1 (0.45) CYP1A2ALDH1A1HTTKDM4ELMNA
SCHEMBL580393 0.81 LMNA (0.42) CYP1A2ALDH1A1HPGDHTTKDM4E
SCHEMBL6471271 0.81 ALPL (0.49) CYP1A2ALDH1A1KDM4ELMNAHSD17B10
SCHEMBL8071559 0.81 ALPL (0.49) CYP1A2ALDH1A1KDM4ELMNAHSD17B10
SCHEMBL1479636 0.81 LMNA (0.42) CYP1A2ALDH1A1HPGDHTTKDM4E
SCHEMBL5110077 0.81 KDM4E (0.42) CYP1A2ALDH1A1HPGDHTTUSP2
SCHEMBL8071556 0.81 ALPL (0.49) CYP1A2ALDH1A1KDM4ELMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080207683-A1 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. 2008-08-28 US claimed
WO-2008100622-A2 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. (US) 2008-08-21 WO claimed
US-20260138071-A1 SULFIDE GAS REMOVAL PROCESS KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2026-05-21 US disclosed
US-20260014197-A1 DRUG DELIVERY SYSTEM IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2026-01-15 US disclosed
US-20260014517-A1 HYDROGEN SULFIDE REMOVAL METHOD FROM DRILLING MUD COMPOSITION KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2026-01-15 US disclosed
US-20260014514-A1 METHOD FOR SCAVENGING HYDROGEN SULFIDE FROM A GASEOUS COMPOSITION IN A STIRRED TANK REACTOR KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2026-01-15 US disclosed
US-20260008009-A1 PROCESS FOR REMOVING HYDROGEN SULFIDE FROM A HYDROCARBON GASEOUS COMPOSITION KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2026-01-08 US disclosed
US-20260002088-A1 PROCESS TO REMOVE HYDROGEN SULFIDE FROM A HYDROCARBON-CONTAINING GAS COMPOSITION KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2026-01-01 US disclosed
US-20250381514-A1 METHOD FOR REMOVING HYDROGEN SULFIDE FROM SOUR GAS KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2025-12-18 US disclosed
US-12459862-B2 Cement paste composition KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2025-11-04 US disclosed
US-12427499-B2 Process for removing hydrogen sulfide from sour gases KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2025-09-30 US disclosed
US-20230404932-A1 METHOD FOR TREATING BLASTOCYSTIS INFECTION IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2023-12-21 US disclosed
US-20230404931-A1 METHOD FOR FORMING A NANOMEDICINAL COMPOSITION IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2023-12-21 US disclosed
US-20230404930-A1 METAL ORGANIC FRAMEWORK/POROUS SILICATE AND/OR ALUMINOSILICATE NANOCARRIER FOR BLASTOCYSTOSIS TREATMENT IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2023-12-21 US disclosed
US-11826477-B1 Metal organic framework/porous silicate and/or aluminosilicate nanocarrier for blastocystosis treatment IMAM ABDULRAHMAN BIN FAISAL UNIVERSITY (SA) 2023-11-28 US disclosed
US-11746278-B1 Method of removing sulfide-containing scale KING FAHD UNIVERSITY OF PETROLEUM AND (SA) 2023-09-05 US disclosed
US-11708517-B1 Hydrogen sulfide mitigating drilling fluid and method of drilling subterranean geological formation KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2023-07-25 US disclosed
US-20200269194-A1 POROUS MEMBRANE CONTAINING METAL-ORGANIC FRAMEWORKS KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2020-08-27 US disclosed
US-20080207683-A1 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. 2008-08-28 US disclosed
WO-2008100622-A2 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S SUNESIS PHARMACEUTICALS, INC. (US) 2008-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260008009-A1 PROCESS FOR REMOVING HYDROGEN SULFIDE FROM A HYDROCARBON GASEOUS COMPOSITION HMOX2, HMOX1, SCO2 CYP1A2 1297/4885ALDH1A1 3365/4885HPGD 2831/4885
US-20260014517-A1 HYDROGEN SULFIDE REMOVAL METHOD FROM DRILLING MUD COMPOSITION TST, SOD1, SAMM50 CYP1A2 3591/4885ALDH1A1 3428/4885HPGD 2825/4885
US-11826477-B1 Metal organic framework/porous silicate and/or aluminosilicate nanocarrier for blastocystosis treatment CAT, GPX1, SLC39A11 CYP1A2 1780/4885ALDH1A1 1463/4885HPGD 4114/4885
US-20230404930-A1 METAL ORGANIC FRAMEWORK/POROUS SILICATE AND/OR ALUMINOSILICATE NANOCARRIER FOR BLASTOCYSTOSIS TREATMENT CAT, GPX1, SLC39A11 CYP1A2 1780/4885ALDH1A1 1463/4885HPGD 4114/4885
US-20230404932-A1 METHOD FOR TREATING BLASTOCYSTIS INFECTION CAT, GPX1, GPX4 CYP1A2 969/4885ALDH1A1 1263/4885HPGD 3657/4885
US-20260002088-A1 PROCESS TO REMOVE HYDROGEN SULFIDE FROM A HYDROCARBON-CONTAINING GAS COMPOSITION SAMM50, SOD1, HNRNPH3 CYP1A2 1844/4885ALDH1A1 3149/4885HPGD 2333/4885
US-20260138071-A1 SULFIDE GAS REMOVAL PROCESS SAMM50, SRSF1, GTF2F1 CYP1A2 3087/4885ALDH1A1 4587/4885HPGD 2762/4885
US-20260014514-A1 METHOD FOR SCAVENGING HYDROGEN SULFIDE FROM A GASEOUS COMPOSITION IN A STIRRED TANK REACTOR SOD1, MAFG, HMOX2 CYP1A2 3587/4885ALDH1A1 4774/4885HPGD 1662/4885
US-20230404931-A1 METHOD FOR FORMING A NANOMEDICINAL COMPOSITION GPX1, GPX4, CAT CYP1A2 1324/4885ALDH1A1 1362/4885HPGD 2867/4885
US-20260014197-A1 DRUG DELIVERY SYSTEM IPO8, SLC39A11, SLC2A8 CYP1A2 2705/4885ALDH1A1 3703/4885HPGD 4499/4885
US-20080207683-A1 BIARYL-SUBSTITUTED TETRAHYDRO-PYRAZOLO-PYRIDINE MODULATORS OF CATHEPSIN S CTSS, CTSK, CTSZ CYP1A2 2244/4885ALDH1A1 4560/4885HPGD 2447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.